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Endothelin Receptor
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN13675 | Zibotentan | 186497-07-4 | Zibotentan is an orally administered potent and specific ETA-receptor endothelin A receptor antagonist IC50 21 nM |
| CSN29551 | ZD-1611 | 186497-38-1 | ZD1611 is an endothelin receptor antagonist. |
| CSN12014 | Sulfisoxazole | 127-69-5 | Sulfisoxazole is an antagonist of endothelin receptor that can be used as a sulfonamide antibacterial agent |
| CSN11008 | Sodium Ferulate | 24276-84-4 | Sodium ferulate is the sodium salt of ferulic acid which is used for the treatment of cardiovascular disease |
| CSN12974 | Sitaxsentan Sodium | 210421-74-2 | Sitaxsentan sodium has selectory antagonism of endothelin A ETA receptor with the IC50 and Ki value of 14 nM and 043 nM respectively |
| CSN12975 | Sitaxsentan | 184036-34-8 | Sitaxsentan is a selective endothelin A (ETA) receptor antagonist. |
| CSN24483 | Ro 46-8443 | 175556-12-4 | Ro 46-8443 is the first non-peptide Endothelin Receptor B selective antagonist with IC50 value of 110nM. |
| CSN17902 | Ro 46-2005 | 150725-87-4 | Ro 46-2005 is an antagonist of endothelin receptor |
| CSN25744 | IRL-2500 | 169545-27-1 | IRL-2500 is a potent endothelin receptor antagonist with IC50 values of 1.3 and 94 nM for ETB and ETA receptors respectively. |
| CSN23533 | Darusentan | 171714-84-4 | Darusentan is an antagonist of endothelin ETA receptor and it can be used to treat congestive heart failure and hypertension |
| CSN19760 | Clazosentan | 180384-56-9 | Clazosentan is a potent endothelin A antagonist, improves cerebral blood flow and behavior after traumatic brain injury. |
| CSN17348 | BQ-788 Sodium | 156161-89-6 | BQ-788 sodium salt is a potent selective ETB receptor antagonist with IC50 of 12 nM for inhibition of ET-1 binding to human Girardi heart cells poorly inhibiting the binding to ETA receptors in human neuroblastoma cell line SK-N-MC cells with IC50 of 1300 nM |
| CSN17753 | BQ-123 | 136553-81-6 | BQ-123 is a specific antagonist of endothelin A receptor ETA and the IC50 is 73 nM |
| CSN10481 | Bosentan Hydrate | 157212-55-0 | Bosentan is an endothelin (ET) receptor antagonist of ET-A (Ki 4.7 nM) and ET-B (Ki 95 nM). |
| CSN10480 | Bosentan | 147536-97-8 | Bosentan is an endothelin (ET) receptor antagonist for ET-A and ET-B with Ki of 4.7 nM and 95 nM, respectively. |
| CSN18015 | Atrasentan | 173937-91-2 | Atrasentan is an endothelin receptor antagonist (IC500.0551 nM, ETA) being developed for the treatment of prostate cancer. |
| CSN13753 | Atrasentan HCl | 195733-43-8 | Atrasentan HCl is an endothelin receptor antagonist (IC50=0.0551 nM, ETA) being developed for the treatment of prostate cancer. |
| CSN10496 | Ambrisentan | 177036-94-1 | Ambrisentan is an oral, once-daily endothelin receptor antagonist that is selective for the endothelin type A receptor (IC50s 0.251, 0.316, 0.398, 251, and 630 nM for rat preparations of heart, bladder, kidney, lung, and cerebral cortex, respectively). |
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