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Opioid Receptor
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN22049 | [Met5]-Enkephalin Amide | 60117-17-1 | [Met5]-Enkephalin, amide is an agonist for δ opioid receptors as well as putative ζ (zeta) opioid receptors. |
| CSN20210 | TRV0109101 | 1401027-29-9 | TRV0109101 a G protein-biased agonist of the -opioid receptor which may be an effective therapeutic avenue for managing chronic pain with reduced propensity for opioid-induced hyperalgesia |
| CSN12642 | Trimebutine Maleate | 34140-59-5 | Trimebutine Maleate is an agonist effect on peripheral k and opiate receptors and also shows antimuscarinic effect |
| CSN12147 | Trimebutine | 39133-31-8 | Trimebutine is an agonist effect on peripheral k and opiate receptors and also shows antimuscarinic effect |
| CSN21214 | PZM-21 | 1997387-43-5 | PZM21 is a potent and selective opioid receptor agonist with an EC50 of 18 nM |
| CSN12166 | Porcine Dynorphin A(1-13) | 72957-38-1 | Porcine dynorphin A(1-13) is a potent, endogenous -agonist. |
| CSN22475 | ORL1 Antagonist 1 | 1174985-59-1 | ORL1 antagonist 1 is an opioid receptor-like 1 ORL1 antagonist with an IC50 of 61 nM |
| CSN21766 | Nociceptin | 170713-75-4 | Nociceptin, a 17 amino acid neuropeptide, is endogenous ligand for the opioid-like G-protein coupled receptor, ORL1 (opioid receptor-like 1). |
| CSN11529 | N-Desmethylclozapine | 6104-71-8 | N-Desmethylclozapine is a dengue virus inhibitor and an agonist of -opioid receptor |
| CSN11162 | Met-Enkephalin | 58569-55-4 | Met-enkephalin is an Opioid related peptide work as a potent agonist of the -opioid receptor and to a lesser extent the -opioid receptor with little to no effect on the -opioid receptor |
| CSN11381 | Meptazinol HCl | 59263-76-2 | Meptazinol HCl is both a partial agonist of 1 opioid receptor and an AChE inhibitor |
| CSN17469 | MCOPPB triHCl | 1108147-88-1 | MCOPPB 3HCl is a nociceptin receptor agonist with pKi of 10.07, displaying weaker activity at other opioid receptors. |
| CSN17719 | LY2795050 | 1346133-08-1 | LY2795050 is a selective -opioid Receptor KOR antagonist IC50072 nM and has the potential as a PET tracer to image KOR in vivo |
| CSN20227 | LY2444296 | 1346133-11-6 | LY2444296 is a short-acting kappa opioid receptor antagonist |
| CSN23719 | LY-2940094 Tartrate | 1307245-87-9 | LY-2940094 tartrate is the tartrate form of LY-2940094 which is an antagonist of nociceptin receptor that is used for the treatment of major depressive disorder and alcoholism |
| CSN20601 | LY2456302 | 1174130-61-0 | LY-2456302 is a potent and centrally-penetrant kappa opioid receptor antagonist with a Ki of 0.807 nM. |
| CSN11328 | Loperamide HCl | 34552-83-5 | Loperamide HCl is a potent and selective -opioid receptor agonist |
| CSN21707 | Leu-Enkephalinamide | 60117-24-0 | Leu-enkephalin amide, found naturally in the brains of many animals, is an endogenous opioid peptide neurotransmitter with the amino acid sequence Tyr-Gly-Gly-Phe-Leu. |
| CSN16622 | JTC-801 | 244218-51-7 | JTC-801 is a selective opioid receptor-like1 ORL1 receptor antagonist with IC50 of 94 nM and weakly inhibits receptors and |
| CSN16488 | JDTic | 361444-66-8 | JDTic is a highly selective antagonist for the -opioid receptor and without affecting the - or -opioid receptors |
| CSN18435 | JDTic 2HCl | 785835-79-2 | JDTic 2HCl is a highly selective antagonist for the κ-opioid receptor without affecting the μ- or δ-opioid receptors. |
| CSN21596 | Gluten Exorphin C | 142479-62-7 | Gluten exorphin C, an opioid peptide derived from wheat gluten, can inhibit μ opioid and δ opioid with IC50 values of 40 μM and 13.5 μM in the GPI and MVD assays. |
| CSN10947 | Ethoheptazine | 77-15-6 | Ethoheptazine is an opioid analgesic from the phenazepane family |
| CSN10924 | Eptazocine | 72522-13-5 | Eptazocine interacts with opioid receptor and is classified as one of the opiate agonist-antagonist analgesics |
