Bombesin Receptor
Cat. No. | Product Name | CAS No. | Information |
---|---|---|---|
CSN21385 | PD176252 | 204067-01-6 | PD176252 is a potent antagonist of neuromedin-B preferring BB1 and gastrin-releasing peptide-preferring BB2 receptor with Kis of 017 nM and 1 nM for human BB1 and BB2 receptors and 066 nM 16 nM for Rat BB1 and BB2 receptors respectively also an agonist of N-Formyl peptide receptor12 FPR1FPR2 with EC50s of 031 and 066 M in HL-60 cells |
CSN24208 | ML-18 | 1422269-30-4 | ML-18 is a nonpeptide BRS-3 antagonist with IC50 value of 4.8μM. |
CSN17401 | MK-5046 | 1022152-70-0 | MK-5046 is a BRS-3 agonist, binds to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM). |