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Cat. No. Product Name CAS No. Information
CSN11752 Tesmilifene 98774-23-3 Tesmilifene is an agent that augments cytotoxicity of various chemotherapeutic agents both in vitro and in vivo
CSN16637 Tectoridin   611-40-5 Tectoridin, an isoflavone, is a natural product isolated and purified from the rhizomes of belamcanda chinensis (L.) DC. with anti-inflammatory activities.
CSN25280 SR19881 2213490-89-0 SR19881 is a ERRγ agonist.
CSN22304 SNIPER(ER)-110 N/A SNIPERER-110 is a nongenetic IAP-dependent protein eraser SNIPER targeting estrogen receptor ER induces ER degradation and induces apoptosis in MCF-7 human breast cancer cells inhibits the growth of MCF-7 tumor xenografts in mice more potently than the previously characterized SNIPERER-87 preferentially recruits XIAP rather than cIAP1 to degrade ER
CSN23201 Y 134 849662-80-2 Selective estrogen receptor modulator (SERM), selective for ERα
CSN11817 Quinestrol   152-43-2 Quinestrol is a synthetic estrogen which is used in hormone replacement therapy.
CSN17566 Protirelin Acetate 120876-23-5 Protirelin is used to test the response of the anterior pituitary gland.
CSN19099 MGL-3196   920509-32-6 MGL-3196 is a selective thyroid hormone receptor agonist with EC50s of 0.21 and 3.74 M for TR and TR respectively.
CSN11387 Mestranol 72-33-3 Mestranol is an agonist of estrogen receptor. It is used as contraceptives.
CSN24502 MB-07811 852948-13-1 MB-07811 is an orally active HepDirect prodrug of MB07344, a liver-targeted thyroid hormone receptor-β agonist with cholesteroland triglycerides lowering activity.
CSN12274 Liquiritigenin 578-86-9 Liquiritigenin is an estrogenic compound which fuctions as a selective agonist of the estrogen receptor ER and an partial agonist of ER. It also has choleretic effect. Liquiritigenin is a flavanone extracted from glycyrrhiza uralensis with antitumour action.
CSN16424 Licochalcone A 58749-22-7 Licochalcone A an estrogenic flavanoid can be an inhibitor of p-glycoprotein and has anti-inflammatory actions
CSN16955 Lasofoxifene Tartrate 190791-29-8 Lasofoxifene tartrate a non-steroidal compound is a modulator of estrogen receptor
CSN19318 L-Thyroxine Sodium Pentahydrate 6106-07-6 L-Thyroxine sodium is an iodine containing hormone produced from thyroglobulin in the thyroid follicular cells and reduces total cholesterol level, low-density lipoprotein cholesterol as well as waist to hip ratio in subclinical hypothyroidism pateints.
CSN12271 L-Thyroxine   51-48-9 L-Thyroxine is an iodine-containing hormone produced from thyroglobulin in the thyroid follicular cells.
CSN11148 Hexestrol 84-16-2 Hexestrol can bind to ER and ER selectively with EC50 of 007 nM and 0175 nM respectively
CSN22924 H3B-5942 2052128-15-9 H3B-5942 is a selective, irreversible and orally active estrogen receptor covalent antagonist, inactivates both wild-type and mutant ERα by targeting Cys530, with Kis of 1 nM and 0.41 nM, respectively.
CSN16250 Gypenoside XVII 80321-69-3 Gypenoside XVII is a natural product.
CSN19421 Genistin   529-59-9 Genistin is a isoflavone which has a role in blocking cell cycle and inducing apoptosis. It is also a modulator of estrogen receptor. Genistin can be isolated from the seeds of glycine max (L.) merr. and used as negative control of genistein.
CSN21091 GDC-0927 1642297-01-5 GDC-0927, also known as SRN-927, is a next-generation oral SERD, appears to have greater potential than GDC-0810 to be a best-in-class SERD molecule.
CSN24207 GDC-0927 HCl 1642297-02-6 GDC-0927 is a next-generation oral SERD.
CSN10946 Ethisterone   434-03-7 Ethisterone is a progestogen hormone that could be used to treat prostate cancer.
CSN10938 Estropipate   7280-37-7 Estropipate, deriving from estrogen, is used to treat symptoms of menopause and to prevent osteoporosis.
CSN25302 Estrogen receptor modulator 1 63676-22-2 Estrogen receptor modulator 1 is an orally active and selective estrogen receptor modulator (SERM), with a pIC50 of 0.46. It has been found to be both estrogenic and antiproliferative in ER-positive endocrine-resistant breast cancer cell lines that overexpress protein kinase C alpha (PKCα).
CSN10935 Estradiol Benzoate   50-50-0 Estradiol benzoate is an estradiol analog which binds to the human, murine and chicken ER with IC50 of 22-28 nM.
CSN24698 ERRα degrader ligand 4a 2306388-57-6 ERRα degrader ligand 4a block the protein-protein interaction of ERRα with PGC-1α coactivator with IC50 value of 5.67nM in a TR-FRET assay.