| CSN21628 | Endomorphin 2 | 141801-26-5 | Endomorphin 2, an endogenous neuropeptide, is agonist of μ-opioid receptor with Ki of 0.69 nM that has analgesic and gastrointestinal properties. |
| CSN21627 | Endomorphin 1 | 189388-22-5 | Endomorphin 1 is a selective agonist of μ-opioid receptor with reasonable affinities for kappa3 binding sites (Ki value between 20 and 30 nM). |
| CSN21597 | Deltorphin I | 122752-15-2 | Deltorphin I is a selective agonist of δ-opioid receptor. |
| CSN21598 | Deltorphin 2 | 122752-16-3 | Deltorphin 2 is selective δ2 opioid receptor agonist. |
| CSN19110 | Cebranopadol (1α,4α)stereoisomer | 863513-93-3 | Cebranopadol14stereoisomer is a stereoisomer of cebranopadol |
| CSN13503 | Cebranopadol | 863513-91-1 | Cebranopadol is an analgesic NOP and opioid receptor agonist with KisEC50s of 09 nM13 nM 07 nM12 nM 26 nM17 nM 18 nM110 nM for human NOP MOP KOP and delta-opioid peptide DOP receptor respectively |
| CSN25444 | BRL 52537 hydrochloride | 112282-24-3 | BRL-52537 hydrochloride is a potent and highly selective κ-opioid agonist. It has neuroprotective effects in animal studies, and is used for research into potential treatments for stroke and heart attack as well as more general brain research. |
| CSN27537 | Bevenopran | 676500-67-7 | Bevenopran is a peripheral μ-opioid receptor antagonist. |
| CSN24259 | BAN ORL 24diHCl- | 475150-69-7 | BAN ORL 24 is a potent and selective NOP receptor antagonist. (IC50 values are 0.27, 2500, 6700 and > 10000 nM for NOP, κ-, μ- and δ-receptors respectively). |
| CSN17791 | BAN ORL 24 | 1401463-54-4 | BAN ORL 24 is a potent and selective NOP receptor antagonist IC50 values are 027 2500 6700 and 10000 nM for NOP - - and -receptors respectively |
| CSN21495 | Asimadoline | 153205-46-0 | Asimadoline is an agonist of κ-opioid receptor (KOR) with IC50 of 1.2 nM. |
| CSN23662 | AR-M 1000390 HCl | 209808-47-9 | AR-M 1000390 HCl is a non-peptidic and low-internalizing -selective opioid receptor agonist |
| CSN13513 | Alvimopan | 156053-89-3 | Alvimopan is a peripherally selective opioid mu receptor antagonist. |
| CSN17774 | Alvimopan Monohydrate | 1383577-62-5 | Alvimopan is a peripherally acting mu-opioid receptor PAM-OR IC50 17 nM antagonist for accelerating gastrointestinal recovery after surgery |
| CSN13650 | Alvimopan Dihydrate | 170098-38-1 | Alvimopan is a peripherally acting mu-opioid receptor (PAM-OR, IC50 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery. |
| CSN14746 | Akuammigine | 642-17-1 | Akuammidine, a natural product isolated and purified from the herbs of Picralima nitida with in vitro antimalarial activity, shows a preference for mu-opioid binding sites with Ki values of 0.6, 2.4 and 8.6 mM at mu-, delta- and kappa-opioid binding sites, respectively and the agonist actions of akuammidine in the mouse-isolated vas deferens were antagonised by naloxone and the mu-opioid receptor selective antagonist D-Phe-Cys-Tyr-D-Trp-Orn-Thr-Pen-Thr-NH2 (CTOP) confirming an action at mu-opioid receptors, and competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding pA2 values of 4.68. |
| CSN21463 | Adrenorphin | 88377-68-8 | Adrenorphin is an agonist of μ-opioid receptor with Ki of 12 nM. |
| CSN12425 | ADL-5859 HCl | 850173-95-4 | ADL-5859 HCl is both a -opioid receptor agonist Ki084 nM EC5020 nM and selectivity against opioid receptor and weak inhibitory activity at the hERG channel with IC50 value of 78 M |
| CSN11317 | (-)-Menthol | 2216-51-5 | --Menthol is a natural product obtained from the oils of corn mint peppermint or other mints as a weak kappa opioid receptor agonist It has local anesthetic and counterirritant qualities and used to relieve minor throat irritation |
| CSN14992 | (Z)-Akuammidine | 113973-31-2 | (Z)-Akuammidine is a potent -opioid agonist isolated and purified from the roots of Gelsemium elegans. |
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