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P2X Receptor

P2X Receptor

Cat. No. Product Name CAS No. Information
CSN21970 PSB-12062 55476-47-6 PSB-12062 is a potent and selective P2X4 antagonist with IC50 of 1.38 μM for human P2X4.
CSN21352 BzATP Triethylammonium Salt 112898-15-4 Prototypic P2X7 receptor agonist that exhibits 5 - 10 fold greater potency than ATP EC50 07 M in HEK 293 cells EC50 values are 36 and 285 M for rat and mouse receptors respectively Exhibits partial agonist activity at P2X1 pEC50 87 and P2Y1 receptors and can be used as a photoaffinity label for ATPase
CSN21404 BzATP 81790-82-1 Prototypic P2X7 receptor agonist that exhibits 5 - 10 fold greater potency than ATP EC50 07 M in HEK 293 cells EC50 values are 36 and 285 M for rat and mouse receptors respectively Exhibits partial agonist activity at P2X1 pEC50 87 and P2Y1 receptors and can be used as a photoaffinity label for ATPase
CSN16004 NF449 627034-85-9 NF449 is a potent purinergic receptor antagonist that displays high selectivity for P2X1 IC50 values are 028 069 120 1820 47000 and 300000 nM for rP2X1 rP2X15 rP2X23 rP2X3 rP2X2 and P2X4 receptors respectively Provides antithrombotic protection in vivo Also acts as a Gs-selective antagonist
CSN20323 NF023 104869-31-0 NF023 a subtype-selective competitive and reversible P2X1 receptor antagonist displays IC50 values of 021 289 50 and 100 M for human P2X1 P2X3 P2X2 and P2X4-mediated responses respectively
CSN19839 JNJ 47965567 1428327-31-4 JNJ 47965567 is a potent and selective P2X7 antagonist pIC50 values are 83 75 and 72 for human mouse and rat receptors respectively
CSN18197 GW791343 3HCl 309712-55-8 GW791343 3HCl is a P2X7 allosteric modulator and exhibits species-specific activity and acts as a negative allosteric modulator of human P2X7 (pIC50 = 6.9 - 7.2).
CSN10731 CTP Disodium Dihydrate   81012-87-5 CTP Disodium Dihydrate is a P2X4 purinergic receptor agonist
CSN25312 BX430 688309-70-8 BX430 is selective P2X4 allosteric antagonist with IC50 of 0.54 μM.
CSN27579 AZ10606120 2HCl 607378-18-7 AZ10606120 dihydrochloride is a selective, high affinity antagonist for P2X7 receptor (P2X7R) at human and rat with an IC50 of ~10 nM. AZ10606120 dihydrochloride is little or no effect at other P2XR subtypes. AZ10606120 dihydrochloride has anti-depressant effects and reduces tumour growth .
CSN19020 A-804598   1125758-85-1 A-804598 is a competitive and selective P2X7 receptor antagonist with IC50 of 10 nM 9 nM and 11 nM in rat mouse and human P2X7 receptors respectively
CSN13107 A-740003 861393-28-4 A-740003 is potent selective and competitive P2X7 receptor antagonist IC50 values are 18 and 40 nM for rat and human receptors respectively
CSN18546 A 438079 HCl   899431-18-6 A 438079 hydrochloride is a competitive P2X7 receptor antagonist pIC50 69 for the inhibition of Ca2 influx in the human recombinant P2X7 cell line
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