Welcome to CSNpharm! For Research Use Only!

CCR

CCR

Cat. No. Product Name CAS No. Information
CSN12197 Vicriviroc Maleate 599179-03-0 Vicriviroc maleate is a CCR5 antagonist with IC50 of 0.91 nM in clinical development for the treatment of HIV-1.
CSN16904 TAK-220 333994-00-6 TAK-220 is an orally bioavailable small-molecule CCR5 antagonist
CSN22613 SB297006   58816-69-6 SB297006 is a selective antagonist of CCR3 with IC50 of 39 nM
CSN12845 RS-504393 300816-15-3 RS 504393 is a selective CCR2 chemokine receptor antagonist (IC50 values are 98 nM and 100 M for inhibition of human recombinant CCR2b and CCR1 receptors respectively).
CSN23164 Teijin Compound 1 1313730-14-1 Potent CCR2b antagonist
CSN17712 PF-4136309 1341224-83-6 PF-4136309 is a potent, Selective, and orally bioavailable CCR2 antagonist.
CSN17807 NSC 5844 140926-75-6 NSC 5844 is a bisquinoline compound with C-C chemokine receptor type 1 CCR1-agonistic properties
CSN11361 Maraviroc 376348-65-1 Maraviroc is a selective CCR5 antagonist (IC50 6.4 nM) and displays potent anti-HIV-1 activity.
CSN17640 INCB3344 1262238-11-8 INCB3344 is a potent and selective small molecule antagonist of the mouse CCR2 receptor and inhibits the binding of CCL2 to mouse monocytes with nanomolar potency (IC50 10 nM).
CSN23233 DAPTA   106362-34-9 DAPTA is a potent and selective CCR5 antagonist
CSN22175 CCR5 Antagonist 1 716354-86-8 CCR5 antagonist 1 is a CCR5 antagonist which can inhibit HIV replication extracted from WO 2004054974 A2
CSN18114 BX471 217645-70-0 BX471 is a potent, selective non-peptide CCR1 antagonist (Ki 1 nM for human CCR1) and exhibits 250-fold selectivity for CCR1 over CCR2, CCR5 and CXCR4.
CSN18182 BX471 HCl 288262-96-4 BX471 HCl is a potent, selective non-peptide CCR1 antagonist (Ki = 1 nM for human CCR1) and exhibits 250-fold selectivity for CCR1 over CCR2, CCR5 and CXCR4.
<< PREV 1 NEXT >>