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PKC

PKC

Cat. No. Product Name CAS No. Information
CSN18071 TAS-301 193620-69-8 TAS-301 is an inhibitor of smooth muscle cell migration and proliferation, inhibits intimal thickening after balloon injury to rat carotid arteries.
CSN11854 Ro 31-8220 Mesylate   138489-18-6 Ro 31-8220 mesylate is a pan-PKC inhibitor with IC50 of 5 nM, 24 nM, 14 nM, 27 nM, and 24 nM for PKC-, PKC-I, PKC-II, PKC-, and PKC-, respectively.
CSN11701 Phorbol 12-Myristate 13-Acetate 16561-29-8 Phorbol 12-myristate 13-acetate is a PKC-activating phorbol ester, increases the intracellular Ca2 concentration (Ca2i) in a dose-dependent manner, with an EC50 of 11.7 nM.
CSN11485 Myricitrin   17912-87-7 Myricitrin a flavonoid compound isolated from the root bark of Myrica cerifera which exerts antinociceptive effects
CSN12991 LY333531 HCl 169939-93-9 LY333531 is a -specific protein kinase C inhibitor. It competitively and reversibly inhibits PKC1 and PKC2 with IC50 values of 4.7 and 5.9 nM respectively.
CSN11206 Ingenol   30220-46-3 Ingenol is a diterpenoid with unique architecture and has derivatives possessing important anticancer activity.
CSN16527 Go6983   133053-19-7 Go6983 is a pan-PKC inhibitor against for PKC PKC PKC and PKC with IC50 of 7 nM 7 nM 6 nM and 10 nM respectively and less potent to PKC and inactive to PKC
CSN10464 Bisindolylmaleimide I 133052-90-1 GF109203X is a potent PKC inhibitor with IC50 of 20 nM, 17 nM, 16 nM, and 20 nM for PKC, PKCI, PKCII, and PKC in cell-free assays, respectively, showing more than 3000-fold selectivity for PKC as compared to EGFR, PDGFR and insulin receptor.
CSN12444 Enzastaurin   170364-57-5 Enzastaurin is a potent PKC selective inhibitor with IC50 of 6 nM 6- to 20-fold selectivity against PKC PKC and PKC
CSN26161 D-Sphingosine 123-78-4 D-Sphingosine inhibits protein kinase C.
CSN10607 Chelerythrine Chloride   3895-92-9 Chelerythrine Chloride is a potent, cell-permeable inhibitor of protein kinase C (IC50 = 660 nM) and competitive with respect to the phosphate acceptor and non-competitive with respect to ATP.
CSN17986 CGP-60474 164658-13-3 CGP60474 is a promising inhibitor of PKC with a high degree of selectivity versus other serinethreonine and tyrosine kinases and show competitive kinetics relative to ATP
CSN25331 Bisindolylmaleimide IV 119139-23-0 Bisindolylmaleimide IV is an inhibitor of protein kinase C.
CSN11220 Acteoside 61276-17-3 Acteoside, is a natural product isolated and purified from the herbs of Cistanche deserticola Y.C. Ma with known antioxidant activity. It is a protein kinase C inhibitor (IC50 25 M).
CSN12210 α-Tocopherol   59-02-9 -Tocopherol is a type of vitamin E and an antagonist of PKC.
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