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Opioid Receptor

Opioid Receptor

Cat. No. Product Name CAS No. Information
CSN22049 [Met5]-Enkephalin Amide 60117-17-1 [Met5]-Enkephalin, amide is an agonist for δ opioid receptors as well as putative ζ (zeta) opioid receptors.
CSN20210 TRV0109101 1401027-29-9 TRV0109101 a G protein-biased agonist of the -opioid receptor which may be an effective therapeutic avenue for managing chronic pain with reduced propensity for opioid-induced hyperalgesia
CSN12642 Trimebutine Maleate   34140-59-5 Trimebutine Maleate is an agonist effect on peripheral k and opiate receptors and also shows antimuscarinic effect
CSN12147 Trimebutine   39133-31-8 Trimebutine is an agonist effect on peripheral k and opiate receptors and also shows antimuscarinic effect
CSN21214 PZM-21 1997387-43-5 PZM21 is a potent and selective opioid receptor agonist with an EC50 of 18 nM
CSN12166 Porcine Dynorphin A(1-13) 72957-38-1 Porcine dynorphin A(1-13) is a potent, endogenous -agonist.
CSN22475 ORL1 Antagonist 1 1174985-59-1 ORL1 antagonist 1 is an opioid receptor-like 1 ORL1 antagonist with an IC50 of 61 nM
CSN21766 Nociceptin 170713-75-4 Nociceptin, a 17 amino acid neuropeptide, is endogenous ligand for the opioid-like G-protein coupled receptor, ORL1 (opioid receptor-like 1).
CSN11529 N-Desmethylclozapine 6104-71-8 N-Desmethylclozapine is a dengue virus inhibitor and an agonist of -opioid receptor
CSN11162 Met-Enkephalin   58569-55-4 Met-enkephalin is an Opioid related peptide work as a potent agonist of the -opioid receptor and to a lesser extent the -opioid receptor with little to no effect on the -opioid receptor
CSN11381 Meptazinol HCl   59263-76-2 Meptazinol HCl is both a partial agonist of 1 opioid receptor and an AChE inhibitor
CSN17469 MCOPPB triHCl 1108147-88-1 MCOPPB 3HCl is a nociceptin receptor agonist with pKi of 10.07, displaying weaker activity at other opioid receptors.
CSN17719 LY2795050 1346133-08-1 LY2795050 is a selective -opioid Receptor KOR antagonist IC50072 nM and has the potential as a PET tracer to image KOR in vivo
CSN20227 LY2444296 1346133-11-6 LY2444296 is a short-acting kappa opioid receptor antagonist
CSN23719 LY-2940094 Tartrate 1307245-87-9 LY-2940094 tartrate is the tartrate form of LY-2940094 which is an antagonist of nociceptin receptor that is used for the treatment of major depressive disorder and alcoholism
CSN20601 LY2456302 1174130-61-0 LY-2456302 is a potent and centrally-penetrant kappa opioid receptor antagonist with a Ki of 0.807 nM.
CSN11328 Loperamide HCl   34552-83-5 Loperamide HCl is a potent and selective -opioid receptor agonist
CSN21707 Leu-Enkephalinamide 60117-24-0 Leu-enkephalin amide, found naturally in the brains of many animals, is an endogenous opioid peptide neurotransmitter with the amino acid sequence Tyr-Gly-Gly-Phe-Leu.
CSN16622 JTC-801 244218-51-7 JTC-801 is a selective opioid receptor-like1 ORL1 receptor antagonist with IC50 of 94 nM and weakly inhibits receptors and
CSN16488 JDTic 361444-66-8 JDTic is a highly selective antagonist for the -opioid receptor and without affecting the - or -opioid receptors
CSN18435 JDTic 2HCl 785835-79-2 JDTic 2HCl is a highly selective antagonist for the κ-opioid receptor without affecting the μ- or δ-opioid receptors.
CSN21596 Gluten Exorphin C 142479-62-7 Gluten exorphin C, an opioid peptide derived from wheat gluten, can inhibit μ opioid and δ opioid with IC50 values of 40 μM and 13.5 μM in the GPI and MVD assays.
