NK Receptor
Cat. No. | Product Name | CAS No. | Information |
---|---|---|---|
CSN13678 | Talnetant | 174636-32-9 | Talnetant is a potent and selective NK3 receptor antagonist ki14 nM hNK-3-CHO and is 100-fold selective for the hNK-3 versus hNK-2 receptor with no affinity for the hNK-1 at concentrations up to 100 M |
CSN17283 | SB-222200 | 174635-69-9 | SB-222200 is a selective reversible and competitive antagonist of human NK-3 receptor Ki44 nM that effectively crosses the blood-brain barrier |
CSN16120 | Netupitant | 290297-26-6 | Netupitant a potent and highly selective NK1 receptor antagonist with Ki of 095 nM |
CSN25315 | L-732138 | 148451-96-1 | L-732138 is a potent and highly selective competitive tachykinin NK1 receptor antagonist with IC50 of 2.3 nM. |
CSN18008 | Fosaprepitant | 172673-20-0 | Fosaprepitant is a neurokinin-1 receptor antagonist for the prevention of chemotherapy-induced nausea and vomiting |
CSN12336 | Fosaprepitant Dimeglumine | 265121-04-8 | Fosaprepitant Dimeglumine is a prodrug for aprepitant which is a selective and high-affinity antagonist of NK1 receptor. |
CSN10324 | Aprepitant | 170729-80-3 | Aprepitant is a selective and high-affinity neurokinin-1 receptor antagonist with IC50 of 0.1 nM. |