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Histamine Receptor

Histamine Receptor

Cat. No. Product Name CAS No. Information
CSN20447 VUF 10460   1028327-66-3 VUF 10460 is a selective agonist of histamine H4 receptor with pKi of 8.22.
CSN21874 Tritoqualine 14504-73-5 Tritoqualine is a histamine H1 antagonist.
CSN12374 Tripelennamine HCl   154-69-8 Tripelennamine HCl is an antagonist of H1-receptor that used as a psychoactive drug with antipruritic activity.
CSN17265 Setastine 64294-95-7 Setastine is an antihistamine used to treat allergies and rhinitis.
CSN21826 Rocastine 91833-77-1 Rocastine is a selective antagonist of nonsedative H1 antagonist for antihistamines.
CSN21315 Pirolate 55149-05-8 Pirolate (CP-32,387) is an antihistamine drug with a tricyclic chemical structure which was patented as an antiallergen.
CSN11691 Pheniramine Maleate   132-20-7 Pheniramine maleate can acts as an antihistamine and vasoconstrictor.
CSN11668 Pemirolast Potassium   100299-08-9 Pemirolast potassium is an antagonist of histamine H1 and mast cell stabilizer with antiallergic effect.
CSN11604 Olopatadine HCl   140462-76-6 Olopatadine HCl can block the release of histamine (IC50 = 559 µM) and stabilize mast cell.
CSN11591 Nylidrin HCl 849-55-8 Nylidrin HCl was an effective inhibitor of IgE-mediated release of histamine from passively sensitized rat peritoneal mast cells and human basophils, and of IgG1-mediated release of histamine from passively sensitized guinea pig lung slices.
CSN11565 Nizatidine   76963-41-2 Nizatidine is an antagonist of histamine H2 receptor that can inhibit the secretion of gastric acid.
CSN21744 Niperotidine 84845-75-0 Niperotidine is an antagonist of histamine H2-receptor.
CSN11531 Nedocromil 69049-73-6 Nedocromil is an inhaled anti-inflammatory agent for the preventive management of asthma.
CSN21105 N-omega-Acetylhistamine 673-49-4 N-acetylhistamine is a histamine metabolite. N-acetylhistamine can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.
CSN12482 Mizolastine 108612-45-9 Mizolastine is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions.
CSN17435 Mizolastine 2HCl 1056596-82-7 Mizolastine 2HCl is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions.
CSN11382 Mequitazine 29216-28-2 Mequitazine is a potent, nonsedative and long-acting histamine H1 antagonist.
CSN21134 Mebhydrolin 524-81-2 Mebhydrolin is a specific histamine H1 receptor antagonist.
CSN12956 Loratadine   79794-75-5 Loratadine is an inverse agonist of peripheral histamine H1-receptor with IC50 of 32 M.
CSN11321 Lodoxamide Tromethamine   63610-09-3 Lodoxamide tromethamine is used as an ophthalmic solution that specially applying to the eye.
CSN13135 Levodropropizine 99291-25-5 Levodropropizine is a histamine receptor inhibitor, and is an effective and very well tolerated peripheral antitussive drug.
CSN19403 Ketotifen Fumarate 34580-14-8 Ketotifen fumarate is a noncompetitive H1 receptor antagonist and mast cell stabilizer that is used to treat asthma.
CSN16759 JNJ-7777120   459168-41-3 JNJ-7777120 is a selective antagonist of histamine-4 receptor (H4R) with Ki of 4 1 nM.
CSN22061 JNJ-39758979 1046447-90-8 JNJ-39758979 is a selective, high-affinity histamine H4 receptor antagonist with Ki of 12.5 nM.
CSN11177 Hydroxyzine Pamoate 10246-75-0 Hydroxyzine pamoate is a histamine H1-receptor antagonist.
CSN17063 Hydroxyzine 68-88-2 Hydroxyzine is a histamine H1-receptor antagonist.
CSN21410 H3R-IN-1 HCl N/A H3R-IN-1 HCl is a histamine receptor 3 (H3R) inverse agonist.
CSN22023 FRG8701 108498-50-6 FRG-8701 is a new Histamine H2-receptor antagonist with IC50 of ranging from 0.25 to 0.43 μM.
CSN21734 FPL59360 85118-44-1 FPL59360, a anti-asthmatic compound, is histamine I receptor antagonist that prevents exercise-induced asthma.
CSN11010 Fexofenadine 83799-24-0 Fexofenadine is an antihistamine pharmaceutical drug used in the treatment of allergy symptoms, such as hay fever, nasal congestion, and urticaria.
CSN19386 Epinastine   80012-43-7 Epinastine is mast cell stabilizer and antihistamine that is used to treat allergic conjunctivitis.
CSN10917 Epinastine HCl 108929-04-0 Epinastine HCl is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.
CSN10883 Ebastine   90729-43-4 Ebastine is a selective H1-histamine receptor antagonist.
CSN10775 Desloratadine   100643-71-8 Desloratadine is an antagonist of histamine H1 receptor that is used to treat allergies.
CSN13624 Decloxizine 2HCl 13073-96-6 Decloxizine 2HCl is a histamine 1 receptor antagonist.
CSN10076 Chlorpheniramine Maleate   113-92-8 Chlorpheniramine maleate is an antagonist of histamine H1 receptor with IC50 of 12 nM.
CSN12995 Cetirizine 2HCl   83881-52-1 Cetirizine 2HCl, a metabolite of hydroxyzine, is racemic selective and inverse agonist of H1 receptor used in the treatment of allergies and hay fever.
CSN22167 BMY-25271 78441-82-4 BMY-25271 is a histamine H2 receptor antagonist.
CSN16768 Azelastine 58581-89-8 Azelastine is a potent, second-generation, selective, histamine antagonist.
CSN16787 Azelastine HCl   79307-93-0 Azelastine HCl is a selective antagonist of histamine receptor used in the treatment of rhinitis.
CSN21455 Acrivastine 87848-99-5 Acrivastine, an H1-receptor antagonist, is a second-generation antihistamine.
CSN10156 6-Methoxyluteolin 520-11-6 6-Methoxyluteolin is a natural product isolated and purified from the flower of Chrysanthemum zawadskii var. latilobum with antioxidant activity and is also a potent inhibitor of histamine release and calcium influx via down-regulation of the FcRI chain.
CSN21849 Tazifylline 79712-55-3 (±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.
CSN14575 Marmin 14957-38-1
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