Chemokine Receptor | GPCR/G Protein|Immunology/Inflammation| CSNpharm

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Cat. No.	Product Name	CAS No.	Information
CSN12197	Vicriviroc Maleate	599179-03-0	Vicriviroc maleate is a CCR5 antagonist with IC50 of 0.91 nM in clinical development for the treatment of HIV-1.
CSN18397	Vercirnon	698394-73-9	Vercirnon is a highly potent antagonist of CCR9, which has been implicated in the aetiology of inflammatory bowel diseases such as Crohns disease.
CSN16904	TAK-220	333994-00-6	TAK-220 is an orally bioavailable small-molecule CCR5 antagonist
CSN22613	SB297006	58816-69-6	SB297006 is a selective antagonist of CCR3 with IC50 of 39 nM
CSN18192	RS-102895	300815-41-2	RS102895 is a potent and specific CCR2 antagonist with binding IC50 of 360 nM, no significant inhibition on CCR1 (IC50 17 M).
CSN13797	RS-102895 HCl	1173022-16-6	RS102895 hydrochloride is a potent and specific CCR2 antagonist with binding IC50 of 360 nM, no significant inhibition on CCR1 (IC50 17 M).
CSN12845	RS-504393	300816-15-3	RS 504393 is a selective CCR2 chemokine receptor antagonist (IC50 values are 98 nM and 100 M for inhibition of human recombinant CCR2b and CCR1 receptors respectively).
CSN17712	PF-4136309	1341224-83-6	PF-4136309 is a potent, Selective, and orally bioavailable CCR2 antagonist.
CSN17807	NSC 5844	140926-75-6	NSC 5844 is a bisquinoline compound with C-C chemokine receptor type 1 CCR1-agonistic properties
CSN18995	MK-0812 Succinate	851916-42-2	MK-0812 succinate is a potent and selective CCR2 antagonist with low nM affinity for CCR2 on human monocytes
CSN13664	MK-0812	624733-88-6	MK-0812 is a potent and selective CCR2 antagonist with low nM affinity for CCR2 on human monocytes.
CSN11361	Maraviroc	376348-65-1	Maraviroc is a selective CCR5 antagonist (IC50 6.4 nM) and displays potent anti-HIV-1 activity.
CSN17640	INCB3344	1262238-11-8	INCB3344 is a potent and selective small molecule antagonist of the mouse CCR2 receptor and inhibits the binding of CCL2 to mouse monocytes with nanomolar potency (IC50 10 nM).
CSN13799	INCB 3284 Dimesylate	887401-93-6	INCB 3284 is a potent, selective and orally bioavailable hCCR2 antagonist with IC50 of 3.7 nM.
CSN18528	INCB 3284	887401-92-5	INCB 3284 is a potent, selective and orally bioavailable hCCR2 antagonist with IC50 of 3.7 nM (inhibition of monocyte chemoattractant protein-1 binding to hCCR2).
CSN22186	GW 766994	408303-43-5	GW 766994 is a specific and oral chemokine receptor-3 (CCR3) antagonist, which has entered clinical trial for asthma and eosinophilic bronchitis.
CSN22234	GSK2239633A	1240516-71-5	GSK2239633A is a CC-chemokine receptor 4 CCR4 antagonist which inhibits the binding of 125I-TARC to human CCR4 with a pIC50 of 796011
CSN23233	DAPTA	106362-34-9	DAPTA is a potent and selective CCR5 antagonist
CSN15987	Cenicriviroc	497223-25-3	Cenicriviroc is an oral, dual CCR2CCR5 antagonist, and displays potent anti-inflammatory and aninfective activity.
CSN22175	CCR5 Antagonist 1	716354-86-8	CCR5 antagonist 1 is a CCR5 antagonist which can inhibit HIV replication extracted from WO 2004054974 A2
CSN18114	BX471	217645-70-0	BX471 is a potent, selective non-peptide CCR1 antagonist (Ki 1 nM for human CCR1) and exhibits 250-fold selectivity for CCR1 over CCR2, CCR5 and CXCR4.
CSN18182	BX471 HCl	288262-96-4	BX471 hydrochloride is a potent, selective non-peptide CCR1 antagonist (Ki 1 nM for human CCR1) and exhibits 250-fold selectivity for CCR1 over CCR2, CCR5 and CXCR4.
CSN20665	AZD-2098	566203-88-1	AZD2098 is a potent CC-chemokine receptor 4 (CCR4) inhibitor, used for asthma research.
CSN20666	AZD-1678	942137-41-9	AZD1678 is a potent CC-chemokine receptor 4 (CCR4) inhibitor, used for asthma research.
CSN22732	C 021 2HCl	864289-85-0
CSN22729	BX 513 HCl	1216540-18-9
CSN22720	BMS CCR2 22	445479-97-0
CSN23102	SB 328437	247580-43-4
CSN23164	Teijin Compound 1	1313730-14-1

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