Welcome to CSNpharm! For Research Use Only!
Opioid Receptor
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN12642 | Trimebutine Maleate | 34140-59-5 | Trimebutine Maleate is an agonist effect on peripheral k and opiate receptors and also shows antimuscarinic effect |
| CSN12147 | Trimebutine | 39133-31-8 | Trimebutine is an agonist effect on peripheral k and opiate receptors and also shows antimuscarinic effect |
| CSN26718 | SB-612111 | 371980-98-2 | SB-612111 is a novel and potent human opiate receptor-like orphan receptor (ORL-1) antagonist with a high affinity for hORL-1 (Ki=0.33 nM). SB-612111 exhibits selectivity for μ-, κ- and δ-receptors with Ki values of 57.6 nM, 160.5 nM and 2109 nM, respecticely. SB-612111 effectively antagonizes the pronociceptive action of Nociceptin (HY-P0183) in an acute pain model[1]. |
| CSN21214 | PZM-21 | 1997387-43-5 | PZM21 is a potent and selective opioid receptor agonist with an EC50 of 18 nM |
| CSN12166 | Porcine Dynorphin A(1-13) | 72957-38-1 | Porcine dynorphin A(1-13) is a potent, endogenous -agonist. |
| CSN22475 | ORL1 Antagonist 1 | 1174985-59-1 | ORL1 antagonist 1 is an opioid receptor-like 1 ORL1 antagonist with an IC50 of 61 nM |
| CSN26717 | LY2940094 | 1307245-86-8 | LY2940094 is a potent and selective nociceptin receptor antagonist which inhibits excessive feeding behavior in rodents. |
| CSN17719 | LY2795050 | 1346133-08-1 | LY2795050 is a selective -opioid Receptor KOR antagonist IC50072 nM and has the potential as a PET tracer to image KOR in vivo |
| CSN20227 | LY2444296 | 1346133-11-6 | LY2444296 is a short-acting kappa opioid receptor antagonist |
| CSN23719 | LY-2940094 Tartrate | 1307245-87-9 | LY-2940094 tartrate is the tartrate form of LY-2940094 which is an antagonist of nociceptin receptor that is used for the treatment of major depressive disorder and alcoholism |
| CSN20601 | LY2456302 | 1174130-61-0 | LY-2456302 is a potent and centrally-penetrant kappa opioid receptor antagonist with a Ki of 0.807 nM. |
| CSN16622 | JTC-801 | 244218-51-7 | JTC-801 is a selective opioid receptor-like1 ORL1 receptor antagonist with IC50 of 94 nM and weakly inhibits receptors and |
| CSN19796 | GSK-1521498 | 1007573-18-3 | GSK-1521498 is a -opioid receptor antagonist It has been shown to attenuate reward-driven compulsive behaviours such as stimulant drug seeking or binge eating in animals and humans |
| CSN19110 | Cebranopadol (1α,4α)stereoisomer | 863513-93-3 | Cebranopadol14stereoisomer is a stereoisomer of cebranopadol |
| CSN13503 | Cebranopadol | 863513-91-1 | Cebranopadol is an analgesic NOP and opioid receptor agonist with KisEC50s of 09 nM13 nM 07 nM12 nM 26 nM17 nM 18 nM110 nM for human NOP MOP KOP and delta-opioid peptide DOP receptor respectively |
| CSN25444 | BRL 52537 hydrochloride | 112282-24-3 | BRL-52537 hydrochloride is a potent and highly selective κ-opioid agonist. It has neuroprotective effects in animal studies, and is used for research into potential treatments for stroke and heart attack as well as more general brain research. |
| CSN27537 | Bevenopran | 676500-67-7 | Bevenopran is a peripheral μ-opioid receptor antagonist. |
| CSN17791 | BAN ORL 24 | 1401463-54-4 | BAN ORL 24 is a potent and selective NOP receptor antagonist IC50 values are 027 2500 6700 and 10000 nM for NOP - - and -receptors respectively |
| CSN21495 | Asimadoline | 153205-46-0 | Asimadoline is an agonist of κ-opioid receptor (KOR) with IC50 of 1.2 nM. |
| CSN23662 | AR-M 1000390 HCl | 209808-47-9 | AR-M 1000390 HCl is a non-peptidic and low-internalizing -selective opioid receptor agonist |
| CSN13513 | Alvimopan | 156053-89-3 | Alvimopan is a peripherally selective opioid mu receptor antagonist. |
| CSN17774 | Alvimopan Monohydrate | 1383577-62-5 | Alvimopan is a peripherally acting mu-opioid receptor PAM-OR IC50 17 nM antagonist for accelerating gastrointestinal recovery after surgery |
| CSN13650 | Alvimopan Dihydrate | 170098-38-1 | Alvimopan is a peripherally acting mu-opioid receptor (PAM-OR, IC50 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery. |
| CSN12425 | ADL-5859 HCl | 850173-95-4 | ADL-5859 HCl is both a -opioid receptor agonist Ki084 nM EC5020 nM and selectivity against opioid receptor and weak inhibitory activity at the hERG channel with IC50 value of 78 M |
| CSN14992 | (Z)-Akuammidine | 113973-31-2 | (Z)-Akuammidine is a potent -opioid agonist isolated and purified from the roots of Gelsemium elegans. |
| CSN29545 | SNC 80 | 156727-74-1 | Highly selective non-peptide δ agonist |
| CSN27869 | SCH 32615 | 83861-02-3 |
+1-708-781-1677
+1-708-286-6026
sales@csnpharm.com
