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GABA Receptor
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN17779 | Vigabatrin HCl | 1391054-02-6 | Vigabatrin HCl is a structural analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA) that irreversibly inhibits the catabolism of GABA by GABA transaminase. |
| CSN12084 | Tiagabine | 115103-54-3 | Tiagabine is an anti-convulsive medication and a selective gamma-aminobutyric acid (GABA) reuptake inhibitor. |
| CSN12085 | Tiagabine HCl | 145821-59-6 | Tiagabine HCl is an inhibitor of gamma-aminobutyric acid (GABA) reuptake (IC50 = 67 nM in vivo) with anticonvulsant effect. |
| CSN12077 | Thiocolchicoside | 602-41-5 | Thiocolchicoside is a small molecule muscle relaxant and anti-inflammatory agent, shown to function as a competitive GABAA (gamma-aminobutyric acid type A) receptor antagonist. |
| CSN23715 | SAGE-217 | 1632051-40-1 | SAGE-217 is an agonist of GABAA receptor with EC50s of 296 nM and 163 nM for 122 and 43 respectively |
| CSN19798 | Ro 48-6791 | 172407-17-9 | Ro 48-6791 is a GABA receptor agonist potentially for the use of anesthesia |
| CSN10515 | Progabide | 62666-20-0 | Progabide is an analog and prodrug of gamma-aminobutyric acid It is commonly used in the treatment of epilepsy with agonistic activity for both the GABAA and GABAB receptors Progabide has been investigated for many diseases besides epilepsy including Parkinsons disease schizophrenia clinical depression and anxiety disorder with varying success |
| CSN21797 | Pipequaline | 77472-98-1 | Pipequaline is a partial agonist of benzodiazepine receptor (Ki = 78 nM) with anxiolytic activity. |
| CSN11714 | Phytol | 150-86-7 | Phytol can activite PPAR and attenuate the inflammatory response by inhibiting neutrophil migration and oxidative stress. Phytol is isolated from the leaves of black tea and acts as an aromatic ingredient. |
| CSN19514 | Oxiracetam(Random Configuration) | 62613-82-5 | Oxiracetam is a derivative of gamma-aminobutyric acid GABA and used as a nootropic drug to improve memory and learning |
| CSN11488 | Nefiracetam | 77191-36-7 | Nefiracetam is a neuronal systems enhancer for Ro 5-4864-induced convulsions. Nefiracetam has GABAergic, cholinergic, and monoaminergic properties. |
| CSN15900 | NCS-382 Sodium | 131733-92-1 | NCS-382 sodium is a -hydroxybutyric acid antagonist, anticonvulsant. |
| CSN23642 | MRX-1024 | 348-67-4 | MRX-1024 can inhibit the activation of GABAA receptor and exhibit relieving effect on hearing loss It can used as a chemoprotective agent |
| CSN18228 | MRK-016 | 342652-67-9 | MRK-016 is a functionally selective, inverse agonist at the benzodiazepine site of GABAA 5 receptors. |
| CSN19855 | MK 0343 | 233275-76-8 | MK 0343 is a selective partial agonist of GABAA3 1 5 and 2 with Ki values of 021 nM-040 nM It displays anxiolytic activity in rodent and primate models |
| CSN24055 | Loreclezole | 117857-45-1 | Loreclezole is a subtype-selective GABAA receptor modulator. Acts as a positive allosteric modulator of β2 or β3-subunit containing receptors. |
| CSN19849 | Loreclezole HCl | 2227372-56-5 | Loreclezole HCl is a subtype-selective GABAA receptor modulator. Acts as a positive allosteric modulator of β2 or β3-subunit containing receptors. |
| CSN16300 | L-Cycloserine | 339-72-0 | L-cycloserine is an inhibitor of serine palmitoyltransferase and block sphingosine biosynthesis It has antibiotic effective against mycobacterium tuberculosis |
| CSN15698 | L-838,417 | 286456-42-6 | L-838417 is a subtype-selective GABAA receptor partial agonist L-838417 selectively binds to 1 2 3 and 5 subunits Ki values are 079 067 067 and 225 nM respectively but displays no efficacy at 1 1-sparing L-838417 exhibits non-sedative anxiolytic antinociceptive and anti-inflammatory activity |
| CSN20905 | Kavain | 3155-48-4 | Kavain is a positive allosteric modulator of α4β2δ subunit-containing GABAA receptors. |
| CSN21680 | Hypotaurine | 300-84-5 | Hypotaurine, a analog of cystamine, is the precursor for taurine synthesis and can act as an antioxidant and singlet oxygen scavenger. it also acts as an endogenous neurotransmitter via action on the glycine receptors. |
