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Bradykinin Receptor

Bradykinin Receptor

Cat. No. Product Name CAS No. Information
CSN21187 SSR240612 464930-42-5 SSR240612 is a potent and selective non-peptide bradykinin B1 receptor antagonist with Kis of 0.48 nM and 0.73 nM for B1 kinin receptors of human fibroblast MRC5 and HEK cells expressing human B1 receptors, 481 nM and 358 nM for B2 receptors of guinea pig ileum membranes and CHO cells expressing human B1 receptor, respectively.
CSN21292 FR167344 free base 215258-13-2 FR167344 free base is an orally active, nonpeptide bradykinin receptor B2 antagonist. FR167344 free base shows a high affinity binding to the B2 receptor with an IC50value of 65 nM and no binding affinity for the B1 receptor.
CSN18567 ELN-441958 913064-47-8 ELN-441958 is a potent neutral antagonist of B1 receptor inhibits the binding of the B1 agonist ligand 3HDAKD to IMR-90 cells with Ki of 026 nM
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