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Opioid Receptor

Opioid Receptor

Cat. No. Product Name CAS No. Information
CSN20211 TRV0109101 HCl 2101210-22-2 TRV0109101 hydrochloride a G protein-biased agonist of the -opioid receptor which may be an effective therapeutic avenue for managing chronic pain with reduced propensity for opioid-induced hyperalgesia
CSN20210 TRV0109101 1401027-29-9 TRV0109101 a G protein-biased agonist of the -opioid receptor which may be an effective therapeutic avenue for managing chronic pain with reduced propensity for opioid-induced hyperalgesia
CSN12642 Trimebutine Maleate   34140-59-5 Trimebutine Maleate is an agonist effect on peripheral k and opiate receptors and also shows antimuscarinic effect
CSN12147 Trimebutine   39133-31-8 Trimebutine is an agonist effect on peripheral k and opiate receptors and also shows antimuscarinic effect
CSN21214 PZM-21 1997387-43-5 PZM21 is a potent and selective opioid receptor agonist with an EC50 of 18 nM
CSN22475 ORL1 Antagonist 1 1174985-59-1 ORL1 antagonist 1 is an opioid receptor-like 1 ORL1 antagonist with an IC50 of 61 nM
CSN11529 N-Desmethylclozapine 6104-71-8 N-Desmethylclozapine is a dengue virus inhibitor and an agonist of -opioid receptor
CSN11162 Met-Enkephalin   58569-55-4 Met-enkephalin is an Opioid related peptide work as a potent agonist of the -opioid receptor and to a lesser extent the -opioid receptor with little to no effect on the -opioid receptor
CSN11381 Meptazinol HCl   59263-76-2 Meptazinol HCl is both a partial agonist of 1 opioid receptor and an AChE inhibitor
CSN17469 MCOPPB triHCl 1108147-88-1 MCOPPB trihydrochloride is a nociceptin receptor agonist with pKi of 1007 displaying weaker activity at other opioid receptors
CSN17719 LY2795050 1346133-08-1 LY2795050 is a selective -opioid Receptor KOR antagonist IC50072 nM and has the potential as a PET tracer to image KOR in vivo
CSN20227 LY2444296 1346133-11-6 LY2444296 is a short-acting kappa opioid receptor antagonist
CSN23719 LY-2940094 Tartrate 1307245-87-9 LY-2940094 tartrate is the tartrate form of LY-2940094 which is an antagonist of nociceptin receptor that is used for the treatment of major depressive disorder and alcoholism
CSN20601 LY2456302 1174130-61-0 LY-2456302 is a potent and centrally-penetrant kappa opioid receptor antagonist with a Ki of 0.807 nM.
CSN11328 Loperamide HCl   34552-83-5 Loperamide HCl is a potent and selective -opioid receptor agonist
CSN16622 JTC-801 244218-51-7 JTC-801 is a selective opioid receptor-like1 ORL1 receptor antagonist with IC50 of 94 nM and weakly inhibits receptors and
CSN16488 JDTic 361444-66-8 JDTic is a highly selective antagonist for the -opioid receptor and without affecting the - or -opioid receptors
CSN18435 JDTic 2HCl 785835-79-2 JDTic dihydrochloride is a highly selective antagonist for the -opioid receptor without affecting the - or -opioid receptors
CSN19796 GSK-1521498 1007573-18-3 GSK-1521498 is a -opioid receptor antagonist It has been shown to attenuate reward-driven compulsive behaviours such as stimulant drug seeking or binge eating in animals and humans
CSN10947 Ethoheptazine 77-15-6 Ethoheptazine is an opioid analgesic from the phenazepane family
CSN10924 Eptazocine 72522-13-5 Eptazocine interacts with opioid receptor and is classified as one of the opiate agonist-antagonist analgesics
CSN19110 Cebranopadol (1α,4α)stereoisomer 863513-93-3 Cebranopadol14stereoisomer is a stereoisomer of cebranopadol
CSN13503 Cebranopadol 863513-91-1 Cebranopadol is an analgesic NOP and opioid receptor agonist with KisEC50s of 09 nM13 nM 07 nM12 nM 26 nM17 nM 18 nM110 nM for human NOP MOP KOP and delta-opioid peptide DOP receptor respectively
CSN17791 BAN ORL 24 1401463-54-4 BAN ORL 24 is a potent and selective NOP receptor antagonist IC50 values are 027 2500 6700 and 10000 nM for NOP - - and -receptors respectively
CSN23662 AR-M 1000390 HCl 209808-47-9 AR-M 1000390 HCl is a non-peptidic and low-internalizing -selective opioid receptor agonist
CSN13513 Alvimopan   156053-89-3 Alvimopan is a peripherally selective opioid mu receptor antagonist.
CSN17774 Alvimopan Monohydrate 1383577-62-5 Alvimopan is a peripherally acting mu-opioid receptor PAM-OR IC50 17 nM antagonist for accelerating gastrointestinal recovery after surgery
CSN13650 Alvimopan Dihydrate 170098-38-1 Alvimopan is a peripherally acting mu-opioid receptor (PAM-OR, IC50 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery.
CSN12425 ADL-5859 HCl 850173-95-4 ADL-5859 HCl is both a -opioid receptor agonist Ki084 nM EC5020 nM and selectivity against opioid receptor and weak inhibitory activity at the hERG channel with IC50 value of 78 M
CSN11317 (-)-Menthol   2216-51-5 --Menthol is a natural product obtained from the oils of corn mint peppermint or other mints as a weak kappa opioid receptor agonist It has local anesthetic and counterirritant qualities and used to relieve minor throat irritation
CSN18860 (R)-ZINC-3573 2089389-15-9 (R)-ZINC-3573 can activate endogenous MRGPRX2 in a human mast cell line and induce degranulation and calcium release.
CSN14746 Akuammigine 642-17-1
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