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GSK-3

GSK-3

Cat. No. Product Name CAS No. Information
CSN15707 TWS119 601514-19-6 TWS119 is inhibitor of glycogen synthase kinase-3 with IC50 of 30 nM
CSN16043 Tideglusib   865854-05-3 Tideglusib is an irreversible GSK-3 inhibitor with IC50 of 5 nM and 60 nM for GSK-3WT (1 h preincubation) and GSK-3C199A (1 h preincubation), respectively.
CSN19500 TDZD-8 327036-89-5 TDZD-8, the derivative of thiadiazolidinone, is a selective inhibitor of GSK-3. It inhibits GSK-3 with IC50 of 2 M.
CSN23157 TCS 2002 1005201-24-0 TCS-2002 is a Potent inhibitor of GSK-3β (IC50 = 35 nM). Oral adminstration inhibits cold water stress-induced tau hyperphosphorylation in the mouse brain.
CSN16568 SB-415286   264218-23-7 SB-415286 is an ATP-competitive inhibitor of GSK3GSK3 with IC50 of 78 nM and Ki of 31 nM
CSN12268 SB-216763 280744-09-4 SB-216763 is potent and selective glycogen synthase kinase-3 GSK-3 inhibitor Ki 9 nM and competes with ATP
CSN23154 TC-G 24 1257256-44-2 Potent and selective GSK-3β inhibitor
CSN18355 LY2090314 603288-22-8 LY2090314 is a potent inhibitor of glycogen synthase kinase-3 (GSK-3) with IC50s of 1.5 nM and 0.9 nM for GSK-3α and GSK-3β respectively.
CSN22886 Lithium Carbonate 554-13-2 Lithium Carbonate inhibits GSK-3 in vivo.
CSN11250 Kenpaullone   142273-20-9 Kenpaullone is an ATP-competitive inhibitor of CDK1cyclin B (IC50 0.4 M), CDK2cyclin A (IC50 0.68 M), CDK5p25 (IC50 0.85 M), lymphocyte kinase (IC50 0.47 M) , and GSK-3 (C50 0.23 M).
CSN11201 Indirubin-3'-Monoxime 160807-49-8 Indirubin-3-monoxime is a powerful inhibitor of GSK-3 with IC50 of 22nM also inhibits CDK15 IC50 180100 nM
CSN17487 IM-12   1129669-05-1 IM-12 is a GSK-3 inhibitor with IC50 of 53 nM
CSN23173 TWS119 Trifluoroacetate 1507095-58-0 GSK-3β inhibitor; induces neuronal differentiation in ESCs
CSN18354 GSK-3 Inhibitor 1 603272-51-1 GSK-3 inhibitor 1 is a potent GSK-3 inhibitor
CSN24803 GNF4877 2041073-22-5 GNF4877 is a potent DYRK1A and GSK3β inhibitor with IC50s of 6 nM and 16 nM, respectively
CSN24779 EHT 5372 1425945-60-3 EHT 5372 is a strong inhibitor of DYRK’s family kinases, with IC50s of 0.22, 0.28 nM for DYRK1A and DYRK1B, respectively.
CSN17624 CP21R7 125314-13-8 CP21R7 is a slective inhibitor of GSK-3
CSN13470 CHIR-99021     252917-06-9 CHIR-99021 is a GSK-3α/β inhibitor with IC50 of 10 nM/6.7 nM, exhibiting > 500-fold selectivity for GSK-3 versus its closest homologs CDC2 and ERK2, as well as other protein kinases.
CSN19176 CHIR-99021 HCl 1797989-42-4 CHIR-99021 HCl is HCl of CHIR-99021, which is a GSK-3α/β inhibitor with IC50 of 10 nM/6.7 nM and shows greater than 500-fold selectivity for GSK-3 versus its closest homologs Cdc2 and ERK2.
CSN19149 CHIR-99021 3HCl 1782235-14-6 CHIR-99021 3HCl is a GSK-3α/β inhibitor with IC50 of 10 nM/6.7 nM, showing > 500-fold selectivity for GSK-3 versus its closest homologs CDC2 and ERK2, as well as other protein kinases.
CSN20636 CHIR-98024 556813-39-9 CHIR-98014 is a reversible inhibitor of GSK3 and GSK3 with IC50 of 065 nM and 058 nM respectively
CSN23355 CHIR-98014 252935-94-7 CHIR-98014 CT98014 is highly selective aminopyrimidine-derivatived inhibitor of GSK-3 with IC50 of 650nM and 580nM for GSK-3 and GSK-3measured by kinase assays respectively and exhibits 1000-fold selectivity for GSK-3 over closely related kinases such as cdc2
CSN16227 BIO-Acetoxime   667463-85-6 BIO-acetoxime is an inhibitor of GSK3 and GSK3 with IC50 of 10 nM.
CSN16080 BIO   667463-62-9 BIO is an inhibitor of GSK-3 and CDK1cyclinB complex. The IC50s of GSK-3, CDK1, CDK5 are 5 nM, 320 nM and 83 nM, respectively.
CSN13082 Bikinin   188011-69-0 Bikinin acts as an ATP-competitive inhibitor of arabidopsis GSK-3 and effective activator of brassinosteroid BR signaling
CSN13894 AZD2858 486424-20-8 AZD2858 is an inhibitor of GSK-3 with IC50 of 68 nM that can inhibit the tau phosphorylation of S396 site and activate Wnt signaling pathway
CSN16226 AZD1080   612487-72-6 AZD1080 is a selective, orally active, brain permeable GSK3 inhibitor of GSK3α and GSK3β with Ki of 6.9 nM and 31 nM, respectively, shows > 14-fold selectivity against CDK2, CDK5, CDK1 and Erk2.
CSN15984 AR-A014418   487021-52-3 AR-A014418 is a selective inhibitor of GSK3 with IC50 of 104 27 nM.
CSN22657 A 1070722 1384424-80-9 A 1070722 is a potent glycogen synthase kinase-3 (GSK-3) inhibitor with Ki of 0.6 nM for GSK-3α and GSK-3β.
CSN23598 5-Bromoindole   10075-50-0 5-bromoindole is an inhibitor ofglycogen synthase kinase 3 GSK-3 it can be used as important pharmaceutical chemical intermediate
CSN22644 2B-(SP) 186901-17-7 2B-(SP) is a selective phosphopeptide substrate for glycogen synthase kinase-3 (GSK-3).
CSN18742 1-Azakenpaullone 676596-65-9 1-Azakenpaullone is a potent and selective GSK-3 inhibitor with IC50 of 18 nM 100-fold selectivity over CDK1cyclin B and CDK5p25
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