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GPCR
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN25229 | SBI-115 | 882366-16-7 | SBI-115 is a GPBAR1 (TGR5) antagonist. |
| CSN22976 | ML 193 | 713121-80-3 | ML 193 is a selective GPR55 antagonist with IC50 of 221 nM. |
| CSN22972 | MK 1903 | 1268882-43-4 | MK 1903 is a potent and selective hydroxycarboxylic acid receptor 2 (HCA2, GPR109A) full agonist. |
| CSN22968 | MEDICA 16 | 87272-20-6 | MEDICA 16 is a free fatty acid 1 (FFA1/GPR40) receptor agonist. |
| CSN23711 | MCHr1 Antagonist 1 | 391610-37-0 | MCHr1 antagonist 1 is a selective antagonist of MCH1 receptor with Kb of 1 nM and Ki of 4 nM at human MCHR1, may be used to reduce the body mass. |
| CSN21714 | Lodoxamide | 53882-12-5 | Lodoxamide is an agonist of GPR35. |
| CSN14893 | Grifolic Acid | 80557-12-6 | Grifolic acid, a natural product isolated and purified from the Cylindrocarpon ianthothele var. majus, with anti-tumour and anti-haemolytic activities. Grifolic acid is a glucose-6-phosphatase inhibitor and a selective partial GPR120 agonist, can induce ERK and Ca2i responses in cells expressing GPR120. |
| CSN12484 | Ginsenoside Rb2 | 11021-13-9 | Ginsenoside Rb2 is a 20 (S)-protopanaxadiol glycoside extracted from ginseng, shows potent antioxidant and anticancer biological activities. |
| CSN10769 | Deoxycholic Acid | 83-44-3 | Deoxycholic Acid is a proinflammatory agent and used in a study to investigate dose-dependent anti-inflammatory effect of ursodeoxycholic acid in experimental colitis. |
| CSN20443 | CYM 5541 | 945128-26-7 | CYM-5541 is an allosteric agonist of S1P3 with EC50 of 72 nM - 132 nM. |
| CSN23236 | CID 1375606 | 313493-80-0 | CID 1375606 is an agonist of GPR27 SREB1 that induces coupling of the receptor to -arrestin 2 |
| CSN23765 | AS 1269574 | 330981-72-1 | AS 1269574 is a GPR119 receptor agonist with EC50 of 25 M in HEK293 cells expressing human GPR119 |
| CSN22671 | AH 7614 | 6326-06-3 | AH 7614 is a selective free fatty acid receptor 4 (FFA4/GPR120) antagonist with pIC50 of 7.1 for human FFA4. |
| CSN23532 | AF64394 | 1637300-25-4 | AF64394 is an inverse agonist of GPR3 with pIC50 of 7.3. |
| CSN16337 | 6-OAU | 83797-69-7 | 6-OAU is a surrogate agonist of GPR84 activating human GPR84 in the presence of Gqi5 chimera in HEK293 cells with an EC50 of 105 nM in the PI assay. |
| CSN25414 | 3-chloro-5-hydroxybenzoic Acid | 53984-36-4 | 3-chloro-5-hydroxybenzoic Acid is a selective GPR81 agonist that exhibited favorable in vivo effects on lipolysis in a mouse model of obesity. |
| CSN23486 | 3,5-Dihydroxybenzoic acid | 99-10-5 | 3 5-dihydroxybenzoic acid is a metabolite of alkylresinols with a certain activation effect on HCA1 It can be used as intermediates in organic synthesis |
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