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GABA Receptor
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN17779 | Vigabatrin HCl | 1391054-02-6 | Vigabatrin hydrochloride is a structural analog of the inhibitory neurotransmitter -aminobutyric acid (GABA) that irreversibly inhibits the catabolism of GABA by GABA transaminase. |
| CSN19031 | U93631 | 152273-12-6 | U93631 is a ligand of GABAA receptor ligand IC50 100 nM which can induce a rapid decay of GABA-induced chloride currents |
| CSN12084 | Tiagabine | 115103-54-3 | Tiagabine is an anti-convulsive medication and a selective gamma-aminobutyric acid (GABA) reuptake inhibitor. |
| CSN12085 | Tiagabine HCl | 145821-59-6 | Tiagabine hydrochloride is an inhibitor of gamma-aminobutyric acid (GABA) reuptake (IC50 67 nM in vivo) with anticonvulsant effect. |
| CSN13133 | Thymol | 89-83-8 | Thymol a natural product isolated and purified from the herbs of Thymus serpyllum L is a positive allosteric modulator of human GABAA receptors and a homo-oligomeric GABA receptor from Drosophila melanogaster |
| CSN12077 | Thiocolchicoside | 602-41-5 | Thiocolchicoside is a small molecule muscle relaxant and anti-inflammatory agent, shown to function as a competitive GABAA (gamma-aminobutyric acid type A) receptor antagonist. |
| CSN21312 | SX-3228 | 156364-04-4 | SX-3228 is a selective benzodiazepine1 BZ1 receptor agonist with an IC50 of 17 nM |
| CSN21079 | SSD114 HCl | N/A | SSD114 is a GABAB positive allosteric modulator SSD114 potentiated GABA-stimulated 35SGTPS binding to native GABAB receptors whereas it had no effect when used alone SSD114 a molecule with a different chemical structure compared to known GABAB PAMs is a novel GABAB PAM with potential usefulness in the GABAB-receptor research field |
| CSN23715 | SAGE-217 | 1632051-40-1 | SAGE-217 is an agonist of GABAA receptor with EC50s of 296 nM and 163 nM for 122 and 43 respectively |
| CSN22497 | RO 4938581 | 883093-10-5 | RO 4938581 is a potent and selective GABAA 5 inverse agonist with a Ki of 46 nM for GABAA 532a and shows a lower affinity at 132a 232a 332a Ki 174 185 80 nM respectively RO 4938581 is used in the research of cognitive dysfunction |
| CSN19798 | Ro 48-6791 | 172407-17-9 | Ro 48-6791 is a GABA receptor agonist potentially for the use of anesthesia |
| CSN20452 | Ro 15-3890 | 84378-44-9 | Ro 15-3890 is an antagonist of benzodiazepine receptor It is a main metabolite of Ro 15-1788 flumazenil |
| CSN11846 | Rilmazafone | 99593-25-6 | Rilmazafone is a water-soluble benzodiazepine prodrug developed in Japan It has sedative and hypnotic effects |
| CSN11821 | (R)-Baclofen HCl | 63701-55-3 | R-Baclofen hydrochloride is a derivative of gamma-aminobutyric acid GABA primarily used to treat spasticity and is in the early research stages for use for the treatment of alcoholism |
| CSN10515 | Progabide | 62666-20-0 | Progabide is an analog and prodrug of gamma-aminobutyric acid It is commonly used in the treatment of epilepsy with agonistic activity for both the GABAA and GABAB receptors Progabide has been investigated for many diseases besides epilepsy including Parkinsons disease schizophrenia clinical depression and anxiety disorder with varying success |
| CSN11714 | Phytol | 150-86-7 | Phytol can activite PPAR and attenuate the inflammatory response by inhibiting neutrophil migration and oxidative stress. Phytol is isolated from the leaves of black tea and acts as an aromatic ingredient. |
| CSN11659 | Pazinaclone | 103255-66-9 | Pazinaclone is a sedative and anxiolytic drug in the cyclopyrrolone family of drugs |
| CSN19514 | Oxiracetam(Random Configuration) | 62613-82-5 | Oxiracetam is a derivative of gamma-aminobutyric acid GABA and used as a nootropic drug to improve memory and learning |
| CSN11488 | Nefiracetam | 77191-36-7 | Nefiracetam is a neuronal systems enhancer for Ro 5-4864-induced convulsions. Nefiracetam has GABAergic, cholinergic, and monoaminergic properties. |
| CSN23642 | MRX-1024 | 348-67-4 | MRX-1024 can inhibit the activation of GABAA receptor and exhibit relieving effect on hearing loss It can used as a chemoprotective agent |
| CSN18575 | Lorediplon | 917393-39-6 | Lorediplon non-benzodiazepine hypnotic drug acts as a modulator of GABAA receptor with the effect of promoting sleep |
| CSN19849 | Loreclezole HCl | 2227372-56-5 | Loreclezole hydrochloride is a subtype-selective GABAA receptor modulator Acts as a positive allosteric modulator of 2 or 3-subunit containing receptors |
