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Cannabinoid Receptor

Cannabinoid Receptor

Cat. No. Product Name CAS No. Information
CSN21516 β-Caryophyllene 87-44-5 β-Caryophyllene is an agonist of the cannabinoid (CB) receptor CB2 with Ki of 155 nM.
CSN12285 Yangonin 500-62-9 Yangonin, a natural product isolated and purified from the roots of Piper methysticum, possess significant binding affinity for the cannabinoid receptor CB1 and inhibits NF-B activation through suppression of the transcriptional activity of the RelAp65 subunit of NF-B.
CSN25626 TM38837 1253641-65-4 TM38837 is a novel, largely peripherally restricted CB1 antagonist with limited penetrance to the brain. Oral dose of TM38837 (100 mg/kg) induced a significant increase in freezing behavior.
CSN24663 PF 514273 851728-60-4 PF 514273 is a selective CB1 receptor antagonist with Ki values of 1 and > 10000 nM at CB1 and CB2 receptors respectively.
CSN24683 OMDM-2 616884-63-0 OMDM-2 is a stable and selective inhibitor of anandamide cellular uptake with Ki of 3 μM.
CSN25339 MAFP 188404-10-6 MAFP is a potent, irreversible inhibitor of fatty acid amide hydrolase (FAAH, anandamide amidase), the enzyme responsible for anandamide hydrolysis (IC50 = 2.5 nM). MAFP also binds irreversibly to CB1 receptors with IC50 of 20 nM.
CSN19472 LY320135 176977-56-3 LY-320135 is a potent and selective Canniboid CB1 receptor antagonistinverse agonist. LY-320135 is selective (70 fold) over Canniboid CB2 receptors. This compound shows weak binding to both 5-HT2 (Ki 6.4 M) and muscarinic receptors (Ki 2.1 M).
CSN24684 JTE-907 282089-49-0 JTE 907 is a highly selective cannabinoid CB2 receptor inverse agonist that binds with high affinity to rat, mouse and human CB2 receptors with Ki of 0.38, 1.55 and 35.9 nM respectively.
CSN20218 JD-5037 1392116-14-1 JD-5037 is a peripherally restricted CB1R antagonist with an IC50 of 15 nM
CSN19173 GW842166X 666260-75-9 GW842166X is a potent and highly selective agonist of cannabinoid receptor CB2 receptor with EC50 of 63 nM shows no significant activity at CB1 receptor
CSN21228 CB2R-IN-1 1257555-79-5 CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 09 nM
CSN20330 CB2 Agonist C8 2052602-31-8 CB2 agonist C8 is an agonists of cannabinoid receptor type 2
CSN20331 CB2 Agonist C36 2097512-96-2 CB2 agonist C36 is an agonists of cannabinoid receptor type 2
CSN17330 CB1-IN-1 1429239-98-4 CB1-IN-1 is a peripherally restricted CB1R antagonist, with Ki of 0.3 nM and 21 nM for CB1R (EC50 = 3 nM) and CB2R, respectively.
CSN10473 BML-190   2854-32-2 BML-190 is a selective cannabinoid CB2 receptor inverse agonist with Ki of 435 nM, with 50-fold selectivity over CB1 receptor.
CSN25672 Arvanil 128007-31-8 Arvanil is an antagonist of cannabinoid CB1 and vanilloid TRPV1 (VR1) with Ki values are 0.5 and 0.3 μM respectively.
CSN24665 CB1 antagonist 2 614726-85-1 AM 4113 is selective CB1 antagonist with Kd of 0.89 nM.
CSN12783 (-)-Gallocatechin 3371-27-5 --Gallocatechin a natural product isolated and purified from the wood of Acacia catechu LF Willd has moderate affinity to the human cannabinoid receptor
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