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Cannabinoid Receptor

Cannabinoid Receptor

Cat. No. Product Name CAS No. Information
CSN21516 β-Caryophyllene 87-44-5 β-Caryophyllene is an agonist of the cannabinoid (CB) receptor CB2 with Ki of 155 nM.
CSN24663 PF 514273 851728-60-4 PF 514273 is a selective CB1 receptor antagonist with Ki values of 1 and > 10000 nM at CB1 and CB2 receptors respectively.
CSN24683 OMDM-2 616884-63-0 OMDM-2 is a stable and selective inhibitor of anandamide cellular uptake with Ki of 3 μM.
CSN13453 MDA 19 1048973-47-2 MDA 19 is a selective human CB2 receptor agonist with Ki of 433 nM
CSN25339 MAFP 188404-10-6 MAFP is a potent, irreversible inhibitor of fatty acid amide hydrolase (FAAH, anandamide amidase), the enzyme responsible for anandamide hydrolysis (IC50 = 2.5 nM). MAFP also binds irreversibly to CB1 receptors with IC50 of 20 nM.
CSN19472 LY320135 176977-56-3 LY-320135 is a potent and selective Canniboid CB1 receptor antagonistinverse agonist. LY-320135 is selective (70 fold) over Canniboid CB2 receptors. This compound shows weak binding to both 5-HT2 (Ki 6.4 M) and muscarinic receptors (Ki 2.1 M).
CSN24684 JTE 907 282089-49-0 JTE 907 is a highly selective cannabinoid CB2 receptor inverse agonist that binds with high affinity to rat, mouse and human CB2 receptors with Ki of 0.38, 1.55 and 35.9 nM respectively.
CSN20218 JD5037 1392116-14-1 JD-5037 is a peripherally restricted CB1R antagonist with an IC50 of 15 nM
CSN19173 GW842166X 666260-75-9 GW842166X is a potent and highly selective agonist of cannabinoid receptor CB2 receptor with EC50 of 63 nM shows no significant activity at CB1 receptor
CSN24670 DEA 150314-35-5 DEA is endocannabinoid and anandamide analog that activates CB1 receptors in microglia and can bind to rat synaptosomal membranes (Ki = 34.4 nM).
CSN21228 CB2R-IN-1 1257555-79-5 CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 09 nM
CSN10473 BML-190   2854-32-2 BML-190 is a selective cannabinoid CB2 receptor inverse agonist with Ki of 435 nM, with 50-fold selectivity over CB1 receptor.
CSN27633 BAY-38-7271 212188-60-8 BAY 38-7271 is selective agonist of cannabinoid CB1/CB2 receptor with Kis of 1.85 nM and 5.96 nM respectively. It has strong neuroprotective properties.
CSN25672 Arvanil 128007-31-8 Arvanil is an antagonist of cannabinoid CB1 and vanilloid TRPV1 (VR1) with Ki values are 0.5 and 0.3 μM respectively.
CSN24665 AM 4113 614726-85-1 AM 4113 is selective CB1 antagonist with Kd of 0.89 nM.
CSN24666 ACPA 229021-64-1 ACPA is a selective agonist of CB1 with Ki of 2.2 nM.
CSN21999 (±)-SLV319   362519-49-1 -SLV319 is a selective antagonist of cannabinoid-1 CB1 receptor with Ki value of 78 nM and it has a weaker activation effect on CB2
CSN15641 (+)-Gallocatechin 970-73-0 -Gallocatechin a natural product isolated and purified from the wood of Acacia catechu LF Willd has moderate affinity to the human cannabinoid receptor
CSN12783 (-)-Gallocatechin 3371-27-5 --Gallocatechin a natural product isolated and purified from the wood of Acacia catechu LF Willd has moderate affinity to the human cannabinoid receptor
CSN24668 (R)-(+)-Methanandamide 157182-49-5 (R)-(+)-Methanandamide, the stable anandamide analog, is a selective agonist for the CB1 receptor with Ki values of 20 and 815 nM for CB1 and CB2 receptors respectively.
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