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Dopamine Receptor

Dopamine Receptor

Cat. No. Product Name CAS No. Information
CSN11417 Trifluoperazine 2HCl   440-17-5 Trifluoperazine 2HCl is a dopamine D2 receptor inhibitor with anti-dopaminergic and anti-adrenergic actions, which belongs to the phenothiazine compounds.
CSN16278 Tetrahydropalmatine   2934-97-6 Tetrahydropalmatine is an isoquinoline alkaloid mainly found in the genus Corydalis with analgesic effects It antagonizes dopamine D1 and D2 receptors as well as actions at dopamine D3 alpha adrenergic and serotonin receptors with Ki values of 124 nM and 388 nM for D1 and D2 dopamine receptors respectively
CSN25548 Tavapadon 1643489-24-0 Tavapadon is an orally active and highly selective dopamine D1/D5 receptor partial agonist. It may be useful in the treatment of Parkinson's disease and Alzheimer's.
CSN12723 Sumanirole Maleate 179386-44-8 Sumanirole maleate is a highly selective D2 receptor full agonist with an ED50 of about 46 nM.
CSN21847 Sultopride 53583-79-2 Sultopride is a selective antagonist of dopamine D2 receptor.
CSN16852 SKF-82958 80751-65-1 SKF-82958 is a D1D5 receptor full agonist.
CSN18415 SKF-82958 Hydrobromide 74115-01-8 SKF-82958 hydrobromide is a D1D5 receptor full agonist.
CSN13576 SKF-38393 HCl   62717-42-4 SKF-38393 HCl is an agonist of dopamine D1 receptor (the IC50 value is 110 nM). It has anorectic and stimulant effects.
CSN25662 SKF 77434 104422-04-0 SKF 77434 is Dopamine D1 receptor partial agonist. Chronic treatment with SKF 77434 produced dose-dependent effects on cocaine self-administration in Rhesus Monkeys.
CSN13078 Ropinirole HCl   91374-20-8 Ropinirole HCl selectively inhibit dopamine D2 receptor with Ki of 29 nM. It is used for the treatment of spontaneous parkinson's disease.
CSN11783 Promazine HCl 53-60-1 Promazine HCl is a D2 dopamine receptor antagonist, belongs to the phenothiazine class of antipsychotics, used to treat schizophrenia.
CSN16556 Prochlorperazine Dimaleate   84-02-6 Prochlorperazine dimaleate is an antagonist of dopamine (D2) receptor with Ki value of 4.7 nM.
CSN10895 Pergolide Mesylate 66104-23-2 Pergolide mesylate is an antiparkinsonian agent which functions as a dopaminergic agonist.
CSN11681 Pergolide 66104-22-1 Pergolide is an ergoline-based dopamine receptor agonist used in some countries for the treatment of Parkinsons disease
CSN23235 PD-168077 190383-31-4 PD168,077 is a dopamine D4 receptor agonist which has a facilitatory effect on memory consolidation.
CSN13887 PD 128907 HCl 112960-16-4 PD 128907 HCl is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 nM, exhibits 53-fold selectivity over dopamine D2 receptor.
CSN18173 Pardoprunox HCl 269718-83-4 Pardoprunox HCl is a partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) and D3 receptor (pKi = 8.6) partial agonist and 5-HT1A receptor (pKi = 8.5) full agonist.
CSN11617 Oroxylin A 480-11-5 Oroxylin A shows inhibition of the dopamine reuptake and allosteric modulation of GABAA receptor. It is a natural active flavonoid isolated from scutellaria baicalensis and oroxylum indicum.
CSN11546 Neuromedin N 92169-45-4 Neuromedin N is a potent modulator of dopamine D2 receptor agonist binding in rat neostriatal membranes
CSN11472 Mosapramine 89419-40-9 Mosapramine is an atypical antipsychotic used in Japan It is a potent dopamine antagonist with high affinity to the D2 D3 and D4 receptors and with moderate affinity for the 5-HT2 receptors
CSN11461 Molindone HCl   15622-65-8 Molindone HCl the salt form of molindone which is a dopamine receptor antagonist can be used in the treatment of schizophrenia and act as a therapeutic antipsychotic
CSN11425 Metoclopramide   364-62-5 Metoclopramide is an antagonist of dopamine D2 and is commonly used as an antiemetic
CSN11426 Metoclopramide HCl 7232-21-5 Metoclopramide HCl is a selective dopamine D2 receptor antagonist, used for the treatment of nausea and vomiting.
CSN11390 Metergoline 17692-51-2 Metergoline is a psychoactive drug of the ergoline chemical class which acts as a ligand for various serotonin and dopamine receptors
CSN23832 Mesoridazine Besylate 32672-69-8 Mesoridazine besylate is a phenothiazine dopamine receptor anatagonist. Mesoridazine besylate is described to demonstrate inhibition for D2DR and D4DR. It has a high affinity for dopamine D4 receptor. Mesoridazine besylate is an antipsychotic agent.
