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Endothelin Receptor

Endothelin Receptor

Cat. No. Product Name CAS No. Information
CSN13675 Zibotentan 186497-07-4 Zibotentan is an orally administered potent and specific ETA-receptor endothelin A receptor antagonist IC50 21 nM
CSN12014 Sulfisoxazole   127-69-5 Sulfisoxazole is an antagonist of endothelin receptor that can be used as a sulfonamide antibacterial agent
CSN24483 Ro 46-8443 175556-12-4 Ro 46-8443 is the first non-peptide Endothelin Receptor B selective antagonist with IC50 value of 110nM.
CSN17902 Ro 46-2005 150725-87-4 Ro 46-2005 is an antagonist of endothelin receptor
CSN25744 IRL-2500 169545-27-1 IRL-2500 is a potent endothelin receptor antagonist with IC50 values of 1.3 and 94 nM for ETB and ETA receptors respectively.
CSN23533 Darusentan   171714-84-4 Darusentan is an antagonist of endothelin ETA receptor and it can be used to treat congestive heart failure and hypertension
CSN17753 BQ-123 136553-81-6 BQ-123 is a specific antagonist of endothelin A receptor ETA and the IC50 is 73 nM
CSN13753 Atrasentan HCl 195733-43-8 Atrasentan HCl is an endothelin receptor antagonist (IC50=0.0551 nM, ETA) being developed for the treatment of prostate cancer.
CSN10496 Ambrisentan   177036-94-1 Ambrisentan is an oral, once-daily endothelin receptor antagonist that is selective for the endothelin type A receptor (IC50s 0.251, 0.316, 0.398, 251, and 630 nM for rat preparations of heart, bladder, kidney, lung, and cerebral cortex, respectively).
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