NMDAR
Cat. No. | Product Name | CAS No. | Information |
---|---|---|---|
CSN21328 | UK-240455 | 178908-09-3 | UK-240455 is a potent and selective N-methyl D-aspartate NMDA glycine site antagonist |
CSN24287 | Traxoprodil mesylate | 189894-57-3 | Traxoprodil a selective antagonist of the NR2B subunit of the NMDA receptor. |
CSN12978 | Traxoprodil | 134234-12-1 | Traxoprodil a selective antagonist of the NR2B subunit of the NMDA receptor |
CSN11907 | SDZ 220-581 | 174575-17-8 | SDZ 220-581 is a potent competitive antagonist at the NMDA glutamate receptor subtype pKi 77 |
CSN15699 | Sarcosine | 107-97-1 | Sarcosine is an NMDAR co-agonist at the glycine binding site. It is an intermediate and byproduct in glycine synthesis and degradation. |
CSN17353 | Ro 25-6981 | 169274-78-6 | Ro 25-6981 is a potent and selective activity-dependent blocker of NMDA receptors containing the NR2B subunit |
CSN17520 | Rapastinel | 117928-94-6 | Rapastinel is a putative NMDAR functional glycine-site partial agonist |
CSN23523 | Quinolinic acid | 89-00-9 | Quinolinic acid is both a selective agonist at NMDA receptors and also a precursor for the formation of NAD |
CSN11780 | Procyclidine HCl | 1508-76-5 | Procyclidine HCl is an potent anti-cholinergic agent, and is also known to have NMDA antagonist properties. |
CSN11618 | Orphenadrine Citrate | 4682-36-4 | Orphenadrine Citrate is both an uncompetitive NMDA receptor antagonist IC50 value of 162 M and a mAChR antagonist with IC50 value of 037 M |
CSN24186 | NMDAR antagonist 1 | 2220162-06-9 | NMDAR antagonist 1 is a NR2B-selective NMDAR antagonist. |
CSN13790 | NMDA | 6384-92-5 | NMDA is an amino acid derived specific agonist at the NMDA receptor |
CSN11379 | Mephenesin | 59-47-2 | Mephenesin is a centrally acting muscle relaxant which may work as an NMDA receptor antagonist. |
CSN13916 | MDL 105519 | 161230-88-2 | MDL 105519 is a potent and selective inhibitor of 3Hglycine binding to the NMDA receptor with Kd of 389 nM |
CSN17128 | L-701,324 | 142326-59-8 | L-701324 is an orally active and long acting anticonvulsant with high affinity and selectivity for the glycine site on the NMDA receptor |
CSN21303 | Kynurenic Acid Sodium | 2439-02-3 | Kynurenic acid, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, 7 nicotinic acetylcholine receptor. Kynurenic acid is also a selective ligand of the GPR35 receptor. |
CSN11186 | Ifenprodil Tartrate | 23210-58-4 | Ifenprodil Tartrate is a high affinity and atypical noncompetitive NMDA receptor antagonist with IC50 of 03 M |
CSN21125 | Ibotenic Acid | 2552-55-8 | Ibotenic acid has agonist activity at both the N-methyl-D-aspartate NMDA and trans-ACPD or metabolotropic quisqualate Qm receptor sites |
CSN10988 | Felbamate | 25451-15-4 | Felbamate is a potent nonsedative anticonvulsant whose clinical effect may be related to the inhibition of N-methyl-D-aspartate NMDA |
CSN10256 | Eliprodil | 119431-25-3 | Eliprodil can antogonize GluN2B-selective NMDA in a non-competitive manner with IC50 value of 1 M It is also a 1 ligand with Ki value of 0013 M |
CSN21590 | D-AP5 | 79055-68-8 | D-AP5 is an antagonist of NMDA receptor (N-methyl-D-aspartate receptor). |
CSN19842 | CGP 37849 | 127910-31-0 | CGP 37849 is a potent selective and competitive NMDA receptor antagonist Ki 35 nM |
CSN10502 | Budipine | 57982-78-2 | Budipine is an uncompetitive NMDAR antagonist used as an antiparkinson agent |
CSN22086 | 7-Chlorokynurenic Acid Sodium Salt | 1263094-00-3 | 7-Chlorokynurenic acid sodium salt is a selective antagonist at the glycine modulatory site of the N-methyl-D-aspartate receptor complex and also a potent inhibitor of the reuptake of glutamate into synaptic vesicles with Ki of 0.59 μM. |
CSN24923 | 6-Methoxy-2-naphthoic acid | 2471-70-7 | 6-Methoxy-2-naphthoic acid is an modulator of NMDAR. |
CSN25440 | ACBC | 22264-50-2 | 1-Aminocyclobutanecarboxylic acid is a NMDA receptor partial agonist acting at the glycine site, NR1. |
CSN23429 | L-Glutamic Acid | 56-86-0 | (S)-Glutamic acid acts as an excitatory neurotransmitter in the central nervous system. |
CSN25118 | (R)-Serine | 312-84-5 | (R)-Serine is the R-enantiomer of serine, which is used in the biosynthesis of proteins. |
CSN25441 | (-)-Aspartic acid | 1783-96-6 | (-)-Aspartic acid is an endogenous NMDA receptor agonist. |
CSN13883 | (+)-MK 801 Maleate | 77086-22-7 | ()-MK 801 Maleate is a highly potent, selective and non-competitive NMDA receptor antagonist with Ki of 30.5 nM. |