CSN10947 Ethoheptazine 77-15-6 Ethoheptazine is an opioid analgesic from the phenazepane family
CSN10924 Eptazocine 72522-13-5 Eptazocine interacts with opioid receptor and is classified as one of the opiate agonist-antagonist analgesics
CSN21628 Endomorphin 2 141801-26-5 Endomorphin 2, an endogenous neuropeptide, is agonist of μ-opioid receptor with Ki of 0.69 nM that has analgesic and gastrointestinal properties.
CSN21627 Endomorphin 1 189388-22-5 Endomorphin 1 is a selective agonist of μ-opioid receptor with reasonable affinities for kappa3 binding sites (Ki value between 20 and 30 nM).
CSN21597 Deltorphin I 122752-15-2 Deltorphin I is a selective agonist of δ-opioid receptor.
CSN21598 Deltorphin 2 122752-16-3 Deltorphin 2 is selective δ2 opioid receptor agonist.
CSN19110 Cebranopadol (1α,4α)stereoisomer 863513-93-3 Cebranopadol14stereoisomer is a stereoisomer of cebranopadol
CSN13503 Cebranopadol 863513-91-1 Cebranopadol is an analgesic NOP and opioid receptor agonist with KisEC50s of 09 nM13 nM 07 nM12 nM 26 nM17 nM 18 nM110 nM for human NOP MOP KOP and delta-opioid peptide DOP receptor respectively
CSN25444 BRL 52537 hydrochloride 112282-24-3 BRL-52537 hydrochloride is a potent and highly selective κ-opioid agonist. It has neuroprotective effects in animal studies, and is used for research into potential treatments for stroke and heart attack as well as more general brain research.
CSN27537 Bevenopran 676500-67-7 Bevenopran is a peripheral μ-opioid receptor antagonist.
CSN24259 BAN ORL 24diHCl- 475150-69-7 BAN ORL 24 is a potent and selective NOP receptor antagonist. (IC50 values are 0.27, 2500, 6700 and > 10000 nM for NOP, κ-, μ- and δ-receptors respectively).
CSN17791 BAN ORL 24 1401463-54-4 BAN ORL 24 is a potent and selective NOP receptor antagonist IC50 values are 027 2500 6700 and 10000 nM for NOP - - and -receptors respectively
CSN21495 Asimadoline 153205-46-0 Asimadoline is an agonist of κ-opioid receptor (KOR) with IC50 of 1.2 nM.
CSN23662 AR-M 1000390 HCl 209808-47-9 AR-M 1000390 HCl is a non-peptidic and low-internalizing -selective opioid receptor agonist
CSN13513 Alvimopan   156053-89-3 Alvimopan is a peripherally selective opioid mu receptor antagonist.
CSN17774 Alvimopan Monohydrate 1383577-62-5 Alvimopan is a peripherally acting mu-opioid receptor PAM-OR IC50 17 nM antagonist for accelerating gastrointestinal recovery after surgery
CSN13650 Alvimopan Dihydrate 170098-38-1 Alvimopan is a peripherally acting mu-opioid receptor (PAM-OR, IC50 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery.
CSN14746 Akuammigine 642-17-1 Akuammidine, a natural product isolated and purified from the herbs of Picralima nitida with in vitro antimalarial activity, shows a preference for mu-opioid binding sites with Ki values of 0.6, 2.4 and 8.6 mM at mu-, delta- and kappa-opioid binding sites, respectively and the agonist actions of akuammidine in the mouse-isolated vas deferens were antagonised by naloxone and the mu-opioid receptor selective antagonist D-Phe-Cys-Tyr-D-Trp-Orn-Thr-Pen-Thr-NH2 (CTOP) confirming an action at mu-opioid receptors, and competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding pA2 values of 4.68.
CSN21463 Adrenorphin 88377-68-8 Adrenorphin is an agonist of μ-opioid receptor with Ki of 12 nM.
CSN12425 ADL-5859 HCl 850173-95-4 ADL-5859 HCl is both a -opioid receptor agonist Ki084 nM EC5020 nM and selectivity against opioid receptor and weak inhibitory activity at the hERG channel with IC50 value of 78 M
CSN11317 (-)-Menthol   2216-51-5 --Menthol is a natural product obtained from the oils of corn mint peppermint or other mints as a weak kappa opioid receptor agonist It has local anesthetic and counterirritant qualities and used to relieve minor throat irritation
CSN14992 (Z)-Akuammidine 113973-31-2 (Z)-Akuammidine is a potent -opioid agonist isolated and purified from the roots of Gelsemium elegans.
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