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Histamine Receptor

Histamine Receptor

Cat. No. Product Name CAS No. Information
CSN20447 VUF 10460   1028327-66-3 VUF 10460 is a selective agonist of histamine H4 receptor with pKi of 8.22.
CSN12374 Tripelennamine HCl   154-69-8 Tripelennamine hydrochloride is an antagonist of H1-receptor that used as a psychoactive drug with antipruritic activity.
CSN17265 Setastine 64294-95-7 Setastine is an antihistamine used to treat allergies and rhinitis.
CSN12316 Rupatadin Fumarate   182349-12-8 Rupatadine fumarate is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 nM and 102 nM, respectively.
CSN13086 Roxatidine Acetate HCl   93793-83-0 Roxatidine acetate hydrochloride is a slective antagonist of histamin H2 receptor.
CSN21315 Pirolate 55149-05-8 Pirolate (CP-32,387) is an antihistamine drug with a tricyclic chemical structure which was patented as an antiallergen.
CSN11691 Pheniramine Maleate   132-20-7 Pheniramine maleate can acts as an antihistamine and vasoconstrictor.
CSN11668 Pemirolast Potassium   100299-08-9 Pemirolast potassium is an antagonist of histamine H1 and mast cell stabilizer with antiallergic effect.
CSN11604 Olopatadine HCl   140462-76-6 Olopatadine hydrochloride can block the release of histamine (IC50 559 M) and stabilize mast cell.
CSN11565 Nizatidine   76963-41-2 Nizatidine is an antagonist of histamine H2 receptor that can inhibit the secretion of gastric acid.
CSN21105 N-omega-Acetylhistamine 673-49-4 N-acetylhistamine is a histamine metabolite. N-acetylhistamine can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.
CSN12482 Mizolastine 108612-45-9 Mizolastine is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions.
CSN17435 Mizolastine 2HCl 1056596-82-7 Mizolastine dihydrochloride is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions.
CSN11382 Mequitazine 29216-28-2 Mequitazine is a potent, nonsedative and long-acting histamine H1 antagonist.
CSN16435 Mebhydrolin Napadisylate   6153-33-9 Mebhydrolin is an antihistamine that used for symptomatic relief of allergic symptoms.
CSN21134 Mebhydrolin 524-81-2 Mebhydrolin is a specific histamine H1 receptor antagonist.
CSN12956 Loratadine   79794-75-5 Loratadine is an inverse agonist of peripheral histamine H1-receptor with IC50 of 32 M.
CSN11321 Lodoxamide Tromethamine   63610-09-3 Lodoxamide tromethamine is used as an ophthalmic solution that specially applying to the eye.
CSN13135 Levodropropizine 99291-25-5 Levodropropizine is a histamine receptor inhibitor, and is an effective and very well tolerated peripheral antitussive drug.
CSN16072 Levocetirizine 2HCl 130018-87-0 Levocetirizine dihydrochloride is a third-generation non-sedative antihistamine, developed from the second-generation antihistamine cetirizine.
CSN19403 Ketotifen Fumarate 34580-14-8 Ketotifen fumarate is a noncompetitive H1 receptor antagonist and mast cell stabilizer that is used to treat asthma.
CSN16759 JNJ-7777120   459168-41-3 JNJ-7777120 is a selective antagonist of histamine-4 receptor (H4R) with Ki of 4 1 nM.
CSN11177 Hydroxyzine Pamoate 10246-75-0 Hydroxyzine pamoate is a histamine H1-receptor antagonist.
CSN17063 Hydroxyzine 68-88-2 Hydroxyzine is a histamine H1-receptor antagonist.
CSN16192 Hydroxyzine 2HCl   2192-20-3 Hydroxyzine dihydrochloride is an antagonist of histamine H1-receptor that inhibits the binding of 3Hpyrilamine and 3Hdesloratadine to histamine H1 receptor with IC50s of 10 nM and 19 nM.
