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GABA Receptor

GABA Receptor

Cat. No. Product Name CAS No. Information
CSN17779 Vigabatrin HCl 1391054-02-6 Vigabatrin HCl is a structural analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA) that irreversibly inhibits the catabolism of GABA by GABA transaminase.
CSN12084 Tiagabine 115103-54-3 Tiagabine is an anti-convulsive medication and a selective gamma-aminobutyric acid (GABA) reuptake inhibitor.
CSN12085 Tiagabine HCl   145821-59-6 Tiagabine HCl is an inhibitor of gamma-aminobutyric acid (GABA) reuptake (IC50 = 67 nM in vivo) with anticonvulsant effect.
CSN12077 Thiocolchicoside 602-41-5 Thiocolchicoside is a small molecule muscle relaxant and anti-inflammatory agent, shown to function as a competitive GABAA (gamma-aminobutyric acid type A) receptor antagonist.
CSN23715 SAGE-217 1632051-40-1 SAGE-217 is an agonist of GABAA receptor with EC50s of 296 nM and 163 nM for 122 and 43 respectively
CSN19798 Ro 48-6791 172407-17-9 Ro 48-6791 is a GABA receptor agonist potentially for the use of anesthesia
CSN10515 Progabide 62666-20-0 Progabide is an analog and prodrug of gamma-aminobutyric acid It is commonly used in the treatment of epilepsy with agonistic activity for both the GABAA and GABAB receptors Progabide has been investigated for many diseases besides epilepsy including Parkinsons disease schizophrenia clinical depression and anxiety disorder with varying success
CSN21797 Pipequaline 77472-98-1 Pipequaline is a partial agonist of benzodiazepine receptor (Ki = 78 nM) with anxiolytic activity.
CSN11714 Phytol   150-86-7 Phytol can activite PPAR and attenuate the inflammatory response by inhibiting neutrophil migration and oxidative stress. Phytol is isolated from the leaves of black tea and acts as an aromatic ingredient.
CSN19514 Oxiracetam(Random Configuration)   62613-82-5 Oxiracetam is a derivative of gamma-aminobutyric acid GABA and used as a nootropic drug to improve memory and learning
CSN11488 Nefiracetam   77191-36-7 Nefiracetam is a neuronal systems enhancer for Ro 5-4864-induced convulsions. Nefiracetam has GABAergic, cholinergic, and monoaminergic properties.
CSN15900 NCS-382 Sodium 131733-92-1 NCS-382 sodium is a -hydroxybutyric acid antagonist, anticonvulsant.
CSN23642 MRX-1024   348-67-4 MRX-1024 can inhibit the activation of GABAA receptor and exhibit relieving effect on hearing loss It can used as a chemoprotective agent
CSN18228 MRK-016 342652-67-9 MRK-016 is a functionally selective, inverse agonist at the benzodiazepine site of GABAA 5 receptors.
CSN19855 MK 0343 233275-76-8 MK 0343 is a selective partial agonist of GABAA3 1 5 and 2 with Ki values of 021 nM-040 nM It displays anxiolytic activity in rodent and primate models
CSN24055 Loreclezole 117857-45-1 Loreclezole is a subtype-selective GABAA receptor modulator. Acts as a positive allosteric modulator of β2 or β3-subunit containing receptors.
CSN19849 Loreclezole HCl 2227372-56-5 Loreclezole HCl is a subtype-selective GABAA receptor modulator. Acts as a positive allosteric modulator of β2 or β3-subunit containing receptors.
CSN16300 L-Cycloserine   339-72-0 L-cycloserine is an inhibitor of serine palmitoyltransferase and block sphingosine biosynthesis It has antibiotic effective against mycobacterium tuberculosis
CSN15698 L-838,417 286456-42-6 L-838417 is a subtype-selective GABAA receptor partial agonist L-838417 selectively binds to 1 2 3 and 5 subunits Ki values are 079 067 067 and 225 nM respectively but displays no efficacy at 1 1-sparing L-838417 exhibits non-sedative anxiolytic antinociceptive and anti-inflammatory activity
CSN20905 Kavain 3155-48-4 Kavain is a positive allosteric modulator of α4β2δ subunit-containing GABAA receptors.
