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Endothelin Receptor
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN13675 | Zibotentan | 186497-07-4 | Zibotentan is an orally administered potent and specific ETA-receptor endothelin A receptor antagonist IC50 21 nM |
| CSN12014 | Sulfisoxazole | 127-69-5 | Sulfisoxazole is an antagonist of endothelin receptor that can be used as a sulfonamide antibacterial agent |
| CSN24483 | Ro 46-8443 | 175556-12-4 | Ro 46-8443 is the first non-peptide Endothelin Receptor B selective antagonist with IC50 value of 110nM. |
| CSN17902 | Ro 46-2005 | 150725-87-4 | Ro 46-2005 is an antagonist of endothelin receptor |
| CSN25744 | IRL-2500 | 169545-27-1 | IRL-2500 is a potent endothelin receptor antagonist with IC50 values of 1.3 and 94 nM for ETB and ETA receptors respectively. |
| CSN23533 | Darusentan | 171714-84-4 | Darusentan is an antagonist of endothelin ETA receptor and it can be used to treat congestive heart failure and hypertension |
| CSN17753 | BQ-123 | 136553-81-6 | BQ-123 is a specific antagonist of endothelin A receptor ETA and the IC50 is 73 nM |
| CSN13753 | Atrasentan HCl | 195733-43-8 | Atrasentan HCl is an endothelin receptor antagonist (IC50=0.0551 nM, ETA) being developed for the treatment of prostate cancer. |
| CSN10496 | Ambrisentan | 177036-94-1 | Ambrisentan is an oral, once-daily endothelin receptor antagonist that is selective for the endothelin type A receptor (IC50s 0.251, 0.316, 0.398, 251, and 630 nM for rat preparations of heart, bladder, kidney, lung, and cerebral cortex, respectively). |
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