| CSN19501 | Ginsenoside Rc | 11021-14-0 | Ginsenoside Rc is a steroid glycoside, and a triterpene saponin found exclusively in the plant genus Panax (ginseng) with properties that inhibit or prevent tumors growth. |
| CSN12568 | Ginkgolide A | 15291-75-5 | Ginkgolide A is an antagonist of g-aminobutyric acid (GABA) with Ki of 14.5 M and also can activate PAF. It is purified from the leaves of ginkgo biloba tree. |
| CSN10697 | Gelsemine | 509-15-9 | Gelsemine a natural indole alkaloid isolated from flowering plants of the genus Gelsemium with potent activity as an agonist of the mammalian glycine receptor, showing effect on pathwayssystems related to xenobiotic- or diet-induced oxidative stress, and in the treatment of anxiety and other conditions. |
| CSN15872 | Gabazine Hydrobromide | 104104-50-9 | Gabazine hydrobromide is a drug that acts as an antagonist at GABAA receptors It is used in scientific research and has no role in medicine as it would be expected to produce convulsions if used in humans |
| CSN16786 | Flumazenil | 78755-81-4 | Flumazenil is a non-selective antagonist of benzodiazepine towards 1 2 3 or 5-containing GABAA receptors |
| CSN18321 | Etomidate HCl | 53188-20-8 | Etomidate HCl is a GABAA receptors agonist, which is a short acting intravenous anaesthetic agent used for the induction of general anaesthesia. |
| CSN18338 | Etifoxine HCl | 56776-32-0 | Etifoxine HCl is a potentiator of β2 or β3 subunit-containing GABAA receptor that promotes axonal regeneration. It shows anxiolytic activity with no effects. |
| CSN17006 | Emamectin Benzoate | 155569-91-8 | Emamectin benzoate acts as an activator of chloride channel via binding gamma aminobutyric acid GABA receptor and glutamate-gated chloride channels It can disrupt nerve signals in arthropods |
| CSN21616 | Doxefazepam | 40762-15-0 | Doxefazepam is a benzodiazepine medication with anxiolyti and anticonvulsant properties. It is used therapeutically as a hypnotic. |
| CSN17574 | DMCM HCl | 1215833-62-7 | DMCM HCl is benzodiazepine inverse agonist that displays anxiogenic and potent convulsant activity. |
| CSN21600 | Deramciclane | 120444-71-5 | Deramciclane is an antagonist of 5-HT2A and inverse agonist of 5-HT2C receptor. It also functions as a GABA reuptake inhibitor. |
| CSN17089 | Bemegride | 64-65-3 | Bemegride can stimulate central nervous system and release barbiturate poisoning |
| CSN19034 | Basmisanil | 1159600-41-5 | Basmisanil is a selective modulator of GABAA5 with negative allosteric regulation. |
| CSN10524 | Baclofen | 1134-47-0 | Baclofen a gamma-amino-butyric acid derivative is a selective GABAB agonist with IC50 of 200 nM which used as a skeletal muscle relaxant |
| CSN10198 | Acamprosate Calcium | 77337-73-6 | Acamprosate calcium is an agonist of GABA receptor It can act as a modulator of glutamatergic systems and reduce alcohol consumption in animal models of alcohol addiction |
| CSN22026 | 6,2'-Dihydroxyflavone | 92439-20-8 | 6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor. |
| CSN12782 | 4-Aminobutyric Acid | 56-12-2 | 4-Aminobutyric acid exhibits inhibitory activity on central nervous system (CNS). It is a natural neurotransmitter. |
| CSN10435 | (+)-Bicuculline | 485-49-4 | -Bicuculline is an antagonist of GABAA receptor with IC50 of 2 M and also shows inhibition of Ca2-activated potassium channels |
| CSN23429 | L-Glutamic Acid | 56-86-0 | (S)-Glutamic acid acts as an excitatory neurotransmitter in the central nervous system. |
| CSN17026 | (R)-Baclofen | 69308-37-8 | (R)-Baclofen is a derivative of gamma-aminobutyric acid with the selective activation of GABAB receptor that is used to treat spasticity. |
| CSN14755 | (-)-Corlumine | 79082-64-7 | (-)-Corlumine is a natural product isolated and purified from the herbs of Fumaria parviflora with spasmolytic and GABA antagonist activity. |
| CSN23331 | 6-Hydroxyflavone | 6665-83-4 |
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