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GABA Receptor

GABA Receptor

Cat. No. Product Name CAS No. Information
CSN17779 Vigabatrin HCl 1391054-02-6 Vigabatrin HCl is a structural analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA) that irreversibly inhibits the catabolism of GABA by GABA transaminase.
CSN24498 TP003 628690-75-5 TP003 is a GABAA receptor partial agonist that demonstrates affinity for the benzodiazepine site.
CSN12084 Tiagabine 115103-54-3 Tiagabine is an anti-convulsive medication and a selective gamma-aminobutyric acid (GABA) reuptake inhibitor.
CSN12085 Tiagabine HCl   145821-59-6 Tiagabine HCl is an inhibitor of gamma-aminobutyric acid (GABA) reuptake (IC50 = 67 nM in vivo) with anticonvulsant effect.
CSN12077 Thiocolchicoside 602-41-5 Thiocolchicoside is a small molecule muscle relaxant and anti-inflammatory agent, shown to function as a competitive GABAA (gamma-aminobutyric acid type A) receptor antagonist.
CSN11911 Securinine 5610-40-2 Securinine, a natural product isolated and purified from the leaves and twigs of Securinega suffruticosa with antifungal activity, induces apoptosis in human leukemia HL-60 cells, is a promising monocytic differentiation inducing agent for Acute Myeloid Leukemia (AML).
CSN19979 Sanggenon D 81422-93-7 Sanggenon D, a natural product isolated and purified from the root bark of Morus alba L.
CSN20452 Ro 15-3890 84378-44-9 Ro 15-3890 is an antagonist of benzodiazepine receptor It is a main metabolite of Ro 15-1788 flumazenil
CSN10515 Progabide 62666-20-0 Progabide is an analog and prodrug of gamma-aminobutyric acid It is commonly used in the treatment of epilepsy with agonistic activity for both the GABAA and GABAB receptors Progabide has been investigated for many diseases besides epilepsy including Parkinsons disease schizophrenia clinical depression and anxiety disorder with varying success
CSN21797 Pipequaline 77472-98-1 Pipequaline is a partial agonist of benzodiazepine receptor (Ki = 78 nM) with anxiolytic activity.
CSN11714 Phytol   150-86-7 Phytol can activite PPAR and attenuate the inflammatory response by inhibiting neutrophil migration and oxidative stress. Phytol is isolated from the leaves of black tea and acts as an aromatic ingredient.
CSN23337 Phenibut 1078-21-3 Phenibut, a GABA analogue, is a central nervous system depressant with anxiolytic and sedative effects.
CSN11488 Nefiracetam   77191-36-7 Nefiracetam is a neuronal systems enhancer for Ro 5-4864-induced convulsions. Nefiracetam has GABAergic, cholinergic, and monoaminergic properties.
CSN15900 NCS-382 Sodium 131733-92-1 NCS-382 sodium is a -hydroxybutyric acid antagonist, anticonvulsant.
CSN18228 MRK-016 342652-67-9 MRK-016 is a functionally selective, inverse agonist at the benzodiazepine site of GABAA 5 receptors.
CSN19855 MK 0343 233275-76-8 MK 0343 is a selective partial agonist of GABAA3 1 5 and 2 with Ki values of 021 nM-040 nM It displays anxiolytic activity in rodent and primate models
CSN24055 Loreclezole 117857-45-1 Loreclezole is a subtype-selective GABAA receptor modulator. Acts as a positive allosteric modulator of β2 or β3-subunit containing receptors.
CSN19849 Loreclezole HCl 2227372-56-5 Loreclezole HCl is a subtype-selective GABAA receptor modulator. Acts as a positive allosteric modulator of β2 or β3-subunit containing receptors.
CSN17671 L-655,708 130477-52-0 L-655708 is a potent 5 subunit-selective GABAA receptor inverse agonist Ki 045 nM
CSN20905 Kavain 3155-48-4 Kavain is a positive allosteric modulator of α4β2δ subunit-containing GABAA receptors.
CSN21680 Hypotaurine 300-84-5 Hypotaurine, a analog of cystamine, is the precursor for taurine synthesis and can act as an antioxidant and singlet oxygen scavenger. it also acts as an endogenous neurotransmitter via action on the glycine receptors.
