Welcome to CSNpharm! For Research Use Only!
Home +1-708-781-1677 sales@csnpharm.com    

Sigma Receptor

Sigma Receptor

Cat. No. Product Name CAS No. Information
CSN16114 Siramesine 147817-50-3 Siramesine is a selective sigma-2 receptor agonist which has been shown to trigger cell death of cancer cells and to exhibit a potent anticancer activity in vivo
CSN16281 Siramesine HCl 224177-60-0 Siramesine hydrochloride is an agonist of sigma-2 receptor which can trigger cell death and exhibit anticancer activity
CSN11878 SA4503 2HCl   165377-44-6 SA4503 is the dihydrochloride form of SA4503 which is an agonist of opioid sigma1 receptor (1R) with IC50 of 17.4 nM.
CSN17988 SA4503   165377-43-5 SA4503 is an agonist of opioid sigma1 receptor (1R) with IC50 of 17.4 nM.
CSN16936 S1RA 878141-96-9 S1RA is a potent and selective sigma-1 receptor 1R Ki17 nM antagonist showed good selectivity against 2R Ki 1000 nM
CSN17645 S1RA HCl 1265917-14-3 S1RA hydrochloride is a potent and selective sigma-1 receptor 1R Ki17 nM antagonist showed good selectivity against 2R Ki 1000 nM
CSN11834 Remoxipride 80125-14-0 Remoxipride is an atypical antipsychotic which was previously used in Europe for the treatment of schizophrenia and acute mania but was withdrawn due to toxicity concerns incidence of aplastic anemia in 110000 patients
CSN21927 Pridopidine 346688-38-8 Pridopidine exhibits high affinity towards sigma 1 receptor S1R Ki 70-80 nM which can counteract the effects of excessive or insufficient dopaminergic transmission and it can used as a dopamine DA stabilizer
CSN18418 PRE-084 HCl 75136-54-8 PRE-084 hydrochloride is a high affinity selective 1 agonist has an IC50 of 44 nM in the sigma receptor assay
CSN16267 BD-1047 Dihydrobromide   138356-21-5 BD-1047 dihydrobromide is a selective functional antagonist of sigma receptors shows antipsychotic activity in animal models predictive of efficacy in schizophrenia
CSN17929 4-IBP   155798-08-6 4-IBP is selective 1 agonist with Ki of 17 nM and 252 nM for 2 receptor
CSN21074 Anavex 2-73 HCl 195615-84-0 1 agonist IC50 860 nM also displays affinity for muscarinic M1-M4 receptors Ki values 500 nM but not for 2 receptors Exhibits neuroprotective effects prevents tau hyperphosphorylation and attenuates scopolamine- and -MK 801-induced learning deficits in a mouse model of amyloid toxicity
CSN23812 Dimemorfan Phosphate 36304-84-4
<< PREV 1 NEXT >>