| CSN16300 | L-Cycloserine | 339-72-0 | L-cycloserine is an inhibitor of serine palmitoyltransferase and block sphingosine biosynthesis It has antibiotic effective against mycobacterium tuberculosis |
| CSN15698 | L-838,417 | 286456-42-6 | L-838417 is a subtype-selective GABAA receptor partial agonist L-838417 selectively binds to 1 2 3 and 5 subunits Ki values are 079 067 067 and 225 nM respectively but displays no efficacy at 1 1-sparing L-838417 exhibits non-sedative anxiolytic antinociceptive and anti-inflammatory activity |
| CSN17671 | L-655,708 | 130477-52-0 | L-655708 is a potent 5 subunit-selective GABAA receptor inverse agonist Ki 045 nM |
| CSN12568 | Ginkgolide A | 15291-75-5 | Ginkgolide A is an antagonist of g-aminobutyric acid (GABA) with Ki of 14.5 M and also can activate PAF. It is purified from the leaves of ginkgo biloba tree. |
| CSN16036 | Gaboxadol HCl | 85118-33-8 | Gaboxadol hydrochloride is a systemically active GABAA receptor agonist and GABAA- receptor antagonist Displays antinociceptive anticonvulsant and sedative effects Hypnotic agent that enhances delta activity within non-REM sleep in rats |
| CSN15872 | Gabazine Hydrobromide | 104104-50-9 | Gabazine hydrobromide is a drug that acts as an antagonist at GABAA receptors It is used in scientific research and has no role in medicine as it would be expected to produce convulsions if used in humans |
| CSN12825 | Gabapentin | 60142-96-3 | Gabapentin is an analogue of GABA that used to treat seizures and neuropathic pain |
| CSN16669 | Gabapentin HCl | 60142-95-2 | Gabapentin is a GABA analogue used to treat seizures and neuropathic pain |
| CSN16786 | Flumazenil | 78755-81-4 | Flumazenil is a non-selective antagonist of benzodiazepine towards 1 2 3 or 5-containing GABAA receptors |
| CSN10967 | Etomidate | 33125-97-2 | Etomidate is an agonist of GABAA receptor and used as a short acting intravenous anaesthetic agent |
| CSN18321 | Etomidate HCl | 53188-20-8 | Etomidate hydrochloride is a GABAA receptors agonist which is a short acting intravenous anaesthetic agent used for the induction of general anaesthesia |
| CSN10962 | Etifoxine | 21715-46-8 | Etifoxine is potentiator of GABAA receptor function in cultured neurons |
| CSN18338 | Etifoxine HCl | 56776-32-0 | Etifoxine hydrochloride is a potentiator of 2 or 3 subunit-containing GABAA receptor that promotes axonal regeneration It shows anxiolytic activity with no effects |
| CSN17006 | Emamectin Benzoate | 155569-91-8 | Emamectin benzoate acts as an activator of chloride channel via binding gamma aminobutyric acid GABA receptor and glutamate-gated chloride channels It can disrupt nerve signals in arthropods |
| CSN16005 | Cloxacillin Sodium | 642-78-4 | Cloxacillin is a semisynthetic antibiotic that belongs to the group of the isoxazolylpenicillins and is used to treat infections caused by species of staphylococci that produce beta-lactamase due to its inhibitory effects on beta-lactamase binding |
| CSN11041 | Chlormezanone | 80-77-3 | Chlormezanone can bind to central benzodiazepine receptors used in the management of anxiety and in the treatment of muscle spasm |
| CSN18672 | CGS-9896 | 77779-36-3 | CGS-9896 is an anxiolytic drug used in scientific research |
| CSN21178 | CGP52432 | 139667-74-6 | CGP52432 is an antagonist of GABAB receptor with an IC50 of 85 nM |
| CSN19034 | Basmisanil | 1159600-41-5 | Basmisanil is a selective modulator of GABAA5 with negative allosteric regulation. |
| CSN16275 | AWD 131-138 | 188116-07-6 | AWD 131-138 is a partial agonist of benzodiazepine receptor with effective anticonvulsant and anxiolytic properties |
| CSN10198 | Acamprosate Calcium | 77337-73-6 | Acamprosate calcium is an agonist of GABA receptor It can act as a modulator of glutamatergic systems and reduce alcohol consumption in animal models of alcohol addiction |
| CSN12782 | 4-Aminobutyric Acid | 56-12-2 | 4-Aminobutyric acid exhibits inhibitory activity on central nervous system (CNS). It is a natural neurotransmitter. |
| CSN10435 | (+)-Bicuculline | 485-49-4 | -Bicuculline is an antagonist of GABAA receptor with IC50 of 2 M and also shows inhibition of Ca2-activated potassium channels |
| CSN17026 | (R)-Baclofen | 69308-37-8 | (R)-Baclofen is a derivative of gamma-aminobutyric acid with the selective activation of GABAB receptor that is used to treat spasticity. |
| CSN11911 | Securinine | 5610-40-2 | |
| CSN23331 | 6-Hydroxyflavone | 6665-83-4 | |
| CSN23337 | Phenibut | 1078-21-3 |
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