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Cat. No. Product Name CAS No. Information
CSN20458 WAY200070 440122-66-7 WAY200070 selectively activates ER EC50 2 nM receptor over ER EC50 155 nM It shows anti-depressive and anti-anxiolytic activities
CSN22522 TR Antagonist 1 500794-88-7 TR antagonist 1 is a high-affinity thyroid hormone receptor TR antagonist with IC50s of 36 and 22 nM for TR and TR respectively
CSN11752 Tesmilifene 98774-23-3 Tesmilifene is an agent that augments cytotoxicity of various chemotherapeutic agents both in vitro and in vivo
CSN16637 Tectoridin   611-40-5 Tectoridin, an isoflavone, is a natural product isolated and purified from the rhizomes of belamcanda chinensis (L.) DC. with anti-inflammatory activities.
CSN22304 SNIPER(ER)-110 N/A SNIPERER-110 is a nongenetic IAP-dependent protein eraser SNIPER targeting estrogen receptor ER induces ER degradation and induces apoptosis in MCF-7 human breast cancer cells inhibits the growth of MCF-7 tumor xenografts in mice more potently than the previously characterized SNIPERER-87 preferentially recruits XIAP rather than cIAP1 to degrade ER
CSN21407 MPP 2HCl 911295-24-4 Selective high affinity silent antagonist at ER receptors Displays 200-fold selectivity for ER over ER Ki values are 27 and 1800 nM at ER and ER receptors respectively
CSN11817 Quinestrol   152-43-2 Quinestrol is a synthetic estrogen which is used in hormone replacement therapy.
CSN17566 Protirelin Acetate 120876-23-5 Protirelin is used to test the response of the anterior pituitary gland.
CSN22305 PAC1 2158322-33-7 PAC1 Compound PAC1 is a PROTAC antibody conjugate more potent estrogen receptor-alpha ER degrader compared to PROTAC without antibody conjugation
CSN21337 Nitromifene 10448-84-7 Nitromifene is an antagonist of estrogen receptor ER
CSN13823 Nafoxidine HCl 1847-63-8 Nafoxidine HCl is a non-steroidal selective estrogen receptor modulator (SERM) or partial antiestrogen of the triphenylethylene group that was developed for the treatment of advanced breast cancer.
CSN19099 MGL-3196 920509-32-6 MGL-3196 is a selective thyroid hormone receptor agonist with EC50s of 0.21 and 3.74 M for TR and TR respectively.
CSN11387 Mestranol 72-33-3 Mestranol is an agonist of estrogen receptor. It is used as contraceptives.
CSN12274 Liquiritigenin 578-86-9 Liquiritigenin is an estrogenic compound which fuctions as a selective agonist of the estrogen receptor ER and an partial agonist of ER. It also has choleretic effect. Liquiritigenin is a flavanone extracted from glycyrrhiza uralensis with antitumour action.
CSN16955 Lasofoxifene Tartrate 190791-29-8 Lasofoxifene tartrate a non-steroidal compound is a modulator of estrogen receptor
CSN19318 L-Thyroxine Sodium Pentahydrate 6106-07-6 L-Thyroxine sodium is an iodine containing hormone produced from thyroglobulin in the thyroid follicular cells and reduces total cholesterol level, low-density lipoprotein cholesterol as well as waist to hip ratio in subclinical hypothyroidism pateints.
CSN12271 L-Thyroxine   51-48-9 L-Thyroxine is an iodine-containing hormone produced from thyroglobulin in the thyroid follicular cells.
CSN11148 Hexestrol 84-16-2 Hexestrol can bind to ER and ER selectively with EC50 of 007 nM and 0175 nM respectively
CSN22924 H3B-5942 2052128-15-9 H3B-5942 is a selective, irreversible and orally active estrogen receptor covalent antagonist, inactivates both wild-type and mutant ERα by targeting Cys530, with Kis of 1 nM and 0.41 nM, respectively.
CSN16250 Gypenoside XVII 80321-69-3 Gypenoside XVII is a natural product.
