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MCT

MCT

Cat. No. Product Name CAS No. Information
CSN22752 α-Cyano-4-hydroxycinnamic acid   28166-41-8 α-Cyano-4-hydroxycinnamic acid is a MCT inhibitor with antitumoral and antiangiogenic activity.
CSN23125 MCT1-IN-2 227321-12-2 SR13800 is a cell-permeable inhibitor of monocarboxylate transporter 1 (MCT1).
CSN23771 BAY-8002 724440-27-1 BAY-8002 is a potent MCT Inhibitor with IC50 value of 8nM for inhibition of L-lactate uptake.
CSN13789 AZD3965 1448671-31-5 AZD3965 is a potent selective and orally available monocarboxylate transporter 1 MCT1 inhibitor with a binding affinity of 16 nM
CSN15986 AR-C155858 496791-37-8 AR-C155858 is an inhibitor of the monocarboxylate transporters MCTs MCT1 and MCT2 Ki values are 23 and 10 nM respectively and exhibits no activity at MCT4
CSN17889 7ACC2 1472624-85-3 7ACC2 is a potent MCT inhibitor with IC50 of 11 nM for inhibition of 14C-lactate influx for antitumor treatment targeting lactate transport in cancer cells
CSN12098 7ACC1 50995-74-9 7ACC1 selectively interfere with lactate fluxes in the lactate-rich tumor microenvironment and inhibits lactate influx but not efflux in tumor cells expressing MCT1 and MCT4 transporters.
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