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Bombesin Receptor

Bombesin Receptor

Cat. No. Product Name CAS No. Information
CSN21385 PD176252 204067-01-6 PD176252 is a potent antagonist of neuromedin-B preferring BB1 and gastrin-releasing peptide-preferring BB2 receptor with Kis of 017 nM and 1 nM for human BB1 and BB2 receptors and 066 nM 16 nM for Rat BB1 and BB2 receptors respectively also an agonist of N-Formyl peptide receptor12 FPR1FPR2 with EC50s of 031 and 066 M in HL-60 cells
CSN24208 ML-18   1422269-30-4 ML-18 is a nonpeptide BRS-3 antagonist with IC50 value of 4.8μM.
CSN17401 MK-5046 1022152-70-0 MK-5046 is a BRS-3 agonist, binds to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM).
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