Kainate receptors, or kainic acid receptors (KARs), are ionotropic receptors that respond to the neurotransmitter glutamate.
Cat. No. | Product Name | CAS No. | Information |
---|---|---|---|
CSN23175 | UBP-282 | 544697-47-4 | UBP-282 is an α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) and kainate receptor antagonist. |
CSN24615 | UBP310 | 902464-46-4 | UBP 310 is an antagonist of GluK1 (formerly GLUK5) kainate receptor with IC50 of 130 nM. |
CSN24617 | UBP 302 | 745055-91-8 | UBP 302 is a potent and selective GluK1 (formally GluR5)-subunit containing kainate receptor antagonist with KD of 402 nM. |
CSN20167 | Selurampanel | 912574-69-7 | Selurampanel is a competitive AMPAkainate receptor antagonist drug for epilepsy |
CSN11876 | (S)-Willardiine | 21416-43-3 | S-Willardiine is a potent agonist of AMPAkainate receptors with EC50 of 448 M |
CSN29466 | (2S,3S,4S)-4-((R,2Z,4E)-6-carboxyhepta-2,4-dien-2-yl)-3-(carboxymethyl)pyrrolidine-2-carboxylic acid | 14277-97-5 | Potent and selective kainate agonist. |
CSN16600 | L-Theanine | 3081-61-6 | L-theanine is an amino acid found most commonly in tea leaves and binds to ionotropic glutamate receptors in the micromolar range including the AMPA and kainate receptors and to a lesser extent the NMDA receptor |
CSN19846 | Kainic acid | 487-79-6 | Kainic acid is a selective agonist at kainate receptors Potent excitant and neurotoxin |
CSN24616 | ATPA | 140158-50-5 | ATPA is a selective and potent GluK1 kainate receptor agonist with Ki of 4.3 nM. |