Histone Acetyltransferase
Cat. No. | Product Name | CAS No. | Information |
---|---|---|---|
CSN22467 | WM-1119 | 2055397-28-7 | WM-1119 is an inhibitor of KAT6A (MOZ) which is a member of histone acetyltransferases with IC50 of 0.051 μM. |
CSN28764 | WM-3835 | 2229025-70-9 | WM 3835 is a highly potent HBO1 inhibitor and demonstrate its mode of activity as a competitive analogue of acetyl-CoA. It reduced H3K14ac levels and inhibits growth and viability of acyte myeloid leukemia cell lines in vitro. |
CSN17961 | Remodelin hydrobromide | 1622921-15-6 | Remodelin hydrobromide is a selective inhibitor of acetyl-transferase protein NAT10 |
CSN24831 | NU9056 | 1450644-28-6 | NU9056 is a selective Tip60 histone acetyltransferase inhibitor with IC50 values of 2μM, 60μM and 36μM for KAT5, p300 and pCAF, respectively. |
CSN27616 | NEO2734 | 2081072-29-7 | NEO2734 is an orally dual p300/CBP and BET bromodomain inhibitor with IC50 values of <30 nM for both p300/CBP and BET bromodomains. |
CSN21259 | WM-8014 | 2055397-18-5 | MOZ-IN-3 is an inhibitor of MOZ a member of histone acetyltransferases with an IC50 of 55 nM |
CSN22468 | MOZ-IN-2 | 2055397-88-9 | MOZ-IN-2 is an inhibitor of protein MOZ a member of histone acetyltransferases with an IC50 of 125 M |
CSN16635 | MG 149 | 1243583-85-8 | MG149 is a potent histone acetyltransferase inhibitor with IC50 of 74 M and 47 M for Tip60 and MOFrespectively |
CSN12696 | ICG001 | 868774-16-7 | ICG-001 is an inhibitor of β-catenin/cyclic AMP responsive element binding protein binding protein (CBP)-mediated transcription with IC50 of 3 µM. |
CSN16033 | ICG-001 | 780757-88-2 | ICG 001 can bind to element-binding protein (CREB)-binding protein (CBP) with IC50 of 3 M and antagonize the Wnt-cateninTCF-mediated transcription. |
CSN16945 | Histone Acetyltransferase Inhibitor II | 932749-62-7 | Histone Acetyltransferase inhibitor II insulin producing cells capable of secreting blood glucose regulating hormones specially insulin in response to physiological signals method of production of said cells and uses thereof |
CSN22203 | HAT-IN-1 | 1889281-94-0 | HAT-IN-1 is an inhibitor of HAT used in the research of cancer |
CSN28526 | GSK699 | 2260944-68-9 | GSK699 is a potent, cell penetrant PCAF/GCN5 PROTAC. |
CSN22422 | GSK 4027 | 2079896-25-4 | GSK 4027 is a chemical probe for the PCAFGCN5 bromodomain with an pIC50 of 7.40.11 for PCAF in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. |
CSN19424 | Curcumin | 458-37-7 | Curcumin is a natural phenolic compound with impressive antioxidant properties. |
CSN15965 | CPTH2 | 357649-93-5 | CPTH2 is a histone acetyltransferase (HAT) inhibitor modulating the Gcn5 network where HATs act as transcriptional coactivators. |
CSN12895 | Procyanidin B3 | 23567-23-9 | Cercosporamide is a potent and selective Mnk inhibitor and an orally bioavailable antifungal agent suppresses phosphorylation of eIF4E and exhibits antileukemic effects |
CSN16094 | C646 | 328968-36-1 | C646 is a selective inhibitor of histone acetyltransferase p300 with Ki of 400 nM |
CSN13640 | Anacardic Acid | 16611-84-0 | Anacardic acid is a potent inhibitor of p300 and p300CBP-associated factor histone acetyltranferases which also has antibacterial activity antimicrobial activityprostaglandin synthase inhibition and tyrosinase and lipoxygenase inhibition |
CSN22658 | A-485 | 1889279-16-6 | A 485 is a potent and selective p300/CREB-binding protein (CBP) HAT domain inhibitor with IC50 of 2.6 and 9.8 nM for the CBP-bromodomain HAT-C/H3 (BHC) and p300-BHC domains, respectively. |
CSN32736 | PF-9363 | 2569009-58-9 | |
CSN32741 | NiCur | 63476-70-0 | |
CSN40845 | Garcinol | 78824-30-3 |