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Bradykinin Receptor

Bradykinin Receptor

Cat. No. Product Name CAS No. Information
CSN21187 SSR240612 464930-42-5 SSR240612 is a potent and selective non-peptide bradykinin B1 receptor antagonist with Kis of 0.48 nM and 0.73 nM for B1 kinin receptors of human fibroblast MRC5 and HEK cells expressing human B1 receptors, 481 nM and 358 nM for B2 receptors of guinea pig ileum membranes and CHO cells expressing human B1 receptor, respectively.
CSN24645 R 715 185052-09-9 R 715 is a selective bradykinin B1 receptor antagonist with pA2 of 8.49 with no activity at B2 receptor.
CSN24303 Lobradimil 159768-75-9 Labradimil, also known as RMP 7, is a bradykinin B2 receptor agonist potentially for the treatment of brain cancer. RMP-7) increases the permeability of human brain microvascular endothelial cell monolayers. RMP-7 enhances delivery of hydrophilic chemotherapeutics and increases survival in rats with metastatic tumors in the brain. RMP-7 increases carboplatin levels in brain tumors after pretreatment with dexamethasone.
CSN11154 Icatibant 130308-48-4 Icatibant is a selective and specific antagonist of bradykinin B2 receptor with IC50 and Ki of 107 nM and 0798 nM respectively
CSN23822 Icatibant Acetate 138614-30-9 Icatibant acetate (HOE-140 acetate) is a potent and specific peptide antagonist of bradykinin B2 receptor with IC50 and Ki of 1.07 nM and 0.798 nM respectively.
CSN21292 FR167344 215258-13-2 FR167344 free base is an orally active, nonpeptide bradykinin receptor B2 antagonist. FR167344 free base shows a high affinity binding to the B2 receptor with an IC50value of 65 nM and no binding affinity for the B1 receptor.
CSN18567 ELN-441958 913064-47-8 ELN-441958 is a potent neutral antagonist of B1 receptor inhibits the binding of the B1 agonist ligand 3HDAKD to IMR-90 cells with Ki of 026 nM
CSN21812 Bradykinin 2-9 16875-11-9 Bradykinin 2-9, an amino-truncated bradykinin peptide, is a metabolite of bradykinin with no detectable contractile activity. It can inhibit ACE and potentiate BK.
CSN22721 Bombinakinin M 509151-65-9 Bombinakinin M is a potent bradykinin receptor agonist.
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