Welcome to CSNpharm! For Research Use Only!
Home Promotion +1-708-781-1677 sales@csnpharm.com    

AMPK

AMPK

Cat. No. Product Name CAS No. Information
CSN18405 ZLN024 723249-01-2 ZLN024 is an AMPK allosteric activator and activates 111 and 211 by around 225 fold with an EC50 of about 12 M
CSN18969 ZLN024 HCl 1883548-91-1 ZLN024 HCl is an AMPK allosteric activator and activates α1β1γ1 and α2β1γ1 by around 2–2.5 fold with an EC50 of about 1–2 μM.
CSN17652 YLF-466D 1273323-67-3 YLF-466D is an allosteric AMPK activator
CSN17571 WZ4003 1214265-58-3 WZ4003 is a potent and selective NUAK12 inhibitor with IC50 values of 20 and 100 nM respectively
CSN23058 PT 1 331002-70-1 PT 1 is a AMP-activated protein kinase (AMPK) activator.
CSN15574 Phillyrin   487-41-2 Phillyrin is a naturally occuring AMPK activity enhancer isolated and purified from the fruits of Forsythia suspensa
CSN11690 PHenformin HCl   834-28-6 Phenformin HCl is an AMPK activator which can increase the phosphorylation and activation of AMPKalpha1 and AMPKalpha2
CSN22062 PF-06409577 1467057-23-3 PF-06409577 is a potent and selective allosteric activator of AMPK with EC50 value of 7 nM for AMPK111 but 40000 nM for AMPK121
CSN24788 O-304 1261289-04-6 O-304 is a first-in-class, orally available pan-AMPK activator, which increases AMPK activity by suppressing the dephosphorylation of pAMPK. O-304 exhibits a great potential as a drug to treat type 2 diabetes (T2D) and associated cardiovascular complications [1][2].
CSN21095 ex229 1219739-36-2 Novel AMPK activator increasing AMPK activity of both AMPKgamma1- and AMPKgamma3-containing complexes in mouse skeletal muscle
CSN13488 Norathyriol 3542-72-1 Norathyriol, a natural product isolated and purified from the herbs of Mangifera indica L., can improve the glucose utilization and insulin sensitivity by up-regulation of the phosphorylation of AMPK. Norathyriol exerts a potent chemopreventive activity by inhibiting Akt activation in neoplastic cell transformation.
CSN20178 Mogroside IIIE 88901-37-5 Mogroside IIIE a naturally occuring cucurbitane glycoside which can attenuate gestational diabetes mellitus through activating of AMPK signaling pathway in mice.
CSN20469 MK-8722 1394371-71-1 MK-8722 is a potent, direct, allosteric activator of all twelve mammalian AMPK complexes.
CSN23901 MK-3903 1219737-12-8 MK-3903 is a potent and selective AMPK activator with EC50 value of 8nM.
CSN19218 GSK621 1346607-05-3 In AML cell lines and primary AML samples, GSK621 markedly increases phosphorylation at AMPKα T172, a marker of AMPK activation.
CSN13786 HTH-01-015 1613724-42-7 HTH-01-015 is a selective NUAK1 inhibitor but not NUAK2 with IC50 of 100 nM suppressing NUAK1-mediated MYPT1 phosphorylation
CSN14375 Gomisin J 66280-25-9 Gomisin J is a natural product isolated and purified from the fruits of Schizandra chinensis with vasodilatory activity that mediates mainly by calcium-dependent activation of eNOS with subsequent production of endothelial NO, and inhibits LPO in rat liver mitochondria and protects cultured myocardial cells from being injured by calcium paradox.
CSN19411 Ginkgolide C   15291-76-6 Ginkgolide C can enhance the cardiac function of rats in the body, is a flavone isolated from Ginkgo biloba leaves.
CSN17240 ETC-1002   738606-46-7 ETC-1002 is an AMPK activator and increase the level of AMPK phosphorylation.
CSN13424 Dorsomorphin 866405-64-3 Dorsomorphin is a selective AMPK inhibitor with Ki value of 109 nM.
CSN15887 Dorsomorphin 2HCl 1219168-18-9 Dorsomorphin 2HCl is a selective AMPK inhibitor with Ki value of 109 nM.
CSN17597 Ampkinone 1233082-79-5 Ampkinone is a small molecule activator of AMPK and stimulates functional activation of AMPK via the phosphorylation at Thr172 in cultured L6 muscle cells with an EC50 value of 43 M enhancing glucose uptake by 32-fold
CSN23079 RSVA 405 140405-36-3 AMPK activator; also STAT3 inhibitor
CSN23366 Adenosine 5'-monophosphate, disodium salt   4578-31-8 Adenosine 5-monophosphate disodium salt is an activator of AMPK and can be used as a substrate of AMP-thymidine kinase AMP deaminase and 5-nucleotidase
CSN12424 A-769662 844499-71-4 A-769662 is a reverible and allosteric activator of AMPK through inhibiting dephosphorylation of AMPK on Thr-172
CSN17102 1,8-Dihydroxyanthraquinone 117-10-2 1,8-Dihydroxyanthraquinone is a synthetic anthraquinone derivative, currently used as an antioxidant in synthetic lubricants, in the synthesis of antitumor agents, as a fungicide and as an intermediate for making dyes.
<< PREV 1 NEXT >>