CSN21410 H3R-IN-1 HCl N/A H3R-IN-1 HCl is a histamine receptor 3 (H3R) inverse agonist.
CSN11010 Fexofenadine 83799-24-0 Fexofenadine is an antihistamine pharmaceutical drug used in the treatment of allergy symptoms, such as hay fever, nasal congestion, and urticaria.
CSN19386 Epinastine   80012-43-7 Epinastine is mast cell stabilizer and antihistamine that is used to treat allergic conjunctivitis.
CSN10917 Epinastine HCl 108929-04-0 Epinastine hydrochloride is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.
CSN10884 Ebrotidine 100981-43-9 Ebrotidine is a competitive H2-receptor antagonist (Ki 127.5 nM) with a potent antisecretory activity and evidenced gastroprotection.
CSN10883 Ebastine   90729-43-4 Ebastine is a selective H1-histamine receptor antagonist.
CSN10864 Doxylamine succinate salt   562-10-7 Doxylamine is an antihistamine which inhibits histamine H1 receptors. It can be used as a short-term sedative and anticholinergic agent.
CSN16168 Diphenhydramine HCl   147-24-0 Diphenhydramine hydrochloride is a histamine H1 antagonist that is used as an antiemetic and antitussive.
CSN10783 Dexchlorpheniramine Maleate 2438-32-6 Dexchlorpheniramine maleate is an antihistamine, with anticholinergic properties, used to treat allergic conditions.
CSN10775 Desloratadine   100643-71-8 Desloratadine is an antagonist of histamine H1 receptor that is used to treat allergies.
CSN10757 Decloxizine 3733-63-9 Decloxizine is a histamine 1 receptor antagonist.
CSN13624 Decloxizine 2HCl 13073-96-6 Decloxizine dihydrochloride is a histamine 1 receptor antagonist.
CSN10076 Chlorpheniramine Maleate   113-92-8 Chlorpheniramine maleate is an antagonist of histamine H1 receptor with IC50 of 12 nM.
CSN10600 Cetirizine 83881-51-0 Cetirizine, a second-generation antihistamine, is a major metabolite of hydroxyzine, and a racemic selective H1 receptor inverse agonist used in the treatment of allergies, hay fever, angioedema, and urticaria.
CSN12995 Cetirizine 2HCl   83881-52-1 Cetirizine dihydrochloride, a metabolite of hydroxyzine, is racemic selective and inverse agonist of H1 receptor used in the treatment of allergies and hay fever.
CSN10548 Carbinoxamine Maleate   3505-38-2 Carbinoxamine maleate is a blocker of histamine-H1 receptor with antihistamine and anticholinergic effects.
CSN10492 Brompheniramine Maleate 980-71-2 Brompheniramine maleate is an antagonist of histamine H1 receptors.
CSN22167 BMY-25271 78441-82-4 BMY-25271 is a histamine H2 receptor antagonist.
CSN10402 Bilastine 202189-78-4 Bilastine selectively antagonizes histamine H1 receptor and it is used to treat allergic rhinoconjunctivitis and urticaria.
CSN10415 Bepotastine Besilate   190786-44-8 Bepotastine besilate is a selective antagonist of histamine 1 (H1) receptor with pIC50 of 5.7.
CSN16768 Azelastine 58581-89-8 Azelastine is a potent, second-generation, selective, histamine antagonist.
CSN16787 Azelastine HCl   79307-93-0 Azelastine hydrochloride is a selective antagonist of histamine receptor used in the treatment of rhinitis.
CSN10365 Azatadine 3964-81-6 Azatadine is an histamine and cholinergic inhibitor with IC50 of 6.5 nM and 10 nM, respectively.
CSN10364 Azatadine Dimaleate   3978-86-7 Azatadine dimaleate is an inhibitor of histamine and cholinergic with IC50 of 6.5 nM and 10 nM, respectively.
CSN10231 Alcaftadine 147084-10-4 Alcaftadine is a high affinity ligand for the H1 receptor, with a pKi (8.5) that is comparable with that of other H1 antihistamines.
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