P-glycoprotein | Membrane Transporter/Ion Channel|Neuronal Signaling| CSNpharm

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Cat. No.	Product Name	CAS No.	Information
CSN12903	Zosuquidar	167354-41-8	Zosuquidar is P-gp modulator that inhibited Pgp-ATPase activity 50-60 at 2 and 10M and had no effect at 008 and 04M measured by P-gp ATPase activity
CSN12751	Zosuquidar 3HCl	167465-36-3	Zosuquidar 3HCl is the 3HCl form of Zosuquidar. Zosuquidar is P-gp modulator that inhibited Pgp-ATPase activity 50-60% at 2 and 10μM and had no effect at 0.08 and 0.4μM.
CSN12182	Valspodar	121584-18-7	Valspodar is a P-glycoprotein P-gp inhibitor widely used in preclinical and clinical studies for overcoming multidrug resistance MDR
CSN14774	Taxinine B	18457-44-8	Taxinine B, a natural product isolated and purified from the barks of Taxus chinensis, can inhibit the drug transport by P-glycoprotein in multidrug-resistant cells, and shows stronger inhibitory effects than acetylsalicylic acid (ASA) on platelet aggregation induced by arachidonic acid (AA).
CSN18364	Tariquidar Methanesulfonate Hydrate	625375-83-9	Tariquidar methanesulfonate is a potent and specific inhibitor of P-glycoprotein P-gp with the high affinity Kd5109 nM
CSN12910	Tariquidar	206873-63-4	Tariquidar is a potent and selective noncompetitive inhibitor of P-glycoprotein with Kd of 51 nM reverses drug resistance in MDR cell Lines
CSN13177	Sinapine Thiocyanate	7431-77-8	Sinapine, an alkaloid isolated and purified from the seeds of Raphanus sativus L., possess antioxidant and radio-protective activities, downregulats multi-drug resistance 1 (MDR1) expression.
CSN22057	Sinapine	18696-26-9	Sinapine is an alkaloid from seeds of the cruciferous species which shows antioxidant and radio-protective activities and decreases expression of P-glycoprotein in Caco-2 cells.
CSN19434	Schizandrin	7432-28-2	Schizandrin is a natural product possessing antioxidant and anti-inflammatory activities.
CSN13555	Isosinensetin	17290-70-9	Isosinensetin exhibits HIV-1 protease inhibiting and antioxidant activities. It is a natural product isolated and purified from the fruit of Citrus aurantium L..
CSN15743	HM30181	849675-66-7	HM30181 is a potent and selective inhibitor of P-glycoprotein
CSN20429	Heliosterpenoid B	N/A	Heliosterpenoid B is a natural product isolated and purfied from the whole plants of Euphorbia helioscopia being potent inhibitors of P-glycoprotein ABCB1
CSN20428	Heliosterpenoid A	2109805-68-5	Heliosterpenoid A is a natural product isolated and purfied from the whole plants of Euphorbia helioscopia being potent inhibitors of P-glycoprotein ABCB1 and exhibiting cytotoxicity against MDA-MB-231 cell lines
CSN14838	Epimedokoreanin B	161068-53-7	Epimedokoreanin B is a natural product isolated and purified from the herbs of Epimedium brevicornum
CSN10894	Elacridar	143664-11-3	Elacridar is a P-glycoprotein inhibitor, and has been used both in vitro and in vivo as a tool inhibitor of P-glycoprotein (Pgp) to investigate the role of transporters in the disposition of various test molecules.
CSN13175	Elacridar HCl	143851-98-3	Elacridar HCl is a P-glycoprotein (P-gp) inhibitor, and has been used both in vitro and in vivo as a tool inhibitor of P-gp to investigate the role of transporters in the disposition of various test molecules.
CSN17662	Dofequidar	129716-58-1	Dofequidar is a quinoline compound which can reverse P-glycoprotein P-gp-mediated MDR
CSN17917	Dofequidar Fumarate	153653-30-6	Dofequidar fumarate an orally active quinoline compound has been reported to overcome MDR by inhibiting ABCB1P-gp ABCC1MDR-associated protein 1 or both
CSN22768	CP 100356 HCl	142715-48-8	CP 100356 HCl is a high affinity P-glycoprotein (P-gp) inhibitor with Kis of 58 and 94 nM for mouse Pgp1a and Pgp1b isoforms.
CSN23176	UCLA GP130 2	339303-87-6

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