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Histamine Receptor

Histamine Receptor

Cat. No. Product Name CAS No. Information
CSN20447 VUF 10460   1028327-66-3 VUF 10460 is a selective agonist of histamine H4 receptor with pKi of 8.22.
CSN21874 Tritoqualine 14504-73-5 Tritoqualine is a histamine H1 antagonist.
CSN24558 TC 1698 dihydrochloride 787587-06-8 TC 1698 dihydrochloride is a selective nicotinic α7 receptor agonist with EC50 of 440 nM.
CSN17265 Setastine 64294-95-7 Setastine is an antihistamine used to treat allergies and rhinitis.
CSN24554 SEN 12333 874450-44-9 SEN 12333 is a selective agonist of α7 nicotinic acetylcholine receptor (nAChR) with EC50 and Ki of 1.6 μM, 260 nM in rat. It also displays functional antagonism at histamine H3 receptors (IC50 = 103 nM).
CSN12316 Rupatadin Fumarate   182349-12-8 Rupatadine fumarate is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 nM and 102 nM, respectively.
CSN13086 Roxatidine Acetate HCl   93793-83-0 Roxatidine acetate HCl is a slective antagonist of histamin H2 receptor.
CSN21826 Rocastine 91833-77-1 Rocastine is a selective antagonist of nonsedative H1 antagonist for antihistamines.
CSN21315 Pirolate 55149-05-8 Pirolate (CP-32,387) is an antihistamine drug with a tricyclic chemical structure which was patented as an antiallergen.
CSN11668 Pemirolast Potassium   100299-08-9 Pemirolast potassium is an antagonist of histamine H1 and mast cell stabilizer with antiallergic effect.
CSN11604 Olopatadine HCl   140462-76-6 Olopatadine HCl can block the release of histamine (IC50 = 559 µM) and stabilize mast cell.
CSN11591 Nylidrin HCl 849-55-8 Nylidrin HCl was an effective inhibitor of IgE-mediated release of histamine from passively sensitized rat peritoneal mast cells and human basophils, and of IgG1-mediated release of histamine from passively sensitized guinea pig lung slices.
CSN21744 Niperotidine 84845-75-0 Niperotidine is an antagonist of histamine H2-receptor.
CSN11531 Nedocromil 69049-73-6 Nedocromil is an inhaled anti-inflammatory agent for the preventive management of asthma.
CSN21105 N-omega-Acetylhistamine 673-49-4 N-acetylhistamine is a histamine metabolite. N-acetylhistamine can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.
CSN12482 Mizolastine 108612-45-9 Mizolastine is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions.
CSN17435 Mizolastine 2HCl 1056596-82-7 Mizolastine 2HCl is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions.
CSN11382 Mequitazine 29216-28-2 Mequitazine is a potent, nonsedative and long-acting histamine H1 antagonist.
CSN21134 Mebhydrolin 524-81-2 Mebhydrolin is a specific histamine H1 receptor antagonist.
CSN14575 Marmin 14957-38-1 Marmin, a natural product isolated and purified from the herbs of Citrus maxima with potent anti-ulcer, antibacterial, fungicidal, and algicidal properties, can inhibit contraction of the guinea-pig tracheal smooth muscle, especially by interfering histamine receptor, inhibiting the histamine release from mast, inhibiting intracellular Ca2+ release from the intracellular store and the Ca2+ influx through voltage-dependent Ca2+ channels, is potential to develop as antihistamine agents, especially as histamine H1 receptor antagonists by interacting with amino acid residues, Asp107, Lys179, Lys191, Asn198, and Trp428 of histamine H1 receptor, shows a cell-growth inhibitory effect against L1210 and K562 in vitro.
CSN12956 Loratadine   79794-75-5 Loratadine is an inverse agonist of peripheral histamine H1-receptor with IC50 of 32 M.
CSN25565 LML-134 1542135-76-1 LML134 is an orally active and high selective Histamine 3 receptor (H3R) inverse agonist with Kis of 0.3 nM and 12 nM for hH3R cAMP and hH3R bdg. LML134 penetrates the brain rapidly, leading to high H3R occupancy, and disengages its target with a fast kinetic profile. LML134 has the potential for excessive sleep disorders.
CSN13135 Levodropropizine 99291-25-5 Levodropropizine is a histamine receptor inhibitor, and is an effective and very well tolerated peripheral antitussive drug.
