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ROCK

ROCK

Cat. No. Product Name CAS No. Information
CSN13431 Y-33075 2HCl 173897-44-4 Y-39983 HCl is a selective rho-associated protein kinase(ROCK) inhibitor with an IC50 of 3.6 nM.
CSN18082 Y-33075 199433-58-4 Y-33075 is potent and selective p160 ROCK inhibitor with an Ki value of 014 M 200 fold selectivity for p160ROCK than PKC cAMP-dependent protein kianse and Mypsin light-chain kinase
CSN12226 Y-27632 146986-50-7 Y-27632 is an ATP-competitive inhibitor of ROCK-I and ROCK-II with Ki of 220 nM and 300 nM for ROCK-I and ROCK-II respectively
CSN13895 Y-27632 2HCl   129830-38-2 Y-27632 2HCl is a selective ROCK1 (p160ROCK) inhibitor with Ki of 140 nM, exhibits > 200-fold selectivity over other kinases, including PKC, cAMP-dependent protein kinase, MLCK and PAK.
CSN16953 K-115 223645-67-8 K-115, an isoquinolinesulfonamide compound, is a highly selective and potent (IC50 31 nM) Rho-kinase inhibitor, and used for treating POAG or ocular hypertension.
CSN17105 Hydroxyfasudil 105628-72-6 Hydroxyfasudil metabolite of Fasudil is a potent Rho-kinase inhibitor and vasodilator
CSN15927 Hydroxyfasudil HCl 155558-32-0 Hydroxyfasudil HCl, metabolite of fasudil, is a potent Rho-kinase inhibitor and vasodilator.
CSN16493 H-1152 451462-58-1 H-1152 an isoquinolinesulfonamide derivative is a more specific stronger and membrane-permeable inhibitor of Rho-kinase with a Ki value of 16 nM but poor inhibitor of other serinethreonine kinases
CSN19208 GSK269962 HCl 2095432-71-4 GSK269962 HCl is a selective ROCK (Rho-associated protein kinase) inhibitor with IC50 values of 1.6 and 4 nM for ROCK1 and ROCK2, respectively.
CSN10984 Fasudil HCl   105628-07-7 Fasudil HCl is a potent inhibitor of ROCK-II, PKA, PKG, PKC, and MLCK with Ki of 0.33 μM, 1.6 μM, 1.6 μM, 3.3 μM and 36 μM, respectively.
CSN10983 Fasudil 103745-39-7 Fasudil HCl is a potent inhibitor of ROCK-II, PKA, PKG, PKC, and MLCK with Ki of 0.33 μM, 1.6 μM, 1.6 μM, 3.3 μM and 36 μM, respectively.
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