Cannabinoid Receptor

Cannabinoid Receptor

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Cat. No.	Product Name	CAS No.	Information
CSN21516	β-Caryophyllene	87-44-5	β-Caryophyllene is an agonist of the cannabinoid (CB) receptor CB2 with Ki of 155 nM.
CSN18972	Taranabant (1R,2R)stereoisomer	701977-08-4	Taranabant1R2Rstereoisomer is the R-Enantiomer of taranabant Taranabant is a highly potent and selective cannabinoid 1 CB1 receptor inverse agonist
CSN12382	Taranabant	701977-09-5	Taranabant is a cannabinoid 1 receptor inverse agonist with IC50 of 03 nM
CSN22151	MK-9470	947371-30-4	MK-9470 is a selective high-affinity inverse agonist human IC5007 nM for the cannabinoid CB1 receptor CB1R developed for use in human brain imaging
CSN13453	MDA 19	1048973-47-2	MDA 19 is a selective human CB2 receptor agonist with Ki of 433 nM
CSN25339	MAFP	188404-10-6	MAFP is a potent, irreversible inhibitor of fatty acid amide hydrolase (FAAH, anandamide amidase), the enzyme responsible for anandamide hydrolysis (IC50 = 2.5 nM). MAFP also binds irreversibly to CB1 receptors with IC50 of 20 nM.
CSN19472	LY320135	176977-56-3	LY-320135 is a potent and selective Canniboid CB1 receptor antagonistinverse agonist. LY-320135 is selective (70 fold) over Canniboid CB2 receptors. This compound shows weak binding to both 5-HT2 (Ki 6.4 M) and muscarinic receptors (Ki 2.1 M).
CSN20218	JD5037	1392116-14-1	JD-5037 is a peripherally restricted CB1R antagonist with an IC50 of 15 nM
CSN19173	GW842166X	666260-75-9	GW842166X is a potent and highly selective agonist of cannabinoid receptor CB2 receptor with EC50 of 63 nM shows no significant activity at CB1 receptor
CSN21228	CB2R-IN-1	1257555-79-5	CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 09 nM
CSN20330	CB2 Agonist C8	2052602-31-8	CB2 agonist C8 is an agonists of cannabinoid receptor type 2
CSN20331	CB2 Agonist C36	2097512-96-2	CB2 agonist C36 is an agonists of cannabinoid receptor type 2
CSN17330	CB1-IN-1	1429239-98-4	CB1-IN-1 is a peripherally restricted CB1R antagonist, with Ki of 0.3 nM and 21 nM for CB1R (EC50 = 3 nM) and CB2R, respectively.
CSN20616	Cannabidivarin	24274-48-4	Cannabidivarin is a non-psychoactive cannabinoid found in Cannabis that activates CB2 cannabinoid receptors as well as the transient receptor potential channels TRPA1, TRPV1, and TRPV2 (EC50s 0.42, 3.6, and 7.3 M, respectively). It is also reported to antagonize TRPM8 (IC50 0.9 M) and to inhibit diacylglycerol lipase (IC50 16.6 M).
CSN10421	beta-Amyrin	559-70-6	beta-Amyrin, a natural cannabinoid receptors agonist isolated and purified from the stem bark of Alstonia boonei, has anti-inflammatory activity. Beta-Amyrin significantly inhibits PGE2, IL-6 secretion, and NF-B activation in a concentration-dependent manner on LPS-induced hPBMCs.
CSN15642	beta-Amyrin Acetate	1616-93-9	beta-Amyrin acetrate, a natural cannabinoid receptor isolated and purified from the herbs of Alstonia boone, shows significant HMG-CoA-reductase and sEH inhibitory activities.
CSN18739	BAY 59-3074	406205-74-1	Bay 59-3074 is a selective CB1CB2 receptor partial agonist with Kis of 483 and 455 nM at human CB1 and CB2 receptors respectively
CSN21999	(±)-SLV319	362519-49-1	-SLV319 is a selective antagonist of cannabinoid-1 CB1 receptor with Ki value of 78 nM and it has a weaker activation effect on CB2
CSN15641	(+)-Gallocatechin	970-73-0	-Gallocatechin a natural product isolated and purified from the wood of Acacia catechu LF Willd has moderate affinity to the human cannabinoid receptor
CSN12783	(-)-Gallocatechin	3371-27-5	--Gallocatechin a natural product isolated and purified from the wood of Acacia catechu LF Willd has moderate affinity to the human cannabinoid receptor

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Cannabinoid Receptor

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