CSN21680 Hypotaurine 300-84-5 Hypotaurine, a analog of cystamine, is the precursor for taurine synthesis and can act as an antioxidant and singlet oxygen scavenger. it also acts as an endogenous neurotransmitter via action on the glycine receptors.
CSN19501 Ginsenoside Rc   11021-14-0 Ginsenoside Rc is a steroid glycoside, and a triterpene saponin found exclusively in the plant genus Panax (ginseng) with properties that inhibit or prevent tumors growth.
CSN12568 Ginkgolide A 15291-75-5 Ginkgolide A is an antagonist of g-aminobutyric acid (GABA) with Ki of 14.5 M and also can activate PAF. It is purified from the leaves of ginkgo biloba tree.
CSN10697 Gelsemine 509-15-9 Gelsemine a natural indole alkaloid isolated from flowering plants of the genus Gelsemium with potent activity as an agonist of the mammalian glycine receptor, showing effect on pathwayssystems related to xenobiotic- or diet-induced oxidative stress, and in the treatment of anxiety and other conditions.
CSN15872 Gabazine Hydrobromide 104104-50-9 Gabazine hydrobromide is a drug that acts as an antagonist at GABAA receptors It is used in scientific research and has no role in medicine as it would be expected to produce convulsions if used in humans
CSN16786 Flumazenil 78755-81-4 Flumazenil is a non-selective antagonist of benzodiazepine towards 1 2 3 or 5-containing GABAA receptors
CSN18321 Etomidate HCl 53188-20-8 Etomidate HCl is a GABAA receptors agonist, which is a short acting intravenous anaesthetic agent used for the induction of general anaesthesia.
CSN18338 Etifoxine HCl   56776-32-0 Etifoxine HCl is a potentiator of β2 or β3 subunit-containing GABAA receptor that promotes axonal regeneration. It shows anxiolytic activity with no effects.
CSN17006 Emamectin Benzoate 155569-91-8 Emamectin benzoate acts as an activator of chloride channel via binding gamma aminobutyric acid GABA receptor and glutamate-gated chloride channels It can disrupt nerve signals in arthropods
CSN21616 Doxefazepam 40762-15-0 Doxefazepam is a benzodiazepine medication with anxiolyti and anticonvulsant properties. It is used therapeutically as a hypnotic.
CSN17574 DMCM HCl 1215833-62-7 DMCM HCl is benzodiazepine inverse agonist that displays anxiogenic and potent convulsant activity.
CSN21600 Deramciclane 120444-71-5 Deramciclane is an antagonist of 5-HT2A and inverse agonist of 5-HT2C receptor. It also functions as a GABA reuptake inhibitor.
CSN17089 Bemegride 64-65-3 Bemegride can stimulate central nervous system and release barbiturate poisoning
CSN19034 Basmisanil   1159600-41-5 Basmisanil is a selective modulator of GABAA5 with negative allosteric regulation.
CSN10524 Baclofen   1134-47-0 Baclofen a gamma-amino-butyric acid derivative is a selective GABAB agonist with IC50 of 200 nM which used as a skeletal muscle relaxant
CSN10198 Acamprosate Calcium   77337-73-6 Acamprosate calcium is an agonist of GABA receptor It can act as a modulator of glutamatergic systems and reduce alcohol consumption in animal models of alcohol addiction
CSN22026 6,2'-Dihydroxyflavone 92439-20-8 6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor.
CSN12782 4-Aminobutyric Acid   56-12-2 4-Aminobutyric acid exhibits inhibitory activity on central nervous system (CNS). It is a natural neurotransmitter.
CSN10435 (+)-Bicuculline   485-49-4 -Bicuculline is an antagonist of GABAA receptor with IC50 of 2 M and also shows inhibition of Ca2-activated potassium channels
CSN23429 L-Glutamic Acid   56-86-0 (S)-Glutamic acid acts as an excitatory neurotransmitter in the central nervous system.
CSN17026 (R)-Baclofen   69308-37-8 (R)-Baclofen is a derivative of gamma-aminobutyric acid with the selective activation of GABAB receptor that is used to treat spasticity.
CSN14755 (-)-Corlumine 79082-64-7 (-)-Corlumine is a natural product isolated and purified from the herbs of Fumaria parviflora with spasmolytic and GABA antagonist activity.
CSN23331 6-Hydroxyflavone 6665-83-4
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