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Cannabinoid Receptor
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN21516 | β-Caryophyllene | 87-44-5 | β-Caryophyllene is an agonist of the cannabinoid (CB) receptor CB2 with Ki of 155 nM. |
| CSN13453 | MDA 19 | 1048973-47-2 | MDA 19 is a selective human CB2 receptor agonist with Ki of 433 nM |
| CSN25339 | MAFP | 188404-10-6 | MAFP is a potent, irreversible inhibitor of fatty acid amide hydrolase (FAAH, anandamide amidase), the enzyme responsible for anandamide hydrolysis (IC50 = 2.5 nM). MAFP also binds irreversibly to CB1 receptors with IC50 of 20 nM. |
| CSN19472 | LY320135 | 176977-56-3 | LY-320135 is a potent and selective Canniboid CB1 receptor antagonistinverse agonist. LY-320135 is selective (70 fold) over Canniboid CB2 receptors. This compound shows weak binding to both 5-HT2 (Ki 6.4 M) and muscarinic receptors (Ki 2.1 M). |
| CSN20218 | JD5037 | 1392116-14-1 | JD-5037 is a peripherally restricted CB1R antagonist with an IC50 of 15 nM |
| CSN21228 | CB2R-IN-1 | 1257555-79-5 | CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 09 nM |
| CSN10473 | BML-190 | 2854-32-2 | BML-190 is a selective cannabinoid CB2 receptor inverse agonist with Ki of 435 nM, with 50-fold selectivity over CB1 receptor. |
| CSN10421 | beta-Amyrin | 559-70-6 | beta-Amyrin, a natural cannabinoid receptors agonist isolated and purified from the stem bark of Alstonia boonei, has anti-inflammatory activity. Beta-Amyrin significantly inhibits PGE2, IL-6 secretion, and NF-B activation in a concentration-dependent manner on LPS-induced hPBMCs. |
| CSN18739 | BAY 59-3074 | 406205-74-1 | Bay 59-3074 is a selective CB1CB2 receptor partial agonist with Kis of 483 and 455 nM at human CB1 and CB2 receptors respectively |
| CSN25672 | Arvanil | 128007-31-8 | Arvanil is an antagonist of cannabinoid CB1 and vanilloid TRPV1 (VR1) with Ki values are 0.5 and 0.3 μM respectively. |
| CSN21999 | (±)-SLV319 | 362519-49-1 | -SLV319 is a selective antagonist of cannabinoid-1 CB1 receptor with Ki value of 78 nM and it has a weaker activation effect on CB2 |
| CSN15641 | (+)-Gallocatechin | 970-73-0 | -Gallocatechin a natural product isolated and purified from the wood of Acacia catechu LF Willd has moderate affinity to the human cannabinoid receptor |
| CSN12783 | (-)-Gallocatechin | 3371-27-5 | --Gallocatechin a natural product isolated and purified from the wood of Acacia catechu LF Willd has moderate affinity to the human cannabinoid receptor |
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