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Vasopressin Receptor

Vasopressin Receptor

Cat. No. Product Name CAS No. Information
CSN16162 Xipamide   14293-44-8 Xipamide a sulfonamide diuretic drug can block sodium reabsorption in distal tubules of the kidney and the cystic fibrosis transmembrane conductance regulator CFTR chloride channel It is used for the treatment of oedema and hypertension
CSN20586 SR49059 150375-75-0 SR49059 is a potent and selective non-peptide vasopressin V1A receptor antagonist which is devoid of agonist activity SR49059 displays high affinity and efficacy at both rat Ki 16 nM and human Ki 11 - 63 nM V1A receptors and potently antagonizes arginine vasopressin-induced effects in vitro IC50 37 nM for inhibition of human platelet aggregation and is orally active in vivo
CSN20548 Selepressin 876296-47-8 Selepressin is a potent, selective vasopressin V1a receptor agonist potentially for the treatment of septic shock.
CSN12760 Mozavaptan 137975-06-5 Mozavaptan is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 12 M and 14 nM respectively
CSN21908 Lixivaptan 168079-32-1 Lixivaptan is an orally active and selective vasopressin receptor V2 antagonist with IC50 values of 1.2 and 2.3 nM for human and rat V2, respectively.
CSN13437 Conivaptan HCl   168626-94-6 Conivaptan HCl is an inhibitor of antidiuretic hormone or antagonist of vasopressin receptor. It can inhibit rat liver V1A receptor and kidney V2 receptor with Ki of 0.48 nM and 3.04 nM, respectively.
CSN22355 Balovaptan 1228088-30-9 Balovaptan is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) receptors, and is used for the research of autism.
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