CSN19501 Ginsenoside Rc 11021-14-0 Ginsenoside Rc is a steroid glycoside, and a triterpene saponin found exclusively in the plant genus Panax (ginseng) with properties that inhibit or prevent tumors growth.
CSN12568 Ginkgolide A 15291-75-5 Ginkgolide A is an antagonist of g-aminobutyric acid (GABA) with Ki of 14.5 M and also can activate PAF. It is purified from the leaves of ginkgo biloba tree.
CSN10697 Gelsemine 509-15-9 Gelsemine a natural indole alkaloid isolated from flowering plants of the genus Gelsemium with potent activity as an agonist of the mammalian glycine receptor, showing effect on pathwayssystems related to xenobiotic- or diet-induced oxidative stress, and in the treatment of anxiety and other conditions.
CSN20431 EVT-201 308239-86-3 EVT-201 is a benzodiazepine derivative drug and partial positive allosteric modulator of the benzodiazepine site of the GABA receptor
CSN21616 Doxefazepam 40762-15-0 Doxefazepam is a benzodiazepine medication with anxiolyti and anticonvulsant properties. It is used therapeutically as a hypnotic.
CSN17574 DMCM HCl 1215833-62-7 DMCM HCl is benzodiazepine inverse agonist that displays anxiogenic and potent convulsant activity.
CSN21600 Deramciclane 120444-71-5 Deramciclane is an antagonist of 5-HT2A and inverse agonist of 5-HT2C receptor. It also functions as a GABA reuptake inhibitor.
CSN17089 Bemegride 64-65-3 Bemegride can stimulate central nervous system and release barbiturate poisoning
CSN19034 Basmisanil   1159600-41-5 Basmisanil is a selective modulator of GABAA5 with negative allosteric regulation.
CSN25262 AZD7325 942437-37-8 AZD-7325 is a GABA-Aα2,3 selective receptor modulator.
CSN24752 AZD6280 942436-93-3 AZD-6280 is a selective GABAA Receptor α2/3 modulator, used for treatment of generalized anxiety disorder.
CSN10198 Acamprosate Calcium   77337-73-6 Acamprosate calcium is an agonist of GABA receptor It can act as a modulator of glutamatergic systems and reduce alcohol consumption in animal models of alcohol addiction
CSN23521 6-Methyl-2-phenyl-4H-chromen-4-one 29976-75-8 6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.
CSN23331 6-Hydroxyflavone 6665-83-4 6-Hydroxyflavone is a naturally occurring flavone, with anti-inflammatory activity. 6-Hydroxyflavone exhibits inhibitory effect towards bovine hemoglobin (BHb) glycation. 6-Hydroxyflavone can activate AKT, ERK 1/2, and JNK signaling pathways to effectively promote osteoblastic differentiation. 6-Hydroxyflavone inhibits the LPS-induced NO production[1] [2].
CSN22026 6,2'-Dihydroxyflavone 92439-20-8 6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor.
CSN23335 5-methoxyflavone 42079-78-7 5-Methoxyflavone, belonged to Flavonoid family, is a DNA polymerase-beta inhibitor and neuroprotective agent against beta-amyloid toxicity. possess central nervous system (CNS) depressant effect mediated through the ionotropic GABAA receptors.
CSN12782 4-Aminobutyric Acid   56-12-2 4-Aminobutyric acid exhibits inhibitory activity on central nervous system (CNS). It is a natural neurotransmitter.
CSN10435 (+)-Bicuculline   485-49-4 -Bicuculline is an antagonist of GABAA receptor with IC50 of 2 M and also shows inhibition of Ca2-activated potassium channels
CSN23429 L-Glutamic Acid   56-86-0 (S)-Glutamic acid acts as an excitatory neurotransmitter in the central nervous system.
CSN17026 (R)-Baclofen   69308-37-8 (R)-Baclofen is a derivative of gamma-aminobutyric acid with the selective activation of GABAB receptor that is used to treat spasticity.
CSN14755 (-)-Corlumine 79082-64-7 (-)-Corlumine is a natural product isolated and purified from the herbs of Fumaria parviflora with spasmolytic and GABA antagonist activity.
CSN25408 Isonipecotic acid 498-94-2
CSN25410 Saclofen 125464-42-8
CSN25409 Ganaxolone 38398-32-2
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