CSN16072 Levocetirizine 2HCl 130018-87-0 Levocetirizine 2HCl is a third-generation non-sedative antihistamine, developed from the second-generation antihistamine cetirizine.
CSN19403 Ketotifen Fumarate 34580-14-8 Ketotifen fumarate is a noncompetitive H1 receptor antagonist and mast cell stabilizer that is used to treat asthma.
CSN16759 JNJ-7777120   459168-41-3 JNJ-7777120 is a selective antagonist of histamine-4 receptor (H4R) with Ki of 4 1 nM.
CSN25273 JNJ-5207852 398473-34-2 JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
CSN22061 JNJ-39758979 1046447-90-8 JNJ-39758979 is a selective, high-affinity histamine H4 receptor antagonist with Ki of 12.5 nM.
CSN17063 Hydroxyzine 68-88-2 Hydroxyzine is a histamine H1-receptor antagonist.
CSN21410 H3R-IN-1 HCl N/A H3R-IN-1 HCl is a histamine receptor 3 (H3R) inverse agonist.
CSN22023 FRG8701 108498-50-6 FRG-8701 is a new Histamine H2-receptor antagonist with IC50 of ranging from 0.25 to 0.43 μM.
CSN21734 FPL59360 85118-44-1 FPL59360, a anti-asthmatic compound, is histamine I receptor antagonist that prevents exercise-induced asthma.
CSN19386 Epinastine   80012-43-7 Epinastine is mast cell stabilizer and antihistamine that is used to treat allergic conjunctivitis.
CSN24500 Emedastine 87233-61-2 Emedastine is a potent, high affinity histamine H1-receptor-selective antagonist with Ki of 1.3 ±0.1 nM for H1-receptors while considerably weaker at H2- (Ki = 49,067 ± 11,113 nM) and H3-receptors (Ki = 12,430 ± 1,282 nM).
CSN13624 Decloxizine 2HCl 13073-96-6 Decloxizine 2HCl is a histamine 1 receptor antagonist.
CSN22573 Cyclizine 2HCl 5897-18-7 Cyclizine is a histamine H1 receptor antagonist of the piperazine class.
CSN10076 Chlorpheniramine Maleate   113-92-8 Chlorpheniramine maleate is an antagonist of histamine H1 receptor with IC50 of 12 nM.
CSN23808 Chlorcyclizine HCl 14362-31-3 Chlorcyclizine hydrochloride is a histamine H1 antagonist.
CSN12995 Cetirizine 2HCl   83881-52-1 Cetirizine 2HCl, a metabolite of hydroxyzine, is racemic selective and inverse agonist of H1 receptor used in the treatment of allergies and hay fever.
CSN25269 Bromazine HCl 1808-12-4 Bromazine hydrochloride is an antagonist of histamine H1 receptor.
CSN22167 BMY-25271 78441-82-4 BMY-25271 is a histamine H2 receptor antagonist.
CSN25225 Betahistine 5638-76-6 Betahistine is a histamine analog and H1 receptor agonist.
CSN16768 Azelastine 58581-89-8 Azelastine is a potent, second-generation, selective, histamine antagonist.
CSN16787 Azelastine HCl   79307-93-0 Azelastine HCl is a selective antagonist of histamine receptor used in the treatment of rhinitis.
CSN24556 AR-R 17779 hydrochloride 178419-42-6 AR-R 17779 hydrochloride is a selective alpha7 nicotinic agonist with Ki value of 190 nM for rat.
CSN21455 Acrivastine 87848-99-5 Acrivastine, an H1-receptor antagonist, is a second-generation antihistamine.
CSN24555 A 844606 861119-08-6 A 844606 is a selective α7 nicotinic acetylcholine receptor (nAChR) partial agonist with EC50 values are 1.4 and 2.2 μM at human and rat receptors, respectively.
CSN10156 6-Methoxyluteolin 520-11-6 6-Methoxyluteolin is a natural product isolated and purified from the flower of Chrysanthemum zawadskii var. latilobum with antioxidant activity and is also a potent inhibitor of histamine release and calcium influx via down-regulation of the FcRI chain.
CSN21849 Tazifylline 79712-55-3 (±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.
CSN24562 (S)-(+)-Dimethindene maleate 136152-65-3 (S)-(+)-Dimethindene maleate is a subtype-selective M2 muscarinic receptor antagonist with pKi of 7.78 and is also a H1 histamine receptor antagonist with pKi of 7.48.
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