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Glucagon Receptor
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN26148 | (S)-2,2',4,4',5,5'-Hexahydroxy-7,7'-dimethyl-[1,1'-bianthracene]-9,9',10,10'-tetraone | 602-06-2 | Skyrin is a fungal bisanthroquinone. It exhibits functional glucagon antagonism by uncoupling the glucagon receptor from adenylate cyclase activation in rat liver membranes. |
| CSN25223 | Danuglipron (PF-06882961) | 2230198-02-2 | PF-06882961 is a potent and orally bioavailable GLP-1R agonist. |
| CSN13565 | MK 0893 | 870823-12-4 | MK 0893 is a potent selective glucagon receptor antagonist with IC50 of 66 nM showing 200 fold selectivity for GIPR PAC1 GLP-1R VPAC1 and VPAC2 |
| CSN23794 | LGD-6972 | 1207989-09-0 | LGD-6972 is a novel and orally-available glucagon receptor antagonist used to treat type 2 diabetes mellitus in Phase 1 study. |
| CSN22875 | L-168049 | 191034-25-0 | L-168,049 is a very potent and selective, non-competitive antagonist of the human glucagon receptor with IC50 of 3.7 nM. |
| CSN18988 | GRA Ex-25 | 307983-31-9 | GRA Ex-25 is an inhibitor of glucagon receptor with IC50 of 56 and 55 nM for rat and human glucagon receptors respectively |
| CSN17234 | PF-06291874 | 1393124-08-7 | Glucagon receptor antagonists-4 is an selective antagonist of glucagon receptor |
| CSN18088 | Glucagon receptor antagonists-3 | 202917-17-7 | Glucagon receptor antagonists-3 is a highly potent glucagon receptor antagonist |
| CSN18089 | Glucagon receptor antagonists-2 | 202917-18-8 | Glucagon receptor antagonists-2 is a highly potent glucagon receptor antagonist |
| CSN13173 | Glucagon receptor antagonists-1 | 503559-84-0 | Glucagon receptor antagonists-1 is a highly potent glucagon receptor antagonist |
| CSN22077 | BETP | 1371569-69-5 | BETP is an agonist of glucagon-like peptide-1 (GLP-1) receptor, with EC50s of 0.66 and 0.755 μM for human and rat GLP-1 receptor, respectively. |
| CSN17364 | Adomeglivant | 1488363-78-5 | Adomeglivant is a potent and selective glucagon receptor antagonist that is used in clinical trial for type 2 diabetes mellitus |
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