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GPCR

GPCR

Cat. No. Product Name CAS No. Information
CSN25229 SBI-115 882366-16-7 SBI-115 is a GPBAR1 (TGR5) antagonist.
CSN22976 ML 193 713121-80-3 ML 193 is a selective GPR55 antagonist with IC50 of 221 nM.
CSN22972 MK 1903 1268882-43-4 MK 1903 is a potent and selective hydroxycarboxylic acid receptor 2 (HCA2, GPR109A) full agonist.
CSN22968 MEDICA 16 87272-20-6 MEDICA 16 is a free fatty acid 1 (FFA1/GPR40) receptor agonist.
CSN23711 MCHr1 Antagonist 1 391610-37-0 MCHr1 antagonist 1 is a selective antagonist of MCH1 receptor with Kb of 1 nM and Ki of 4 nM at human MCHR1, may be used to reduce the body mass.
CSN21714 Lodoxamide 53882-12-5 Lodoxamide is an agonist of GPR35.
CSN14893 Grifolic Acid 80557-12-6 Grifolic acid, a natural product isolated and purified from the Cylindrocarpon ianthothele var. majus, with anti-tumour and anti-haemolytic activities. Grifolic acid is a glucose-6-phosphatase inhibitor and a selective partial GPR120 agonist, can induce ERK and Ca2i responses in cells expressing GPR120.
CSN12484 Ginsenoside Rb2 11021-13-9 Ginsenoside Rb2 is a 20 (S)-protopanaxadiol glycoside extracted from ginseng, shows potent antioxidant and anticancer biological activities.
CSN10769 Deoxycholic Acid   83-44-3 Deoxycholic Acid is a proinflammatory agent and used in a study to investigate dose-dependent anti-inflammatory effect of ursodeoxycholic acid in experimental colitis.
CSN20443 CYM 5541 945128-26-7 CYM-5541 is an allosteric agonist of S1P3 with EC50 of 72 nM - 132 nM.
CSN23236 CID 1375606   313493-80-0 CID 1375606 is an agonist of GPR27 SREB1 that induces coupling of the receptor to -arrestin 2
CSN23765 AS 1269574 330981-72-1 AS 1269574 is a GPR119 receptor agonist with EC50 of 25 M in HEK293 cells expressing human GPR119
CSN22671 AH 7614 6326-06-3 AH 7614 is a selective free fatty acid receptor 4 (FFA4/GPR120) antagonist with pIC50 of 7.1 for human FFA4.
CSN23532 AF64394 1637300-25-4 AF64394 is an inverse agonist of GPR3 with pIC50 of 7.3.
CSN16337 6-OAU 83797-69-7 6-OAU is a surrogate agonist of GPR84 activating human GPR84 in the presence of Gqi5 chimera in HEK293 cells with an EC50 of 105 nM in the PI assay.
CSN25414 3-chloro-5-hydroxybenzoic Acid 53984-36-4 3-chloro-5-hydroxybenzoic Acid is a selective GPR81 agonist that exhibited favorable in vivo effects on lipolysis in a mouse model of obesity.
CSN23486 3,5-Dihydroxybenzoic acid 99-10-5 3 5-dihydroxybenzoic acid is a metabolite of alkylresinols with a certain activation effect on HCA1 It can be used as intermediates in organic synthesis
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