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PKC
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN18071 | TAS-301 | 193620-69-8 | TAS-301 is an inhibitor of smooth muscle cell migration and proliferation, inhibits intimal thickening after balloon injury to rat carotid arteries. |
| CSN11854 | Ro 31-8220 Mesylate | 138489-18-6 | Ro 31-8220 mesylate is a pan-PKC inhibitor with IC50 of 5 nM, 24 nM, 14 nM, 27 nM, and 24 nM for PKC-, PKC-I, PKC-II, PKC-, and PKC-, respectively. |
| CSN11701 | Phorbol 12-Myristate 13-Acetate | 16561-29-8 | Phorbol 12-myristate 13-acetate is a PKC-activating phorbol ester, increases the intracellular Ca2 concentration (Ca2i) in a dose-dependent manner, with an EC50 of 11.7 nM. |
| CSN11485 | Myricitrin | 17912-87-7 | Myricitrin a flavonoid compound isolated from the root bark of Myrica cerifera which exerts antinociceptive effects |
| CSN12991 | LY333531 HCl | 169939-93-9 | LY333531 is a -specific protein kinase C inhibitor. It competitively and reversibly inhibits PKC1 and PKC2 with IC50 values of 4.7 and 5.9 nM respectively. |
| CSN11206 | Ingenol | 30220-46-3 | Ingenol is a diterpenoid with unique architecture and has derivatives possessing important anticancer activity. |
| CSN16527 | Go6983 | 133053-19-7 | Go6983 is a pan-PKC inhibitor against for PKC PKC PKC and PKC with IC50 of 7 nM 7 nM 6 nM and 10 nM respectively and less potent to PKC and inactive to PKC |
| CSN10464 | Bisindolylmaleimide I | 133052-90-1 | GF109203X is a potent PKC inhibitor with IC50 of 20 nM, 17 nM, 16 nM, and 20 nM for PKC, PKCI, PKCII, and PKC in cell-free assays, respectively, showing more than 3000-fold selectivity for PKC as compared to EGFR, PDGFR and insulin receptor. |
| CSN12444 | Enzastaurin | 170364-57-5 | Enzastaurin is a potent PKC selective inhibitor with IC50 of 6 nM 6- to 20-fold selectivity against PKC PKC and PKC |
| CSN26161 | D-Sphingosine | 123-78-4 | D-Sphingosine inhibits protein kinase C. |
| CSN10607 | Chelerythrine Chloride | 3895-92-9 | Chelerythrine Chloride is a potent, cell-permeable inhibitor of protein kinase C (IC50 = 660 nM) and competitive with respect to the phosphate acceptor and non-competitive with respect to ATP. |
| CSN17986 | CGP-60474 | 164658-13-3 | CGP60474 is a promising inhibitor of PKC with a high degree of selectivity versus other serinethreonine and tyrosine kinases and show competitive kinetics relative to ATP |
| CSN25331 | Bisindolylmaleimide IV | 119139-23-0 | Bisindolylmaleimide IV is an inhibitor of protein kinase C. |
| CSN11220 | Acteoside | 61276-17-3 | Acteoside, is a natural product isolated and purified from the herbs of Cistanche deserticola Y.C. Ma with known antioxidant activity. It is a protein kinase C inhibitor (IC50 25 M). |
| CSN12210 | α-Tocopherol | 59-02-9 | -Tocopherol is a type of vitamin E and an antagonist of PKC. |
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