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Cannabinoid Receptor

Cannabinoid Receptor

Cat. No. Product Name CAS No. Information
CSN21516 β-Caryophyllene 87-44-5 β-Caryophyllene is an agonist of the cannabinoid (CB) receptor CB2 with Ki of 155 nM.
CSN13453 MDA 19 1048973-47-2 MDA 19 is a selective human CB2 receptor agonist with Ki of 433 nM
CSN25339 MAFP 188404-10-6 MAFP is a potent, irreversible inhibitor of fatty acid amide hydrolase (FAAH, anandamide amidase), the enzyme responsible for anandamide hydrolysis (IC50 = 2.5 nM). MAFP also binds irreversibly to CB1 receptors with IC50 of 20 nM.
CSN19472 LY320135 176977-56-3 LY-320135 is a potent and selective Canniboid CB1 receptor antagonistinverse agonist. LY-320135 is selective (70 fold) over Canniboid CB2 receptors. This compound shows weak binding to both 5-HT2 (Ki 6.4 M) and muscarinic receptors (Ki 2.1 M).
CSN20218 JD5037 1392116-14-1 JD-5037 is a peripherally restricted CB1R antagonist with an IC50 of 15 nM
CSN21228 CB2R-IN-1 1257555-79-5 CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 09 nM
CSN10473 BML-190   2854-32-2 BML-190 is a selective cannabinoid CB2 receptor inverse agonist with Ki of 435 nM, with 50-fold selectivity over CB1 receptor.
CSN10421 beta-Amyrin 559-70-6 beta-Amyrin, a natural cannabinoid receptors agonist isolated and purified from the stem bark of Alstonia boonei, has anti-inflammatory activity. Beta-Amyrin significantly inhibits PGE2, IL-6 secretion, and NF-B activation in a concentration-dependent manner on LPS-induced hPBMCs.
CSN18739 BAY 59-3074 406205-74-1 Bay 59-3074 is a selective CB1CB2 receptor partial agonist with Kis of 483 and 455 nM at human CB1 and CB2 receptors respectively
CSN25672 Arvanil 128007-31-8 Arvanil is an antagonist of cannabinoid CB1 and vanilloid TRPV1 (VR1) with Ki values are 0.5 and 0.3 μM respectively.
CSN21999 (±)-SLV319   362519-49-1 -SLV319 is a selective antagonist of cannabinoid-1 CB1 receptor with Ki value of 78 nM and it has a weaker activation effect on CB2
CSN15641 (+)-Gallocatechin 970-73-0 -Gallocatechin a natural product isolated and purified from the wood of Acacia catechu LF Willd has moderate affinity to the human cannabinoid receptor
CSN12783 (-)-Gallocatechin 3371-27-5 --Gallocatechin a natural product isolated and purified from the wood of Acacia catechu LF Willd has moderate affinity to the human cannabinoid receptor
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