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Casein Kinase
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN15858 | TTP 22 | 329907-28-0 | TTP 22 is a high affinity ATP-competitive casein kinase 2 CK2 inhibitor with IC50Ki of 01 M40 nM showing selectivity for CK2 over JNK3 ROCK1 and MET IC50 10 M |
| CSN25710 | TMCB | 905105-89-7 | TMCB is a dual-kinase inhibitor of both casein kinase 2 (CK2) and extracellular-signal-regulated kinase 8 (ERK8) with IC50s of 0.50 μM. |
| CSN19438 | TBB | 17374-26-4 | TBB is a highly selective ATPGTP-competitive inhibitor of casein kinase-2 CK2with IC50s of 09 and 16 M for rat liver and human recombinant CK2 respectively |
| CSN18028 | TA-01 | 1784751-18-3 | TA-01 potently inhibits CK1 CK1and p38 IC50values are 64 68 and 67 nM respectively |
| CSN17879 | SR-3029 | 1454585-06-8 | SR-3029 is a potent and highly specific CK1CK1 inhibitor with the IC50 of 97 nM |
| CSN26213 | PI-828 | 942289-87-4 | PI-828 is a dual PI3K and casein kinase 2 (CK2) inhibitor with IC50s of 173 nM, 149 nM, and 1127 nM for p110α, CK2, and CK2α2 in lipid kinase assay, respectively. |
| CSN16518 | PF-670462 | 950912-80-8 | PF-670462 is a potent and selective inhibitor of CK1 with IC50 of 77 22 nM |
| CSN22941 | PF-4800567 | 1188296-52-7 | PF-4800567 is an inhibitor of casein kinase 1 CK1 with IC50 of 32 nM |
| CSN22893 | PF-4800567 HCl | 1391052-28-0 | PF-4800567 HCl is a selective casein kinase 1ε inhibitor with IC50 of 32 nM. |
| CSN24190 | NCC007 | 2342583-66-6 | NCC007 is a dual CK1α and CK1δ inhibitor with IC50 value of 1.8 and 3.6μM, respectively. |
| CSN11346 | LY294002 | 154447-36-6 | LY294002 is the first synthetic molecule known to inhibit PI3Kα/δ/β with IC50 of 0.5 μM/0.57 μM/0.97 μM in cell-free assays. It is an early-stage autophagy inhibitor and also inhibits CK2. |
| CSN16329 | LH846 | 639052-78-1 | LH846 is a selective inhibitor of casein kinase CK 1 with IC50 of 290 nM 13 M and 25 M for CK1 and displays no inhibitory activity at CK2 |
| CSN18054 | IC261 | 186611-52-9 | IC261 is an ATP-competitive inhibitor of CK1 with IC50s about 1 M for CK1 and CK1 16 M for CK1 |
| CSN19160 | H-89 dihydrochloride | 130964-39-5 | H 89 2HCl is a potent and selective inhibitor of cyclic AMP-dependent protein kinase (protein kinase A) with IC50 of 48 nM. It also shows weak inhibition on PKG, PKC, CK1, CK2 and others kinases. |
| CSN19160 | H-89 dihydrochloride | 130964-39-5 | H 89 2HCl is a potent and selective inhibitor of cyclic AMP-dependent protein kinase (protein kinase A) with IC50 of 48 nM. It also shows weak inhibition on PKG, PKC, CK1, CK2 and others kinases. |
| CSN63435 | (E/Z)-GO289 | 694522-87-7 | GO289 is a potent and selective CK2 inhibitor. |
| CSN26540 | CK2/PIM1-IN-1 | 292640-28-9 | for CK2 and PIM1, respectively. CK2/PIM1-IN-1 is developed for the research of proliferative disorders such as cancer, as well as other kinase-associated conditions including inflammation, pain, vascular disorders, pathogenic infections and certain immunological disorders[1]. |
| CSN18468 | Emodin | 518-82-1 | Emodin shows antiproliferative effects in cancer cells that are regulated by different signaling pathways it is a naturally occurring anthraquinone present in the roots and barks of numerous plants |
| CSN10902 | Ellagic acid | 476-66-4 | Ellagic acid is a potent and cell permeable casein kinase 2 (CK2) inhibitor with Ki of 20 nM, acts as a potent antioxidant and anti-mutagenic. |
| CSN16246 | DMAT | 749234-11-5 | DMAT is a potent and specific CK2 inhibitor with an IC50 value of 130 nM |
| CSN13638 | D4476 | 301836-43-1 | D4476 is a potent selective and cell-permeant CK1 casein kinase 1 inhibitor with IC50 of 200 nM and 300 nM in a cell-free assay for CK1 from Schizosaccharomyces pombe and CK1 respectively Also acts as an ALK5 inhibitor with IC50 of 500 nM |
| CSN17673 | Silmitasertib sodium salt | 1309357-15-0 | CX-4945 Sodium is a selective inhibitor of CK2 catalytic subunits with an IC50 value of 1 nmolL. |
| CSN12957 | Silmitasertib | 1009820-21-6 | CX-4945 is a potent and selective ATP-competitive small molecule protein kinase CK2 inhibitor with a Ki and an IC50 of 038 and 1 nM for recombinant human CK2 respectively |
| CSN23747 | CK1-IN-1 | 1784751-20-7 | CK1-IN-1 is a casein kinase 1 (CK1) inhibitor extracted from patent WO2015119579A1, compound 1c, has IC50s of 15 nM, 16 nM, 73 nM for CK1δ, and CK1ε, p38σ MAPK, respectively[1]. |
| CSN21284 | Casein Kinase II Inhibitor IV | 863598-09-8 | Casein Kinase II Inhibitor IV is a small-molecule inducer of epidermal keratinocyte differentiation |
| CSN20162 | CAM4066 | 2101206-81-7 | CAM4066 is a selective Casein Kinase 2 CK2 inhibitor |
| CSN27228 | BioE-1115 | 1268863-35-9 | BioE-1115 is a highly selective and potent PAS kinase (PASK) inhibitor with an IC50 of ~4 nM. BioE-1115 is also a potent casein kinase 2α inhibitor with an IC50 of ~10 μM . |
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