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NK Receptor
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN19815 | Tradipitant | 622370-35-8 | Tradipitant is the 2nd generation neurokinin-1 receptor antagonist, which showed activity in preclinical anxiety models. |
| CSN13678 | Talnetant | 174636-32-9 | Talnetant is a potent and selective NK3 receptor antagonist ki14 nM hNK-3-CHO and is 100-fold selective for the hNK-3 versus hNK-2 receptor with no affinity for the hNK-1 at concentrations up to 100 M |
| CSN18094 | Talnetant HCl | 204519-66-4 | Talnetant hydrochloride is a potent and selective NK3 receptor antagonist (ki1.4 nM, hNK-3-CHO), 100-fold selective for the hNK-3 versus hNK-2 receptor, with no affinity for the hNK-1 at concentrations up to 100 M. |
| CSN22504 | Serlopitant | 860642-69-9 | Serlopitant is a selective Neurokinin-1 (NK-1) receptor antagonist. |
| CSN17283 | SB-222200 | 174635-69-9 | SB-222200 is a selective reversible and competitive antagonist of human NK-3 receptor Ki44 nM that effectively crosses the blood-brain barrier |
| CSN22503 | Saredutant | 142001-63-6 | Saredutant is a selective NK2 receptor antagonist. |
| CSN19715 | Rolapitant | 552292-08-7 | Rolapitant inhibits CYP2D6 breast cancer resistance protein BCRP and Neurokinin NK1 Receptor |
| CSN16098 | Rolapitant HCl H2O | 914462-92-3 | Rolapitant HCl H2O is a long-acting selective and competitive NK-1 receptor antagonist |
| CSN18026 | NKP608 | 177707-12-9 | NKP608 is a non-peptidic derivative of 4-aminopiperidine which acts as a selective specific and potent antagonist at the neurokinin-1 NK-1 receptor both in vitro IC5026 nM and in vivo |
| CSN16120 | Netupitant | 290297-26-6 | Netupitant a potent and highly selective NK1 receptor antagonist with Ki of 095 nM |
| CSN19286 | MLE4901 | 941690-55-7 | MLE4901 is an antagonist of Neurokinin 3 Receptor and a potential drug for Polycystic ovary syndrome and menopausal hot flushes |
| CSN22464 | MEN 15596 | 522664-63-7 | MEN 15596 is a potent and selective tachykinin NK2 receptor antagonist with a pKi of 101 |
| CSN17887 | Maropitant | 147116-67-4 | Maropitant is a neurokinin NK1 receptor antagonist |
| CSN18008 | Fosaprepitant | 172673-20-0 | Fosaprepitant is a neurokinin-1 receptor antagonist for the prevention of chemotherapy-induced nausea and vomiting |
| CSN12336 | Fosaprepitant Dimeglumine | 265121-04-8 | Fosaprepitant Dimeglumine is a prodrug for aprepitant which is a selective and high-affinity antagonist of NK1 receptor. |
| CSN10324 | Aprepitant | 170729-80-3 | Aprepitant is a selective and high-affinity neurokinin-1 receptor antagonist with IC50 of 0.1 nM. |
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