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Androgen Receptor

Androgen Receptor

Cat. No. Product Name CAS No. Information
CSN21357 YK11 1370003-76-1 YK11 is a partial agonist of androgen receptor with osteogenic activity
CSN12743 RU 58841   154992-24-2 RU 58841 is a nonsteroidal antiandrogen for potential use as a topical treatment for androgen-dependent conditions including acne, pattern hair loss, and excessive hair growth.
CSN19838 RD 162 915087-27-3 RD 162 is an orally active and very potent antagonist of androgen receptor AR and is a second-generation of antiandrogen for the treatment of advanced prostate cancer and highly recommended tool in AR research
CSN17523 RAD140 1182367-47-0 RAD140 is a potent orally bioavailable nonsteroidal selective androgen receptor modulator SARM
CSN17663 ORM-15341 1297537-33-7 ORM-15341 is a potent and full antagonist for human AR hAR with IC50 values of 38 nM as shown by transactivation assays in AR-HEK293 cells stably expressing full-length hAR and an androgen-responsive luciferase reporter gene construct
CSN17664 ODM-201 1297538-32-9 ODM-201 is a competitive inhibitor of androgen receptor with IC50 value of 26 nM and inhibits AR nuclear translocation with Ki value of 11 nM.
CSN13442 Nomegestrol 58691-88-6 Nomegestrol is a steroidal progestin
CSN16774 Nilutamide   63612-50-0 Nilutamide is a non-steroidal androgen receptor antagonist and also inhibits androgen biosynthesis in vitro
CSN17614 N-desmethyl Enzalutamide 1242137-16-1 N-Desmethyl enzalutamide is a major metabolite of Enzalutamide Enzalutamide MDV3100 is an androgen-receptor AR antagonist with IC50 of 36 nM
CSN18357 MK-0773 606101-58-0 MK-0773 one of selective androgen receptor modulators SARMs is a 4-aza-steroid that exhibited tissue selectivity in humans IC50 66 nM
CSN13670 LGD-4033 1165910-22-4 LGD-4033 is a nonsteroidal oral SARM that binds to androgen receptor with high affinity Ki of 1 nM and selectivity
CSN10977 Hydroxyflutamide 52806-53-8 Hydroxyflutamide is a derivative of the synthetic steroid ethisterone, that suppresses the production of gonadotrophins, and has some weak androgenic effects.
CSN11169 Hydromadinone 16469-74-2 Hydromadinone is a steroidal progestin of the 17-hydroxyprogesterone group
CSN18667 GSK2881078 1539314-06-1 GSK 2881078 is a selective androgen receptor modulator potentially for the treatment of cachexia
CSN17573 GLPG0492 R-Enantiomer 1215085-93-0 GLPG0492 R-enantiomer is the R-Enantiomer of GLPG-0492 which is a selective androgen receptor modulator
CSN17572 GLPG0492 1215085-92-9 GLPG0492 is a selective androgen receptor modulator and exhibits anabolic activity on muscle strongly dissociated from the androgenic activity on prostate after oral dosing
CSN11095 Gestonorone 2137-18-0 Gestronol is a steroidal progestin of the 19-norprogesterone and 17-hydroxyprogesterone groups
CSN16707 Flutamide   13311-84-7 Flutamide is a competitive non-steroidal antagonist of androgen receptor.
CSN10468 EPI-001 227947-06-0 EPI-001 is an androgen receptor N-terminal domain antagonist with IC50 of 6 M and a selective PPAR-gamma modulator
CSN12389 Enzalutamide   915087-33-1 Enzalutamide is an androgen-receptor AR antagonist with IC50 of 36 nM in LNCaP cells
CSN10728 Cyproterone Acetate   427-51-0 Cyproterone Acetate is an antagonist and partial agonist of androgen receptor with IC50 value of 71 nM and EC50 value of 4M
CSN18075 Cortexolone 17 alpha-Propionate 19608-29-8 Cortexolone 17 alpha-propionate is a topical and peripherally selective androgen antagonist, which is used in treatment of acne and androgenic alopecia.
CSN16582 BMS-564929 627530-84-1 BMS-564929 is an androgen receptor AR agonist binds to androgen receptor AR with a Ki of 211016 nM
CSN12437 Bicalutamide   90357-06-5 Bicalutamide is non-steroidal androgen receptor antagonist with IC50 value of 190 nM
CSN17150 AZD3514 1240299-33-5 AZD3514 is a potent and oral androgen receptor downregulator with Ki of 22 M and has ability of reducing AR protein expression
CSN17338 Dimethylcurcumin 52328-98-0 ASC-J9 an antitumor agent suppresses castration-resistant prostate cancer growth via degradation of full-length and splice variant androgen receptors
CSN13830 ARN-509 956104-40-8 ARN-509 can compeitively and selectively inhibit androgen receptor with IC50 value of 16 nM
CSN20433 Androgen Receptor Modulator C7 2109805-69-6 Androgen receptor modulator C7 is a potent AR ARE EC50 034 nM and tissue-selective NC interaction EC50 1206 nM modulator
CSN22336 ACP-105 899821-23-9 ACP-105 is a potent nonsteroidal selective androgen receptor modulator (SARM) with partial agonist activity relative to the natural androgen testosterone.
CSN19392 3,3'-Diindolylmethane   1968-05-4 3,3-Diindolylmethane is an AR structurally similar androgen receptor antagonist.
CSN23255 1-Phenylpentan-1-ol   583-03-9 1-Phenylpentan-1-ol is an intermediate for synthesis of -amino-carbonyl-based androgen receptor antagonist
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