Welcome to CSNpharm! For Research Use Only!
Home +1-708-781-1677 sales@csnpharm.com    

P-gp

P-gp

Cat. No. Product Name CAS No. Information
CSN12903 Zosuquidar 167354-41-8 Zosuquidar is P-gp modulator that inhibited Pgp-ATPase activity 50-60 at 2 and 10M and had no effect at 008 and 04M measured by P-gp ATPase activity
CSN12751 Zosuquidar 3HCl 167465-36-3 Zosuquidar 3HCl is the 3HCl form of Zosuquidar. Zosuquidar is P-gp modulator that inhibited Pgp-ATPase activity 50-60% at 2 and 10μM and had no effect at 0.08 and 0.4μM.
CSN12182 Valspodar 121584-18-7 Valspodar is a P-glycoprotein P-gp inhibitor widely used in preclinical and clinical studies for overcoming multidrug resistance MDR
CSN14774 Taxinine B 18457-44-8 Taxinine B, a natural product isolated and purified from the barks of Taxus chinensis, can inhibit the drug transport by P-glycoprotein in multidrug-resistant cells, and shows stronger inhibitory effects than acetylsalicylic acid (ASA) on platelet aggregation induced by arachidonic acid (AA).
CSN18364 Tariquidar Methanesulfonate Hydrate 625375-83-9 Tariquidar methanesulfonate is a potent and specific inhibitor of P-glycoprotein P-gp with the high affinity Kd5109 nM
CSN12910 Tariquidar 206873-63-4 Tariquidar is a potent and selective noncompetitive inhibitor of P-glycoprotein with Kd of 51 nM reverses drug resistance in MDR cell Lines
CSN13177 Sinapine Thiocyanate 7431-77-8 Sinapine, an alkaloid isolated and purified from the seeds of Raphanus sativus L., possess antioxidant and radio-protective activities, downregulats multi-drug resistance 1 (MDR1) expression.
CSN22057 Sinapine 18696-26-9 Sinapine is an alkaloid from seeds of the cruciferous species which shows antioxidant and radio-protective activities and decreases expression of P-glycoprotein in Caco-2 cells.
CSN19434 Schizandrin   7432-28-2 Schizandrin is a natural product possessing antioxidant and anti-inflammatory activities.
CSN13555 Isosinensetin   17290-70-9 Isosinensetin exhibits HIV-1 protease inhibiting and antioxidant activities. It is a natural product isolated and purified from the fruit of Citrus aurantium L..
CSN15743 HM30181 849675-66-7 HM30181 is a potent and selective inhibitor of P-glycoprotein
CSN20429 Heliosterpenoid B N/A Heliosterpenoid B is a natural product isolated and purfied from the whole plants of Euphorbia helioscopia being potent inhibitors of P-glycoprotein ABCB1
CSN20428 Heliosterpenoid A 2109805-68-5 Heliosterpenoid A is a natural product isolated and purfied from the whole plants of Euphorbia helioscopia being potent inhibitors of P-glycoprotein ABCB1 and exhibiting cytotoxicity against MDA-MB-231 cell lines
CSN14838 Epimedokoreanin B 161068-53-7 Epimedokoreanin B is a natural product isolated and purified from the herbs of Epimedium brevicornum
CSN10894 Elacridar 143664-11-3 Elacridar is a P-glycoprotein inhibitor, and has been used both in vitro and in vivo as a tool inhibitor of P-glycoprotein (Pgp) to investigate the role of transporters in the disposition of various test molecules.
CSN13175 Elacridar HCl 143851-98-3 Elacridar HCl is a P-glycoprotein (P-gp) inhibitor, and has been used both in vitro and in vivo as a tool inhibitor of P-gp to investigate the role of transporters in the disposition of various test molecules.
CSN17662 Dofequidar 129716-58-1 Dofequidar is a quinoline compound which can reverse P-glycoprotein P-gp-mediated MDR
CSN17917 Dofequidar Fumarate 153653-30-6 Dofequidar fumarate an orally active quinoline compound has been reported to overcome MDR by inhibiting ABCB1P-gp ABCC1MDR-associated protein 1 or both
CSN22768 CP 100356 HCl 142715-48-8 CP 100356 HCl is a high affinity P-glycoprotein (P-gp) inhibitor with Kis of 58 and 94 nM for mouse Pgp1a and Pgp1b isoforms.
CSN23176 UCLA GP130 2 339303-87-6
<< PREV 1 NEXT >>