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Vasopressin Receptor

Vasopressin Receptor

Cat. No. Product Name CAS No. Information
CSN16162 Xipamide   14293-44-8 Xipamide a sulfonamide diuretic drug can block sodium reabsorption in distal tubules of the kidney and the cystic fibrosis transmembrane conductance regulator CFTR chloride channel It is used for the treatment of oedema and hypertension
CSN20586 SR49059 150375-75-0 SR49059 is a potent and selective non-peptide vasopressin V1A receptor antagonist which is devoid of agonist activity SR49059 displays high affinity and efficacy at both rat Ki 16 nM and human Ki 11 - 63 nM V1A receptors and potently antagonizes arginine vasopressin-induced effects in vitro IC50 37 nM for inhibition of human platelet aggregation and is orally active in vivo
CSN20548 Selepressin 876296-47-8 Selepressin is a potent, selective vasopressin V1a receptor agonist potentially for the treatment of septic shock.
CSN21427 RO5028442 920022-47-5 RO5028442 is a potent and selective brain-penetrant vasopressin 1a V1a receptor antagonist with Kis of 1 nM hV1a and 39 nM mV1a
CSN12760 Mozavaptan 137975-06-5 Mozavaptan is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 12 M and 14 nM respectively
CSN13437 Conivaptan HCl   168626-94-6 Conivaptan hydrochloride is an inhibitor of antidiuretic hormone or antagonist of vasopressin receptor It can inhibit rat liver V1A receptor and kidney V2 receptor with Ki of 048 nM and 304 nM respectively
CSN10352 Atosiban   90779-69-4 Atosiban is competitive antagonist of vasopressin and oxytocin receptors It is a nonapeptide and the analogue of desamino-oxytocin
CSN22355 Balovaptan 1228088-30-9
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