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Aurora Kinase

Aurora Kinase

Cat. No. Product Name CAS No. Information
CSN12727 ZM447439 331771-20-1 ZM 447439 is a selective and ATP-competitive inhibitor for Aurora A and Aurora B with IC50 of 110 nM 130 nM respectively 8 fold selectivity than Aurora C MEK1 Src
CSN12326 Tozasertib     639089-54-6 Tozasertib is the inhibitor of Aurora-A, -B, -C kinases with Ki values of 0.6, 18, 4.6 nM respectively.
CSN16128 TAK-901 934541-31-8 TAK-901 is an inhibitor of Aurora AB with IC50 of 21 nM15 nM
CSN18798 SNS-314 Mesylate 1146618-41-8 SNS-314 is a potent and selective inhibitor of Aurora A Aurora B and Aurora C with IC50 of 9 nM 31 nM and 3 nM respectively
CSN13118 SCH-1473759 1094069-99-4 SCH-1473759 is a sub-nanomolar Aurora AB inhibitor with IC50 of 4 nM and 13 nM respectively
CSN17462 SCH-1473759 HCl 1094067-13-6 SCH-1473759 hydrochloride is a sub-nanomolar Aurora AB inhibitor with IC50 of 4 nM and 13 nM respectively
CSN15807 Reversine   656820-32-5 Reversine a synthetic purine analogue26-disubstituted purine is a potent human A3 adenosine receptor antagonist with Ki of 066 M and a pan-aurora ABC kinase inhibitor with IC50 of 12 nM13 nM20 nM respectively
CSN12811 PHA-680632 398493-79-3 PHA-680632 is potent inhibitor of Aurora A B and C with IC50 of 27 nM 135 nM and 120 nM respectively
CSN18615 PF-03814735 942487-16-3 PF-03814735 is a potent orally bioavailable reversible small-molecule Aurora kinase inhibitor with IC50 of 08 5 10 and 22 nM for Aurora A Aurora B Flt 1 and FAk respectively
CSN12363 MLN8054 869363-13-3 MLN8054 is a potent and selective inhibitor of Aurora A with IC50 of 4 nM and exhibits more than 40-fold selective for Aurora A than Aurora B
CSN16817 MK-8745 885325-71-3 MK-8745 is a potent and selective Aurora an inhibitor with IC50 of 06 nM more than 450-fold selectivity for Aurora A over Aurora B
CSN17389 MK-5108 1010085-13-8 MK-5108 is a potent and highly selective Aurora inhibitor with IC50 of 0064 14 and 12 nM for Aurora A B and C
CSN13761 Hesperadin 422513-13-1 Hesperadin is a potent and ATP-competitive inhibitor of Aurora B kinase with IC50 of 250 nM
CSN12395 GSK1070916 942918-07-2 GSK1070916 is a reversible and ATP-competitive inhibitor of Aurora BC with IC50 of 35 nM65 nM and displays 100-fold selectivity against the closely related Aurora A-TPX2 complex IC50490 nM
CSN12423 Danusertib   827318-97-8 Danusertib is a pyrrolo-pyrazole and small molecule Aurora kinases inhibitor with IC50 of 13 79 and 61 nM for Aurora A B and C respectively
CSN17118 CYC-116   693228-63-6 CYC116 is a potent inhibitor of Aurora with Ki of 80 nM92 nM for Aurora AB
CSN17149 CCT137690 1095382-05-0 CCT137690 is a potent inhibitor of Aurora kinases IC50 values are 0015 0019 and 0025 M at Aurora A Aurora C and Aurora B respectively
CSN16415 CCT129202 942947-93-5 CCT129202 is a Aurora kinase inhibitor with IC50 of 0042 0022 0198 005 and 0227 0064 M for Aurora A Aurora B and Aurora C respectively
CSN16205 BI-847325 1207293-36-4 BI-847325 is a selective and orally bioavailable dual MEKAurora kinase inhibitor with IC50 of 3 nM Xenopus laevis Aurora B 25 nM human Aurora A 15 nM human Aurora C 25 nM human MEK1 and 4 nM human MEK2 respectively
CSN17268 AZD1152-HQPA 722544-51-6 AZD1152-HQPA is the active metabolite of AZD-1152 and a highly selective Aurora B inhibitor with IC50 of 0.37 nM, 100 fold selective for Aurora B over Aurora A.
CSN12380 TC-S 7010 1158838-45-9 Aurora an inhibitor I is a potent and selective inhibitor of Aurora A with IC50 of 34 nM in a cell-free assay It is 1000-fold selective for Aurora A than Aurora B
CSN12715 AT9283 896466-04-9 AT9283 is a multi-targeted inhibitor with IC50s of 4 12 11 and approximate 3 nM for Bcr-Abl T315I JAK2 and JAK3 Aurora A and Aurora B respectively
CSN16543 AMG-900 945595-80-2 AMG-900 is a potent and highly selective pan-Aurora kinases inhibitor for Aurora ABC with IC50 of 5 nM4 nM 1 nM and is 10-fold selective for Aurora kinases than p38 Tyk2 JNK2 Met and Tie2
CSN13457 Alisertib   1028486-01-2 Alisertib is a selective Aurora inhibitor with IC50 of 12 nM with 200-fold higher selectivity for Aurora A than Aurora B
CSN23149 TC-A 2317 HCl 1245907-03-2
CSN23770 Aurora Kinase Inhibitor III 879127-16-9
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