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GABA Receptor

GABA Receptor

Cat. No. Product Name CAS No. Information
CSN17779 Vigabatrin HCl 1391054-02-6 Vigabatrin hydrochloride is a structural analog of the inhibitory neurotransmitter -aminobutyric acid (GABA) that irreversibly inhibits the catabolism of GABA by GABA transaminase.
CSN19031 U93631   152273-12-6 U93631 is a ligand of GABAA receptor ligand IC50 100 nM which can induce a rapid decay of GABA-induced chloride currents
CSN12084 Tiagabine 115103-54-3 Tiagabine is an anti-convulsive medication and a selective gamma-aminobutyric acid (GABA) reuptake inhibitor.
CSN12085 Tiagabine HCl   145821-59-6 Tiagabine hydrochloride is an inhibitor of gamma-aminobutyric acid (GABA) reuptake (IC50 67 nM in vivo) with anticonvulsant effect.
CSN13133 Thymol 89-83-8 Thymol a natural product isolated and purified from the herbs of Thymus serpyllum L is a positive allosteric modulator of human GABAA receptors and a homo-oligomeric GABA receptor from Drosophila melanogaster
CSN12077 Thiocolchicoside 602-41-5 Thiocolchicoside is a small molecule muscle relaxant and anti-inflammatory agent, shown to function as a competitive GABAA (gamma-aminobutyric acid type A) receptor antagonist.
CSN21312 SX-3228 156364-04-4 SX-3228 is a selective benzodiazepine1 BZ1 receptor agonist with an IC50 of 17 nM
CSN21079 SSD114 HCl N/A SSD114 is a GABAB positive allosteric modulator SSD114 potentiated GABA-stimulated 35SGTPS binding to native GABAB receptors whereas it had no effect when used alone SSD114 a molecule with a different chemical structure compared to known GABAB PAMs is a novel GABAB PAM with potential usefulness in the GABAB-receptor research field
CSN23715 SAGE-217 1632051-40-1 SAGE-217 is an agonist of GABAA receptor with EC50s of 296 nM and 163 nM for 122 and 43 respectively
CSN22497 RO 4938581 883093-10-5 RO 4938581 is a potent and selective GABAA 5 inverse agonist with a Ki of 46 nM for GABAA 532a and shows a lower affinity at 132a 232a 332a Ki 174 185 80 nM respectively RO 4938581 is used in the research of cognitive dysfunction
CSN19798 Ro 48-6791 172407-17-9 Ro 48-6791 is a GABA receptor agonist potentially for the use of anesthesia
CSN20452 Ro 15-3890 84378-44-9 Ro 15-3890 is an antagonist of benzodiazepine receptor It is a main metabolite of Ro 15-1788 flumazenil
CSN11846 Rilmazafone 99593-25-6 Rilmazafone is a water-soluble benzodiazepine prodrug developed in Japan It has sedative and hypnotic effects
CSN11821 (R)-Baclofen HCl 63701-55-3 R-Baclofen hydrochloride is a derivative of gamma-aminobutyric acid GABA primarily used to treat spasticity and is in the early research stages for use for the treatment of alcoholism
CSN10515 Progabide 62666-20-0 Progabide is an analog and prodrug of gamma-aminobutyric acid It is commonly used in the treatment of epilepsy with agonistic activity for both the GABAA and GABAB receptors Progabide has been investigated for many diseases besides epilepsy including Parkinsons disease schizophrenia clinical depression and anxiety disorder with varying success
CSN11714 Phytol   150-86-7 Phytol can activite PPAR and attenuate the inflammatory response by inhibiting neutrophil migration and oxidative stress. Phytol is isolated from the leaves of black tea and acts as an aromatic ingredient.
CSN11659 Pazinaclone 103255-66-9 Pazinaclone is a sedative and anxiolytic drug in the cyclopyrrolone family of drugs
CSN19514 Oxiracetam(Random Configuration)   62613-82-5 Oxiracetam is a derivative of gamma-aminobutyric acid GABA and used as a nootropic drug to improve memory and learning
CSN11488 Nefiracetam   77191-36-7 Nefiracetam is a neuronal systems enhancer for Ro 5-4864-induced convulsions. Nefiracetam has GABAergic, cholinergic, and monoaminergic properties.
