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| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN23132 | SR8278 | 1254944-66-5 | SR8278 is a rev-erbα antagonist. It inhibits Rev-Erbα transcriptional repression (EC50 = 0.47 μM) and blocks activity of Rev-Erbα agonist GSK 4112 in HEK293 cells. SR8278 increases expression of glucose-regulating genes, G6Pase and PEPCK in HepG2 cells. |
| CSN26216 | SR10067 | 1380548-02-6 | SR10067 is a potent, selective and brain penetrant Rev-Erbα/β agonist, with IC50 values are 160 and 170 nM for Rev-Erbβ and Rev-Erbα, respectively. |
| CSN17576 | GSK4112 | 1216744-19-2 | GSK4112 is an agonist of Rev-erb with EC50 of 04 M and it can be designed to mimic the action of heme |
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