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Histamine Receptor

Histamine Receptor

Cat. No. Product Name CAS No. Information
CSN21826 Rocastine 91833-77-1 Rocastine is a selective antagonist of nonsedative H1 antagonist for antihistamines.
CSN13516 Ranitidine HCl   66357-59-3 Ranitidine HCl is an antagonist of histamine H2-receptor that can inhibit stomach acid production.
CSN26180 PU-02   313984-77-9 PU-02 is an antagonist of serotonin (5-HT) receptor subtype 5-HT3.
CSN17113 Promethazine HCl   58-33-3 Promethazine HCl is the effective antagonist of the H1 receptor and moderate antagonist of mACh receptor.
CSN21315 Pirolate 55149-05-8 Pirolate (CP-32,387) is an antihistamine drug with a tricyclic chemical structure which was patented as an antiallergen.
CSN21744 Niperotidine 84845-75-0 Niperotidine is an antagonist of histamine H2-receptor.
CSN11531 Nedocromil 69049-73-6 Nedocromil is an inhaled anti-inflammatory agent for the preventive management of asthma.
CSN21105 N-omega-Acetylhistamine 673-49-4 N-acetylhistamine is a histamine metabolite. N-acetylhistamine can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.
CSN11809 Mepyramine Maleate   59-33-6 Mepyramine maleate is an antagonist of histamine H1 receptor.
CSN21134 Mebhydrolin 524-81-2 Mebhydrolin is a specific histamine H1 receptor antagonist.
CSN14575 Marmin 14957-38-1 Marmin, a natural product isolated and purified from the herbs of Citrus maxima with potent anti-ulcer, antibacterial, fungicidal, and algicidal properties, can inhibit contraction of the guinea-pig tracheal smooth muscle, especially by interfering histamine receptor, inhibiting the histamine release from mast, inhibiting intracellular Ca2+ release from the intracellular store and the Ca2+ influx through voltage-dependent Ca2+ channels, is potential to develop as antihistamine agents, especially as histamine H1 receptor antagonists by interacting with amino acid residues, Asp107, Lys179, Lys191, Asn198, and Trp428 of histamine H1 receptor, shows a cell-growth inhibitory effect against L1210 and K562 in vitro.
CSN19403 Ketotifen Fumarate 34580-14-8 Ketotifen fumarate is a noncompetitive H1 receptor antagonist and mast cell stabilizer that is used to treat asthma.
CSN25273 JNJ-5207852 398473-34-2 JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
CSN17063 Hydroxyzine 68-88-2 Hydroxyzine is a histamine H1-receptor antagonist.
CSN16192 Hydroxyzine 2HCl   2192-20-3 Hydroxyzine 2HCl is an antagonist of histamine H1-receptor that inhibits the binding of [3H]pyrilamine and [3H]desloratadine to histamine H1 receptor with IC50s of 10 nM and 19 nM.
CSN22023 FRG8701 108498-50-6 FRG-8701 is a new Histamine H2-receptor antagonist with IC50 of ranging from 0.25 to 0.43 μM.
CSN21734 FPL59360 85118-44-1 FPL59360, a anti-asthmatic compound, is histamine I receptor antagonist that prevents exercise-induced asthma.
CSN12462 Fexofenadine HCl 153439-40-8 Fexofenadine inhibits histamine H1 receptor with IC50 of 246 nM.
CSN19386 Epinastine   80012-43-7 Epinastine is mast cell stabilizer and antihistamine that is used to treat allergic conjunctivitis.
CSN24500 Emedastine 87233-61-2 Emedastine is a potent, high affinity histamine H1-receptor-selective antagonist with Ki of 1.3 ±0.1 nM for H1-receptors while considerably weaker at H2- (Ki = 49,067 ± 11,113 nM) and H3-receptors (Ki = 12,430 ± 1,282 nM).
CSN22573 Cyclizine 2HCl 5897-18-7 Cyclizine is a histamine H1 receptor antagonist of the piperazine class.
CSN20584 Clobenpropit Dihydrobromide 145231-35-2 Clobenpropit hydrobromide is a selective histamine H3 receptor antagonist that crosses the blood-brain barrier, inhibiting histamine binding in rat brain.
CSN15935 Ciproxifan Maleate 184025-19-2 Ciproxifan maleate is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at other receptor subtypes.
CSN12549 Cinnarizine   298-57-7 Cinnarizine, an antihistamine, can block calcium channel and promote cerebral blood flow. It is used to treat post-trauma cerebral symptoms and cerebral arteriosclerosis.
CSN23808 Chlorcyclizine HCl 14362-31-3 Chlorcyclizine hydrochloride is a histamine H1 antagonist.
CSN25269 Bromazine HCl 1808-12-4 Bromazine hydrochloride is an antagonist of histamine H1 receptor.
CSN22167 BMY-25271 78441-82-4 BMY-25271 is a histamine H2 receptor antagonist.
CSN16768 Azelastine 58581-89-8 Azelastine is a potent, second-generation, selective, histamine antagonist.
CSN16787 Azelastine HCl   79307-93-0 Azelastine HCl is a selective antagonist of histamine receptor used in the treatment of rhinitis.
CSN21455 Acrivastine 87848-99-5 Acrivastine, an H1-receptor antagonist, is a second-generation antihistamine.
CSN10156 6-Methoxyluteolin 520-11-6 6-Methoxyluteolin is a natural product isolated and purified from the flower of Chrysanthemum zawadskii var. latilobum with antioxidant activity and is also a potent inhibitor of histamine release and calcium influx via down-regulation of the FcRI chain.
CSN21849 Tazifylline 79712-55-3 (±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.
CSN24562 (S)-(+)-Dimethindene maleate 136152-65-3 (S)-(+)-Dimethindene maleate is a subtype-selective M2 muscarinic receptor antagonist with pKi of 7.78 and is also a H1 histamine receptor antagonist with pKi of 7.48.
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