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Sigma Receptor

Sigma Receptor

Cat. No. Product Name CAS No. Information
CSN16114 Siramesine 147817-50-3 Siramesine is a selective sigma-2 receptor agonist which has been shown to trigger cell death of cancer cells and to exhibit a potent anticancer activity in vivo
CSN16281 Siramesine HCl 224177-60-0 Siramesine HCl is an agonist of sigma-2 receptor which can trigger cell death and exhibit anticancer activity.
CSN17988 SA4503   165377-43-5 SA4503 is an agonist of opioid sigma1 receptor (1R) with IC50 of 17.4 nM.
CSN11878 SA4503 2HCl   165377-44-6 SA4503 2HCl is the 2HCl form of SA4503 which is an agonist of opioid sigma1 receptor (σ1R) with IC50 of 17.4 nM.
CSN16936 S1RA 878141-96-9 S1RA is a potent and selective sigma-1 receptor 1R Ki17 nM antagonist showed good selectivity against 2R Ki 1000 nM
CSN17645 S1RA HCl 1265917-14-3 S1RA HCl is a potent and selective sigma-1 receptor (σ1R, Ki=17 nM) antagonist, showed good selectivity against σ2R (Ki > 1000 nM).
CSN33114 Roluperidone 359625-79-9 Roluperidone is a 5-HT2A and sigma 2 receptor antagonist.
CSN21927 Pridopidine 346688-38-8 Pridopidine exhibits high affinity towards sigma 1 receptor S1R Ki 70-80 nM which can counteract the effects of excessive or insufficient dopaminergic transmission and it can used as a dopamine DA stabilizer
CSN18418 PRE-084 HCl 75136-54-8 PRE-084 HCl is a high affinity, selective σ1 agonist, has an IC50 of 44 nM in the sigma receptor assay.
CSN26761 PD-144418 Oxalate 1794760-28-3 PD-144418 Oxalate is a novel selective sigma ligand.
CSN26378 1,3-Di-o-tolylguanidine 97-39-2 Ditolylguanidine (1,3-Di-o-tolylguanidine) is an agonist of sigma receptor (σ1/σ2 receptor)[1].
CSN33115 CYR-101 HCl 2H2O 1937215-88-7 CYR-101 hydrochloride dihydrate is a 5-HT2A and sigma 2 receptor antagonist.
CSN24789 BD1063 dhydrochloride 206996-13-6 BD1063 dhydrochloride is a potent and selective sigma 1 receptor antagonist.
CSN16267 BD-1047 Dihydrobromide   138356-21-5 BD-1047 dihydrobromide is a selective functional antagonist of sigma receptors shows antipsychotic activity in animal models predictive of efficacy in schizophrenia
CSN17929 4-IBP   155798-08-6 4-IBP is selective 1 agonist with Ki of 17 nM and 252 nM for 2 receptor
CSN21074 Anavex 2-73 HCl 195615-84-0 1 agonist IC50 860 nM also displays affinity for muscarinic M1-M4 receptors Ki values 500 nM but not for 2 receptors Exhibits neuroprotective effects prevents tau hyperphosphorylation and attenuates scopolamine- and -MK 801-induced learning deficits in a mouse model of amyloid toxicity
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