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CRTH2

CRTH2

Cat. No. Product Name CAS No. Information
CSN24302 MK-7246     1218918-62-7 MK-7246 is a potent and selective CRTH2 antagonist with Ki value of 2.5nM.
CSN20221 MK-2305 2101206-49-7 MK-2305 is a GPR40 partial agonist lower fasting glucose in the Goto Kakizaki rat via suppression of endogenous glucose production
CSN18830 Fevipiprant   872365-14-5 Fevipiprant is a selective potent reversible competitive CRTh2 antagonist with an in vitro dissociation constant KD value of 11nM at the CRTh2 receptor and an IC50 value of 044 nM for inhibition of PGD2-induced eosinophil shape change in human whole blood
CSN16482 AZD1981     802904-66-1 AZD1981 is a potent and selective CRTh2 antagonist and displaces radio-labelled PGD2 from human recombinant DP2 with high potency (pIC50 8.4).
CSN22681 AMG 853 1169483-24-2 AMG 853 is a potent dual CRTH2 and prostaglandin D2 (PGD2) receptor antagonist (IC50 values are 8 and 35 nM, respectively in plasma).
CSN25231 AM211 1175526-27-8 AM211 is a potent and selective prostaglandin D2 receptor type 2 antagonist with IC50 value of 4.9nM.
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