|α-Cyano-4-hydroxycinnamic acid is a MCT inhibitor with antitumoral and antiangiogenic activity.
|SR13800 is a cell-permeable inhibitor of monocarboxylate transporter 1 (MCT1).
|BAY-8002 is a potent MCT Inhibitor with IC50 value of 8nM for inhibition of L-lactate uptake.
|AZD3965 is a potent selective and orally available monocarboxylate transporter 1 MCT1 inhibitor with a binding affinity of 16 nM
|AR-C155858 is an inhibitor of the monocarboxylate transporters MCTs MCT1 and MCT2 Ki values are 23 and 10 nM respectively and exhibits no activity at MCT4
|7ACC2 is a potent MCT inhibitor with IC50 of 11 nM for inhibition of 14C-lactate influx for antitumor treatment targeting lactate transport in cancer cells
|7ACC1 selectively interfere with lactate fluxes in the lactate-rich tumor microenvironment and inhibits lactate influx but not efflux in tumor cells expressing MCT1 and MCT4 transporters.