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Opioid Receptor

Opioid Receptor

Cat. No. Product Name CAS No. Information
CSN12642 Trimebutine Maleate   34140-59-5 Trimebutine Maleate is an agonist effect on peripheral k and opiate receptors and also shows antimuscarinic effect
CSN12147 Trimebutine   39133-31-8 Trimebutine is an agonist effect on peripheral k and opiate receptors and also shows antimuscarinic effect
CSN26718 SB-612111 371980-98-2 SB-612111 is a novel and potent human opiate receptor-like orphan receptor (ORL-1) antagonist with a high affinity for hORL-1 (Ki=0.33 nM). SB-612111 exhibits selectivity for μ-, κ- and δ-receptors with Ki values of 57.6 nM, 160.5 nM and 2109 nM, respecticely. SB-612111 effectively antagonizes the pronociceptive action of Nociceptin (HY-P0183) in an acute pain model[1].
CSN21214 PZM-21 1997387-43-5 PZM21 is a potent and selective opioid receptor agonist with an EC50 of 18 nM
CSN12166 Porcine Dynorphin A(1-13) 72957-38-1 Porcine dynorphin A(1-13) is a potent, endogenous -agonist.
CSN22475 ORL1 Antagonist 1 1174985-59-1 ORL1 antagonist 1 is an opioid receptor-like 1 ORL1 antagonist with an IC50 of 61 nM
CSN26717 LY2940094 1307245-86-8 LY2940094 is a potent and selective nociceptin receptor antagonist which inhibits excessive feeding behavior in rodents.
CSN17719 LY2795050 1346133-08-1 LY2795050 is a selective -opioid Receptor KOR antagonist IC50072 nM and has the potential as a PET tracer to image KOR in vivo
CSN20227 LY2444296 1346133-11-6 LY2444296 is a short-acting kappa opioid receptor antagonist
CSN23719 LY-2940094 Tartrate 1307245-87-9 LY-2940094 tartrate is the tartrate form of LY-2940094 which is an antagonist of nociceptin receptor that is used for the treatment of major depressive disorder and alcoholism
CSN20601 LY2456302 1174130-61-0 LY-2456302 is a potent and centrally-penetrant kappa opioid receptor antagonist with a Ki of 0.807 nM.
CSN16622 JTC-801 244218-51-7 JTC-801 is a selective opioid receptor-like1 ORL1 receptor antagonist with IC50 of 94 nM and weakly inhibits receptors and
CSN19796 GSK-1521498 1007573-18-3 GSK-1521498 is a -opioid receptor antagonist It has been shown to attenuate reward-driven compulsive behaviours such as stimulant drug seeking or binge eating in animals and humans
CSN19110 Cebranopadol (1α,4α)stereoisomer 863513-93-3 Cebranopadol14stereoisomer is a stereoisomer of cebranopadol
CSN13503 Cebranopadol 863513-91-1 Cebranopadol is an analgesic NOP and opioid receptor agonist with KisEC50s of 09 nM13 nM 07 nM12 nM 26 nM17 nM 18 nM110 nM for human NOP MOP KOP and delta-opioid peptide DOP receptor respectively
CSN25444 BRL 52537 hydrochloride 112282-24-3 BRL-52537 hydrochloride is a potent and highly selective κ-opioid agonist. It has neuroprotective effects in animal studies, and is used for research into potential treatments for stroke and heart attack as well as more general brain research.
CSN27537 Bevenopran 676500-67-7 Bevenopran is a peripheral μ-opioid receptor antagonist.
CSN17791 BAN ORL 24 1401463-54-4 BAN ORL 24 is a potent and selective NOP receptor antagonist IC50 values are 027 2500 6700 and 10000 nM for NOP - - and -receptors respectively
CSN21495 Asimadoline 153205-46-0 Asimadoline is an agonist of κ-opioid receptor (KOR) with IC50 of 1.2 nM.
CSN23662 AR-M 1000390 HCl 209808-47-9 AR-M 1000390 HCl is a non-peptidic and low-internalizing -selective opioid receptor agonist
CSN13513 Alvimopan   156053-89-3 Alvimopan is a peripherally selective opioid mu receptor antagonist.
CSN17774 Alvimopan Monohydrate 1383577-62-5 Alvimopan is a peripherally acting mu-opioid receptor PAM-OR IC50 17 nM antagonist for accelerating gastrointestinal recovery after surgery
CSN13650 Alvimopan Dihydrate 170098-38-1 Alvimopan is a peripherally acting mu-opioid receptor (PAM-OR, IC50 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery.
CSN12425 ADL-5859 HCl 850173-95-4 ADL-5859 HCl is both a -opioid receptor agonist Ki084 nM EC5020 nM and selectivity against opioid receptor and weak inhibitory activity at the hERG channel with IC50 value of 78 M
CSN14992 (Z)-Akuammidine 113973-31-2 (Z)-Akuammidine is a potent -opioid agonist isolated and purified from the roots of Gelsemium elegans.
CSN29545 SNC 80 156727-74-1 Highly selective non-peptide δ agonist
CSN27869 SCH 32615 83861-02-3
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