CSN22143 ERB-196 550997-55-2 ERB-196 is a nonsteroidal selective estrogen receptor- (ER) agonist.
CSN12284 Equol   531-95-3 Equol, a non-steroidal estrogen, is a selective agonist of ER. It is produced from the metabolism of the isoflavonoid phytoestrogen daidzen by human intestinal microflora.
CSN17408 Endoxifen Z-Isomer HCl 1032008-74-4 Endoxifen Z-isomer HCl is the most important Tamoxifen metabolite responsible for eliciting the anti-estrogenic effects of this drug in breast cancer cells expressing estrogen receptor-alpha (ERα). Endoxifen Z-isomer HCl inhibits hERG tail currents at 50 mV in a concentration-dependent manner with IC50 values of 1.6 μM.
CSN17474 Endoxifen Z-Isomer 112093-28-4 Endoxifen is the most important tamoxifen metabolite responsible for eliciting the anti-estrogenic effects of this drug in breast cancer cells expressing estrogen receptor-alpha ER
CSN17545 Endoxifen E-isomer HCl 1197194-61-8 Endoxifen E-isomer HCl is a tamoxifen metabolite and potent Selective Estrogen Response Modifier (SERM).
CSN10805 Diethylstilbestrol   56-53-1 Diethylstilbestrol is a synthetic nonsteroidal estrogen that produces all the pharmacological and therapeutic effects of natural estradiol It is mainly used for functional hemorrhage caused by estrogen hypoxia and hormonal imbalance amenorrhea
CSN10799 Dienestrol   84-17-3 Dienestrol is an agonist of estrogen receptor which is used for the treatment of menopausal symptoms
CSN17329 Daidzein   486-66-8 Daidzein can act as an inhibitor of tyrosine kinase and an activator of estrogen receptor It is inactive analogue of genistein
CSN14669 Cristacarpin 74515-47-2 Cristacarpin, a natural product isolated and purified from the herbs of Erythrina burana, exhibits moderate but selective activity towards DNA repair-deficient yeast mutants, and promotes endoplasmic reticulum (ER) stress, leading to sub-lethal reactive oxygen species (ROS) generation and which eventually terminates by triggering senescence in pancreatic and breast cancer cells through blocking the cell cycle in the G1 phase.
CSN10623 Chlorotrianisene   569-57-3 Chlorotrianisene, a synthetic and non-steroidal estrogen, is a modulator of estrogen receptor.
CSN12352 Calycosin 20575-57-9 Calycosin, a phytoestrogen, is a partial agonist of ER and a calcium channel blocker. It also shows prevention of reperfusion injury. Calycosin can be isolated and purified from the herb of Astragalus membranaceus Bge. var. mongholicus with anti-oxidative activity.
CSN21522 Bifluranol 34633-34-6 Bifluranol is a synthetic nonsteroidal estrogen of the stilbestrol group related to diethylstilbestrol that has been used as an antiandrogen in the United Kingdom in the treatment of benign prostatic hyperplasia.
CSN18837 Bazedoxifene HCl 198480-56-7 Bazedoxifene is a third generation selective estrogen receptor modulator (SERM).
CSN12297 Bazedoxifene 198481-32-2 Bazedoxifene is a selective estrogen receptor modulator SERM currently in development for osteoporosis prevention and treatment
CSN10382 Bazedoxifene Acetate 198481-33-3 Bazedoxifene acetate can selectively modulate estrogen receptor (SERM), the IC50 values are 26 nM and 99 nM for ER and ER respectively.
CSN22351 Arzoxifene HCl 182133-27-3 Arzoxifene HCl is a selective estrogen receptor modulator that is a potent estrogen antagonist in mammary and uterine tissue while acting as an estrogen agonist to maintain bone density and lower serum cholesterol.
CSN22335 Acolbifene 182167-02-8 Acolbifene (EM652) is a fourth-generation selective estrogen receptor antagonist with a LC50 value of 223 nM.
CSN22105 4-Hydroxytamoxifen 68047-06-3 4-Hydroxytamoxifen is the active metabolite of tamoxifen and a selective estrogen receptor (ER) modulator that is widely used in the therapeutic and chemopreventive treatment of breast cancer.
CSN17213 17-Caproxyprogesterone   630-56-8 17-Caproxyprogesterone is a steroidal progestin. It is a synthetic ester derivative of 17-hydroxyprogesterone.
CSN17211 α-Estradiol 57-91-0 -Estradiol is an endogenous estrogen receptor ligand (Ki values are 0.2 and 1.2 nM for ER and ER receptors respectively).
CSN10426 β-Estradiol 17-acetate 1743-60-8 -Estradiol 17-acetate is a metabolite of estradiol.
CSN21921 (R)-Equol 221054-79-1 (R)-Equol is an agonist of both ERα and ERβ with Kis of 27.4 and 15.4 nM, respectively.
CSN25405 (±)-Equol 94105-90-5
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