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CRTH2
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN24302 | MK-7246 | 1218918-62-7 | MK-7246 is a potent and selective CRTH2 antagonist with Ki value of 2.5nM. |
| CSN20221 | MK-2305 | 2101206-49-7 | MK-2305 is a GPR40 partial agonist lower fasting glucose in the Goto Kakizaki rat via suppression of endogenous glucose production |
| CSN18830 | Fevipiprant | 872365-14-5 | Fevipiprant is a selective potent reversible competitive CRTh2 antagonist with an in vitro dissociation constant KD value of 11nM at the CRTh2 receptor and an IC50 value of 044 nM for inhibition of PGD2-induced eosinophil shape change in human whole blood |
| CSN22382 | CRTh2 antagonist 1 | 1379445-54-1 | CRTh2 antagonist 1是 CRTh2 的拮抗剂，IC50 值为89 nM。 |
| CSN26623 | CAY10471 Racemate | 844639-57-2 | CAY 10471 is a potent, highly selective CRTH2/DP 2 receptor antagonist. CAY10471 binds to the human CRTH2/DP2, DP1, and TP receptors with Ki values of 0.6, 1200, and >10,000 nM. Cat#531655 is a racemic mixture of CAY10471. |
| CSN16482 | AZD1981 | 802904-66-1 | AZD1981 is a potent and selective CRTh2 antagonist and displaces radio-labelled PGD2 from human recombinant DP2 with high potency (pIC50 8.4). |
| CSN22681 | Vidupiprant | 1169483-24-2 | AMG 853 is a potent dual CRTH2 and prostaglandin D2 (PGD2) receptor antagonist (IC50 values are 8 and 35 nM, respectively in plasma). |
| CSN25231 | AM211 | 1175526-27-8 | AM211 is a potent and selective prostaglandin D2 receptor type 2 antagonist with IC50 value of 4.9nM. |
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