CSN23642 MRX-1024   348-67-4 MRX-1024 can inhibit the activation of GABAA receptor and exhibit relieving effect on hearing loss It can used as a chemoprotective agent
CSN18575 Lorediplon 917393-39-6 Lorediplon non-benzodiazepine hypnotic drug acts as a modulator of GABAA receptor with the effect of promoting sleep
CSN19849 Loreclezole HCl 2227372-56-5 Loreclezole hydrochloride is a subtype-selective GABAA receptor modulator Acts as a positive allosteric modulator of 2 or 3-subunit containing receptors
CSN16300 L-Cycloserine   339-72-0 L-cycloserine is an inhibitor of serine palmitoyltransferase and block sphingosine biosynthesis It has antibiotic effective against mycobacterium tuberculosis
CSN15698 L-838,417 286456-42-6 L-838417 is a subtype-selective GABAA receptor partial agonist L-838417 selectively binds to 1 2 3 and 5 subunits Ki values are 079 067 067 and 225 nM respectively but displays no efficacy at 1 1-sparing L-838417 exhibits non-sedative anxiolytic antinociceptive and anti-inflammatory activity
CSN17671 L-655,708 130477-52-0 L-655708 is a potent 5 subunit-selective GABAA receptor inverse agonist Ki 045 nM
CSN12568 Ginkgolide A 15291-75-5 Ginkgolide A is an antagonist of g-aminobutyric acid (GABA) with Ki of 14.5 M and also can activate PAF. It is purified from the leaves of ginkgo biloba tree.
CSN16036 Gaboxadol HCl 85118-33-8 Gaboxadol hydrochloride is a systemically active GABAA receptor agonist and GABAA- receptor antagonist Displays antinociceptive anticonvulsant and sedative effects Hypnotic agent that enhances delta activity within non-REM sleep in rats
CSN15872 Gabazine Hydrobromide 104104-50-9 Gabazine hydrobromide is a drug that acts as an antagonist at GABAA receptors It is used in scientific research and has no role in medicine as it would be expected to produce convulsions if used in humans
CSN12825 Gabapentin   60142-96-3 Gabapentin is an analogue of GABA that used to treat seizures and neuropathic pain
CSN16669 Gabapentin HCl 60142-95-2 Gabapentin is a GABA analogue used to treat seizures and neuropathic pain
CSN16786 Flumazenil 78755-81-4 Flumazenil is a non-selective antagonist of benzodiazepine towards 1 2 3 or 5-containing GABAA receptors
CSN10967 Etomidate   33125-97-2 Etomidate is an agonist of GABAA receptor and used as a short acting intravenous anaesthetic agent
CSN18321 Etomidate HCl 53188-20-8 Etomidate hydrochloride is a GABAA receptors agonist which is a short acting intravenous anaesthetic agent used for the induction of general anaesthesia
CSN10962 Etifoxine 21715-46-8 Etifoxine is potentiator of GABAA receptor function in cultured neurons
CSN18338 Etifoxine HCl   56776-32-0 Etifoxine hydrochloride is a potentiator of 2 or 3 subunit-containing GABAA receptor that promotes axonal regeneration It shows anxiolytic activity with no effects
CSN17006 Emamectin Benzoate 155569-91-8 Emamectin benzoate acts as an activator of chloride channel via binding gamma aminobutyric acid GABA receptor and glutamate-gated chloride channels It can disrupt nerve signals in arthropods
CSN16005 Cloxacillin Sodium 642-78-4 Cloxacillin is a semisynthetic antibiotic that belongs to the group of the isoxazolylpenicillins and is used to treat infections caused by species of staphylococci that produce beta-lactamase due to its inhibitory effects on beta-lactamase binding
CSN11041 Chlormezanone   80-77-3 Chlormezanone can bind to central benzodiazepine receptors used in the management of anxiety and in the treatment of muscle spasm
CSN18672 CGS-9896 77779-36-3 CGS-9896 is an anxiolytic drug used in scientific research
CSN21178 CGP52432 139667-74-6 CGP52432 is an antagonist of GABAB receptor with an IC50 of 85 nM
CSN19034 Basmisanil   1159600-41-5 Basmisanil is a selective modulator of GABAA5 with negative allosteric regulation.
CSN16275 AWD 131-138   188116-07-6 AWD 131-138 is a partial agonist of benzodiazepine receptor with effective anticonvulsant and anxiolytic properties
CSN10198 Acamprosate Calcium   77337-73-6 Acamprosate calcium is an agonist of GABA receptor It can act as a modulator of glutamatergic systems and reduce alcohol consumption in animal models of alcohol addiction
CSN12782 4-Aminobutyric Acid   56-12-2 4-Aminobutyric acid exhibits inhibitory activity on central nervous system (CNS). It is a natural neurotransmitter.
CSN10435 (+)-Bicuculline   485-49-4 -Bicuculline is an antagonist of GABAA receptor with IC50 of 2 M and also shows inhibition of Ca2-activated potassium channels
CSN17026 (R)-Baclofen   69308-37-8 (R)-Baclofen is a derivative of gamma-aminobutyric acid with the selective activation of GABAB receptor that is used to treat spasticity.
CSN11911 Securinine 5610-40-2
CSN23331 6-Hydroxyflavone 6665-83-4
CSN23337 Phenibut 1078-21-3
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