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Opioid Receptor
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN20211 | TRV0109101 HCl | 2101210-22-2 | TRV0109101 hydrochloride a G protein-biased agonist of the -opioid receptor which may be an effective therapeutic avenue for managing chronic pain with reduced propensity for opioid-induced hyperalgesia |
| CSN20210 | TRV0109101 | 1401027-29-9 | TRV0109101 a G protein-biased agonist of the -opioid receptor which may be an effective therapeutic avenue for managing chronic pain with reduced propensity for opioid-induced hyperalgesia |
| CSN12642 | Trimebutine Maleate | 34140-59-5 | Trimebutine Maleate is an agonist effect on peripheral k and opiate receptors and also shows antimuscarinic effect |
| CSN12147 | Trimebutine | 39133-31-8 | Trimebutine is an agonist effect on peripheral k and opiate receptors and also shows antimuscarinic effect |
| CSN21214 | PZM-21 | 1997387-43-5 | PZM21 is a potent and selective opioid receptor agonist with an EC50 of 18 nM |
| CSN22475 | ORL1 Antagonist 1 | 1174985-59-1 | ORL1 antagonist 1 is an opioid receptor-like 1 ORL1 antagonist with an IC50 of 61 nM |
| CSN11515 | Nalmefene HCl | 58895-64-0 | Nalmefene hydrochloride originally known as nalmetrene is an opioid antagonistused primarily in the management of alcohol dependence It has also been investigated for the treatment of other addictions such as pathological gambling |
| CSN11529 | N-Desmethylclozapine | 6104-71-8 | N-Desmethylclozapine is a dengue virus inhibitor and an agonist of -opioid receptor |
| CSN11162 | Met-Enkephalin | 58569-55-4 | Met-enkephalin is an Opioid related peptide work as a potent agonist of the -opioid receptor and to a lesser extent the -opioid receptor with little to no effect on the -opioid receptor |
| CSN11381 | Meptazinol HCl | 59263-76-2 | Meptazinol HCl is both a partial agonist of 1 opioid receptor and an AChE inhibitor |
| CSN17469 | MCOPPB triHCl | 1108147-88-1 | MCOPPB trihydrochloride is a nociceptin receptor agonist with pKi of 1007 displaying weaker activity at other opioid receptors |
| CSN17719 | LY2795050 | 1346133-08-1 | LY2795050 is a selective -opioid Receptor KOR antagonist IC50072 nM and has the potential as a PET tracer to image KOR in vivo |
| CSN20227 | LY2444296 | 1346133-11-6 | LY2444296 is a short-acting kappa opioid receptor antagonist |
| CSN23719 | LY-2940094 Tartrate | 1307245-87-9 | LY-2940094 tartrate is the tartrate form of LY-2940094 which is an antagonist of nociceptin receptor that is used for the treatment of major depressive disorder and alcoholism |
| CSN20601 | LY2456302 | 1174130-61-0 | LY-2456302 is a potent and centrally-penetrant kappa opioid receptor antagonist with a Ki of 0.807 nM. |
| CSN11328 | Loperamide HCl | 34552-83-5 | Loperamide HCl is a potent and selective -opioid receptor agonist |
| CSN16622 | JTC-801 | 244218-51-7 | JTC-801 is a selective opioid receptor-like1 ORL1 receptor antagonist with IC50 of 94 nM and weakly inhibits receptors and |
| CSN16488 | JDTic | 361444-66-8 | JDTic is a highly selective antagonist for the -opioid receptor and without affecting the - or -opioid receptors |
| CSN18435 | JDTic 2HCl | 785835-79-2 | JDTic dihydrochloride is a highly selective antagonist for the -opioid receptor without affecting the - or -opioid receptors |
| CSN19796 | GSK-1521498 | 1007573-18-3 | GSK-1521498 is a -opioid receptor antagonist It has been shown to attenuate reward-driven compulsive behaviours such as stimulant drug seeking or binge eating in animals and humans |
| CSN10947 | Ethoheptazine | 77-15-6 | Ethoheptazine is an opioid analgesic from the phenazepane family |
| CSN10924 | Eptazocine | 72522-13-5 | Eptazocine interacts with opioid receptor and is classified as one of the opiate agonist-antagonist analgesics |
| CSN18678 | [D-Ala2]Leucine-Enkephalin | 64963-01-5 | D-Ala2Leucine-Enkephalin is a potent long-acting Leu-enkephalin analog agonist of delta opioid receptor |
| CSN19110 | Cebranopadol (1α,4α)stereoisomer | 863513-93-3 | Cebranopadol14stereoisomer is a stereoisomer of cebranopadol |
| CSN13503 | Cebranopadol | 863513-91-1 | Cebranopadol is an analgesic NOP and opioid receptor agonist with KisEC50s of 09 nM13 nM 07 nM12 nM 26 nM17 nM 18 nM110 nM for human NOP MOP KOP and delta-opioid peptide DOP receptor respectively |
| CSN17791 | BAN ORL 24 | 1401463-54-4 | BAN ORL 24 is a potent and selective NOP receptor antagonist IC50 values are 027 2500 6700 and 10000 nM for NOP - - and -receptors respectively |
| CSN23662 | AR-M 1000390 HCl | 209808-47-9 | AR-M 1000390 HCl is a non-peptidic and low-internalizing -selective opioid receptor agonist |
| CSN13513 | Alvimopan | 156053-89-3 | Alvimopan is a peripherally selective opioid mu receptor antagonist. |
| CSN17774 | Alvimopan Monohydrate | 1383577-62-5 | Alvimopan is a peripherally acting mu-opioid receptor PAM-OR IC50 17 nM antagonist for accelerating gastrointestinal recovery after surgery |
| CSN13650 | Alvimopan Dihydrate | 170098-38-1 | Alvimopan is a peripherally acting mu-opioid receptor (PAM-OR, IC50 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery. |
| CSN12425 | ADL-5859 HCl | 850173-95-4 | ADL-5859 HCl is both a -opioid receptor agonist Ki084 nM EC5020 nM and selectivity against opioid receptor and weak inhibitory activity at the hERG channel with IC50 value of 78 M |
| CSN11317 | (-)-Menthol | 2216-51-5 | --Menthol is a natural product obtained from the oils of corn mint peppermint or other mints as a weak kappa opioid receptor agonist It has local anesthetic and counterirritant qualities and used to relieve minor throat irritation |
| CSN18860 | (R)-ZINC-3573 | 2089389-15-9 | (R)-ZINC-3573 can activate endogenous MRGPRX2 in a human mast cell line and induce degranulation and calcium release. |
| CSN14746 | Akuammigine | 642-17-1 |
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