MCT
Cat. No. | Product Name | CAS No. | Information |
---|---|---|---|
CSN22752 | α-Cyano-4-hydroxycinnamic acid | 28166-41-8 | α-Cyano-4-hydroxycinnamic acid is a MCT inhibitor with antitumoral and antiangiogenic activity. |
CSN23125 | MCT1-IN-2 | 227321-12-2 | SR13800 is a cell-permeable inhibitor of monocarboxylate transporter 1 (MCT1). |
CSN23771 | BAY-8002 | 724440-27-1 | BAY-8002 is a potent MCT Inhibitor with IC50 value of 8nM for inhibition of L-lactate uptake. |
CSN13789 | AZD3965 | 1448671-31-5 | AZD3965 is a potent selective and orally available monocarboxylate transporter 1 MCT1 inhibitor with a binding affinity of 16 nM |
CSN15986 | AR-C155858 | 496791-37-8 | AR-C155858 is an inhibitor of the monocarboxylate transporters MCTs MCT1 and MCT2 Ki values are 23 and 10 nM respectively and exhibits no activity at MCT4 |
CSN17889 | 7ACC2 | 1472624-85-3 | 7ACC2 is a potent MCT inhibitor with IC50 of 11 nM for inhibition of 14C-lactate influx for antitumor treatment targeting lactate transport in cancer cells |
CSN12098 | 7ACC1 | 50995-74-9 | 7ACC1 selectively interfere with lactate fluxes in the lactate-rich tumor microenvironment and inhibits lactate influx but not efflux in tumor cells expressing MCT1 and MCT4 transporters. |