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SRPK
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN24738 | ZT-12-037-01 | 2328073-61-4 | ZT-12-037-01 is a potent and selective STK19 inhibitor with an IC50 value of 24.04nM |
| CSN19078 | WNK463 | 2012607-27-9 | WNK463 is a potant With-No-Lysine WNK kinase inhibitor with IC50s of 5169 nM for WNK1234 |
| CSN22078 | TMPA | 1258275-73-8 | TMPA is an antagonist of nuclear receptor Nur77 and LKB1 interaction. |
| CSN23884 | STK16-IN-1 | 1223001-53-3 | STK16-IN-1 is a serine/threonine protein kinase 16 (STK16) inhibitor with IC50 of 295 nM. |
| CSN13762 | SRPIN340 | 218156-96-8 | SRPIN340 is an inhibitor of serinearginine-rich protein kinase SRPK1 with IC50 of 089 M |
| CSN23673 | SPHINX31 | 1818389-84-2 | SPHINX31 is a potent and selective inhibitor of serine/arginine-rich protein kinase 1 (SRPK1), with an IC50 of 5.9 nM. SPHINX31 inhibits phosphorylation of serine/arginine-rich splicing factor 1 (SRSF1). SPHINX31 is a potential topical therapeutic for neovascular eye disease[1]. |
| CSN20434 | PROTAC TBK1 C3i | 2052306-13-3 | PROTAC TBK1 C3i is a potent hit TBK1 DC50 12 nM Dmax 96 with excellent selectivity against a related kinase IKK which was further used as a chemical tool to assess TBK1 as a target in mutant K-Ras cancer cells |
| CSN17458 | Pim1/AKK1-IN-1 | 1093222-27-5 | Pim1 AKK1-IN-1 is a potent multi-kinase inhibitor with Kd values of 35 nM53 nM75 nM380 nM for Pim1AKK1MST2LKB1 respectively and also inhibits MPSK1 and TNIK |
| CSN23000 | Nek2-IN-5 | 1507367-00-1 | NCL 00017509 is a potent and reversible NIMA related kinase 2 (Nek2) inhibitor with IC50 of 56 nM. |
| CSN17802 | ML281 | 1404437-62-2 | ML281 is a potent and selective serinethreonine kinase STK33 inhibitor with IC50 of 14 nM STK33 downregulation is toxic to KRAS-dependent cancer cell lines |
| CSN27205 | ILK-IN-3 | 6975-75-3 | ILK-IN-3 is an integrin linked kinase inhibitor. |
| CSN18951 | OSU-T315 | 2070015-22-2 | ILK-IN-2 is a ILK inhibitor |
| CSN17699 | ILK-IN-2 | 1333146-24-9 | ILK-IN-1 is an ILK inhibitor with IC50 of 06 M |
| CSN24084 | GSK8612 | 2361659-62-1 | GSK8612 is a potent and highly selective Tank-binding Kinase-1 (TBK1) inhibitor with pIC50 of 6.8 for recombinant TBK1. |
| CSN25836 | CMPD101 | 865608-11-3 | CMPD101 is a selective GRK2/3 inhibitor with IC50 values of 32 and 54 nM for GRK3 and GRK2, respectively. |
| CSN20021 | Bryostatin 1 | 83314-01-6 | Bryostatin 1 is a Protein kinase C (PKC) activator that binds with high affinity (Ki = 1.35 nM). |
| CSN42722 | Belumosudil mesylate | 2109704-99-4 | Belumosudil is a small molecule and selective inhibitor of ROCK2 with IC50 of 105 nM, which is over 200 fold selecivity over ROCK1 (IC50 =24 μM). |
| CSN12528 | 4μ8C | 14003-96-4 | 48C is a potent and selective IRE1 Rnase inhibitor with IC50 of 76 nM. |
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