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c-RET

c-RET

Cat. No. Product Name CAS No. Information
CSN25546 Selpercatinib 2152628-33-4 Selpercatinib is a potent and specific RET inhibitor with IC50 values of 1 nM, 2 nM, 2 nM, 4 nM, 2 nM, 2 nM for WT RET, RET V804M, RET V804L, RET A883F, RET M918T and RET S891A respectively.
CSN13099 Regorafenib 755037-03-7 Regorafenib is a multi-target inhibitor for VEGFR123, PDGFR, Kit, RET and Raf-1 with IC50 of 134.246 nM, 22 nM, 7 nM, 1.5 nM and 2.5 nM, respectively.
CSN23893 LOXO-292 2222755-14-6 LOXO-292 is a selective and potent RET inhibitor and an investigational drug in clinical development for the treatment of patients with cancers that harbor abnormalities in the rearranged during transfection (RET) kinase.
CSN24470 GSK3179106   1627856-64-7 GSK3179106 is a potent, selective and gut-restricted RET kinase inhibitor with IC50 value of 0.4nM.
CSN22922 BLU-667 2097132-94-8 Blu667 is a highly potent and selective RET inhibitor with IC50 value of 0.4nM.
CSN19120 BBT594 882405-89-2 BBT594 is a potentreceptor tyrosine kinase RET inhibitor, used for cancer treatment.
CSN18365 AST-487 630124-46-8 AST-487 is a RET kinase inhibitor with IC50 of 880 nM inhibits RET autophosphorylation and activation of downstream effectors also inhibits Flt-3 with IC50 of 520 nM
CSN22316 AD80   1384071-99-1 AD80 is a multikinase inhibitor with inhibitions onRETRAF SRC andS6K
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