CSN16179 L-Stepholidine 16562-13-3 L-Stepholidine is a naturally occurring chemical compound isolated and purfied from the roots of Stephania japonica. L-Stepholidine is a dual D2 receptor antagonist and D1 receptor agonist.
CSN25316 L-745870 158985-00-3 L-745870 is a high-affinity, selective and orally active human dopamine D4 receptor antagonist with a Ki of 0.43 nM and excellent brain penetration.
CSN15992 Flupenthixol 2HCl   51529-01-2 Flupenthixol 2HCl, a typical antipsychotic drug, is non-selective antagonist of dopamine D1-5 receptors as well as 5-HT2A. It is also known as flupenthixol.
CSN11002 Fenoldopam Mesylate   67227-57-0 Fenoldopam mesylate is a partial specific agonist of D1 receptor, a synthetic benzoxipine derivative.
CSN10871 Droperidol   548-73-2 Droperidol is an antagonist of dopamine-2 receptor.
CSN22033 Dixyrazine 2470-73-7 Dixyrazine, a phenothiazine derivative, can prevent brain oedema induced by intracarotid injection of protamine sulphate.
CSN12899 Dexpramipexole 104632-28-2 Dexpramipexole is a neuroprotective agent and weak non-ergoline dopamine agonist.
CSN17422 Dexpramipexole 2HCl   104632-27-1 Dexpramipexole 2HCl is the HCl form of Dexpramipexole which is a non-ergoline dopamine agonist for treatment of parkinson's disease and restless leg syndrome.Dexpramipexole is an (R)-(+) optical enantiomer of pramipexole.
CSN21571 Clocapramine 47739-98-0 Clocapramine is D2 5-HT2A receptors antagonist.
CSN19084 CGP-25454A 104391-26-6 CGP 25454A is a selective presynaptic dopamine autoreceptor antagonist.
CSN16030 Cariprazine 839712-12-8 Cariprazine exhibits high selectivity and affinity to dopamine D3 receptor Ki009 nM and lower binding activity to dopamine D2 receptor and 5-HT1A with Ki of 05 nM and 26 nM repectively It has been used as antipsychotics in the treatment of schizophrenia and bipolar disorder
CSN10446 B-HT 920 36085-73-1 B-HT 920 is a dopamine D2 receptor agonist 2-adrenoceptor agonist and 5-HT3 receptor antagonist which displays antiParkinsonian activity
CSN12577 Azaperone   1649-18-9 Azaperone functions as a dopamine antagonist that can bind to D1 and D2 receptors. It has the characteristics of antihistamines and anticholinergics.
CSN24171 Ansofaxine HCl 916918-84-8 Ansofaxine HCl is a multiple-target reuptake inhibitor with IC50 values of 723nM, 491nM and 763nM for serotonin, dopamine and norepinephrine reuptake.
CSN10288 Amisulpride   71675-85-9 Amisulpride is a selective dopamine antagonist wit Ki of 28 nM for D2 receptor and Ki of 32 nM D3 receptor its used as an antipsychotic drug
CSN10011 Amantadine HCl   665-66-7 Amantadine HCl is an antiviral and an antiparkinsonian drug. It is used to treat or prevent infections of the respiratory tract caused by a certain virus.
CSN10242 Alizapride 59338-93-1 Alizapride is a dopamine antagonist with prokinetic and antiemetic effects used in the treatment of nausea and vomiting including postoperative nausea and vomiting
CSN10243 Alizapride HCl   59338-87-3 Alizapride HCl is a dopamine receptor antagonist used in the administration of nausea and vomiting
CSN25294 ABT-724 70006-24-5 ABT-724 is a potent and highly selective dopamine D4 receptor agonist with EC50s of 12.4 nM, 14.3 nM and 23.2 nM for human dopamine D4 receptor, rat D4 receptor and ferret D4 receptor.
CSN25293 ABT-724 3HCl 587870-77-7 ABT-724 3HCl is a potent and highly selective dopamine D4 receptor agonist with EC50s of 12.4 nM, 14.3 nM and 23.2 nM for human dopamine D4 receptor, rat D4 receptor and ferret D4 receptor.
CSN21450 Abaperidone 183849-43-6 Abaperidone is an antagonist of 5-HT2A receptor and dopamine D2 receptor with IC50s of 6.2 and 17 nM respectively.
CSN24069 A-381393 726174-00-1 A-381393 is a potent, selective, brain penetrate dopamine D4 receptor antagonist, with Kis of 1.5, 1.9 and 1.6 nM for human dopamine D4.4, D4.2, and D4.7 receptor, respectively, >2700-fold selectivity over D1, D2, D3 and D5 dopamine receptors. A-381393 shows moderate affinity for 5-HT2A (Ki, 370 nM)[1].
CSN13176 (-)-Isocorypalmine 483-34-1 (-)-Isocorypalmine, a natural product isolated and purified from the tubers of Corydalis yanhusuo W. T. Wang, with significant antifungal activity, also acts as a D1 partial agonist and a D2 antagonist to produce its in vivo effects and may be a promising agent for treatment of cocaine addiction.
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