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Cannabinoid Receptor
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN21516 | β-Caryophyllene | 87-44-5 | β-Caryophyllene is an agonist of the cannabinoid (CB) receptor CB2 with Ki of 155 nM. |
| CSN12285 | Yangonin | 500-62-9 | Yangonin, a natural product isolated and purified from the roots of Piper methysticum, possess significant binding affinity for the cannabinoid receptor CB1 and inhibits NF-B activation through suppression of the transcriptional activity of the RelAp65 subunit of NF-B. |
| CSN25626 | TM38837 | 1253641-65-4 | TM38837 is a novel, largely peripherally restricted CB1 antagonist with limited penetrance to the brain. Oral dose of TM38837 (100 mg/kg) induced a significant increase in freezing behavior. |
| CSN24663 | PF 514273 | 851728-60-4 | PF 514273 is a selective CB1 receptor antagonist with Ki values of 1 and > 10000 nM at CB1 and CB2 receptors respectively. |
| CSN24683 | OMDM-2 | 616884-63-0 | OMDM-2 is a stable and selective inhibitor of anandamide cellular uptake with Ki of 3 μM. |
| CSN25339 | MAFP | 188404-10-6 | MAFP is a potent, irreversible inhibitor of fatty acid amide hydrolase (FAAH, anandamide amidase), the enzyme responsible for anandamide hydrolysis (IC50 = 2.5 nM). MAFP also binds irreversibly to CB1 receptors with IC50 of 20 nM. |
| CSN19472 | LY320135 | 176977-56-3 | LY-320135 is a potent and selective Canniboid CB1 receptor antagonistinverse agonist. LY-320135 is selective (70 fold) over Canniboid CB2 receptors. This compound shows weak binding to both 5-HT2 (Ki 6.4 M) and muscarinic receptors (Ki 2.1 M). |
| CSN24684 | JTE-907 | 282089-49-0 | JTE 907 is a highly selective cannabinoid CB2 receptor inverse agonist that binds with high affinity to rat, mouse and human CB2 receptors with Ki of 0.38, 1.55 and 35.9 nM respectively. |
| CSN20218 | JD-5037 | 1392116-14-1 | JD-5037 is a peripherally restricted CB1R antagonist with an IC50 of 15 nM |
| CSN19173 | GW842166X | 666260-75-9 | GW842166X is a potent and highly selective agonist of cannabinoid receptor CB2 receptor with EC50 of 63 nM shows no significant activity at CB1 receptor |
| CSN21228 | CB2R-IN-1 | 1257555-79-5 | CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 09 nM |
| CSN20330 | CB2 Agonist C8 | 2052602-31-8 | CB2 agonist C8 is an agonists of cannabinoid receptor type 2 |
| CSN20331 | CB2 Agonist C36 | 2097512-96-2 | CB2 agonist C36 is an agonists of cannabinoid receptor type 2 |
| CSN17330 | CB1-IN-1 | 1429239-98-4 | CB1-IN-1 is a peripherally restricted CB1R antagonist, with Ki of 0.3 nM and 21 nM for CB1R (EC50 = 3 nM) and CB2R, respectively. |
| CSN10473 | BML-190 | 2854-32-2 | BML-190 is a selective cannabinoid CB2 receptor inverse agonist with Ki of 435 nM, with 50-fold selectivity over CB1 receptor. |
| CSN25672 | Arvanil | 128007-31-8 | Arvanil is an antagonist of cannabinoid CB1 and vanilloid TRPV1 (VR1) with Ki values are 0.5 and 0.3 μM respectively. |
| CSN24665 | CB1 antagonist 2 | 614726-85-1 | AM 4113 is selective CB1 antagonist with Kd of 0.89 nM. |
| CSN12783 | (-)-Gallocatechin | 3371-27-5 | --Gallocatechin a natural product isolated and purified from the wood of Acacia catechu LF Willd has moderate affinity to the human cannabinoid receptor |
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