CSN19421 Genistin   529-59-9 Genistin is a isoflavone which has a role in blocking cell cycle and inducing apoptosis. It is also a modulator of estrogen receptor. Genistin can be isolated from the seeds of glycine max (L.) merr. and used as negative control of genistein.
CSN10938 Estropipate   7280-37-7 Estropipate, deriving from estrogen, is used to treat symptoms of menopause and to prevent osteoporosis.
CSN10935 Estradiol Benzoate   50-50-0 Estradiol benzoate is an estradiol analog which binds to the human, murine and chicken ER with IC50 of 22-28 nM.
CSN22143 ERB-196 550997-55-2 ERB-196 is a nonsteroidal selective estrogen receptor- (ER) agonist.
CSN12284 Equol   531-95-3 Equol, a non-steroidal estrogen, is a selective agonist of ER. It is produced from the metabolism of the isoflavonoid phytoestrogen daidzen by human intestinal microflora.
CSN17408 Endoxifen Z-Isomer HCl 1032008-74-4 Endoxifen Z-isomer HCl is the most important Tamoxifen metabolite responsible for eliciting the anti-estrogenic effects of this drug in breast cancer cells expressing estrogen receptor-alpha (ERα). Endoxifen Z-isomer HCl inhibits hERG tail currents at 50 mV in a concentration-dependent manner with IC50 values of 1.6 μM.
CSN17474 Endoxifen Z-Isomer 112093-28-4 Endoxifen is the most important tamoxifen metabolite responsible for eliciting the anti-estrogenic effects of this drug in breast cancer cells expressing estrogen receptor-alpha ER
CSN17545 Endoxifen E-isomer HCl 1197194-61-8 Endoxifen E-isomer HCl is a tamoxifen metabolite and potent Selective Estrogen Response Modifier (SERM).
CSN10799 Dienestrol   84-17-3 Dienestrol is an agonist of estrogen receptor which is used for the treatment of menopausal symptoms
CSN17329 Daidzein   486-66-8 Daidzein can act as an inhibitor of tyrosine kinase and an activator of estrogen receptor It is inactive analogue of genistein
CSN10623 Chlorotrianisene   569-57-3 Chlorotrianisene, a synthetic and non-steroidal estrogen, is a modulator of estrogen receptor.
CSN12352 Calycosin   20575-57-9 Calycosin, a phytoestrogen, is a partial agonist of ER and a calcium channel blocker. It also shows prevention of reperfusion injury. Calycosin can be isolated and purified from the herb of Astragalus membranaceus Bge. var. mongholicus with anti-oxidative activity.
CSN21522 Bifluranol 34633-34-6 Bifluranol is a synthetic nonsteroidal estrogen of the stilbestrol group related to diethylstilbestrol that has been used as an antiandrogen in the United Kingdom in the treatment of benign prostatic hyperplasia.
CSN12297 Bazedoxifene 198481-32-2 Bazedoxifene is a selective estrogen receptor modulator SERM currently in development for osteoporosis prevention and treatment
CSN10382 Bazedoxifene Acetate 198481-33-3 Bazedoxifene acetate can selectively modulate estrogen receptor (SERM), the IC50 values are 26 nM and 99 nM for ER and ER respectively.
CSN17980 AZD9496 1639042-08-2 AZD9496 is a selective antagonist of estrogen receptor Er IC50 028 nM
CSN22351 Arzoxifene HCl 182133-27-3 Arzoxifene HCl is a selective estrogen receptor modulator that is a potent estrogen antagonist in mammary and uterine tissue while acting as an estrogen agonist to maintain bone density and lower serum cholesterol.
CSN22335 Acolbifene 182167-02-8 Acolbifene (EM652) is a fourth-generation selective estrogen receptor antagonist with a LC50 value of 223 nM.
CSN17211 α-Estradiol 57-91-0 -Estradiol is an endogenous estrogen receptor ligand (Ki values are 0.2 and 1.2 nM for ER and ER receptors respectively).
CSN10426 β-Estradiol 17-acetate 1743-60-8 -Estradiol 17-acetate is a metabolite of estradiol.
CSN21921 (R)-Equol 221054-79-1 (R)-Equol is an agonist of both ERα and ERβ with Kis of 27.4 and 15.4 nM, respectively.
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