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AMPAR

AMPAR

Cat. No. Product Name CAS No. Information
CSN21669 gamma-DGG 6729-55-1 γDGG is a blocker of AMPA receptor.
CSN17953 Fanapanel 161605-73-8 ZK200775 is a highly selective AMPAkainate antagonist with little activity against NMDA with Ki values of 3.2 nM, 100 nM, and 8.5 M against quisqualate, kainate, and NMDA, respectively.
CSN17630 Fanapanel hydrate 1255517-78-2 ZK200775 is a highly selective AMPAkainate antagonist with little activity against NMDA and has Ki values of 3.2 nM, 100 nM, and 8.5 M against quisqualate, kainate, and NMDA, respectively.
CSN22000 Zonampanel 210245-80-0 YM 872 is an AMPA receptor antagonists and acts as antiepileptic drugs.
CSN23175 UBP-282 544697-47-4 UBP-282 is an α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) and kainate receptor antagonist.
CSN24615 UBP310 902464-46-4 UBP 310 is an antagonist of GluK1 (formerly GLUK5) kainate receptor with IC50 of 130 nM.
CSN24617 UBP 302 745055-91-8 UBP 302 is a potent and selective GluK1 (formally GluR5)-subunit containing kainate receptor antagonist with KD of 402 nM.
CSN24618 U-54494A 112465-94-8 U-54494A hydrochloride is a selective non-competitive AMPA receptor antagonist with IC50 of 10-20 mM.
CSN13864 Sunifiram 314728-85-3 Sunifiram is a piperazine derived ampakine-like drug(acting via AMPA receptors) which has nootropic effects in animal studies with significantly higher potency than piracetam.
CSN20167 Selurampanel 912574-69-7 Selurampanel is a competitive AMPAkainate receptor antagonist drug for epilepsy
CSN11876 (S)-Willardiine 21416-43-3 S-Willardiine is a potent agonist of AMPAkainate receptors with EC50 of 448 M
CSN19840 (RS)-AMPA hydrobromide 171259-81-7 RS-AMPA hydrobromide is a class of glutamate agonist structurally related to ibotenic acid
CSN24155 Philanthotoxin 74 2HCl 1227301-51-0 Philanthotoxin 74 dihydrochloride (PhTx 74) is an AMPAR antagonist; inhibits GluR3 and GluR1 with IC50s of 263 and 296 nM, respectively.
CSN22487 PF-4778574 1219633-99-4 PF-4778574 is a positive allosteric modulation of AMPA receptor with EC50 of 45 to 919 nM in differenct cells
CSN32485 Pesampator 1258963-59-5 PF-04958242 is an AMPA receptor positive allosteric modulator.
CSN17813 PEPA 141286-78-4 PEPA is an allosteric modulator of AMPA receptors and binds to the GluA2o and GluA3o LBDs and can be utilized as an indicator of AMPA receptor heterogeneity
CSN23006 NPEC-caged-(S)-AMPA 1257323-84-4 NPEC-caged-(S)-AMPA is an agonist at the AMPA receptor.
CSN13580 Omberacetam   157115-85-0 Noopept is a potent nootropic that improves cognitive ability.
CSN22241 NBQX 118876-58-7 NBQX is a potent, selective and competitive AMPAR antagonist, which shows activity of neuroprotective and anticonvulsant.
CSN22999 NBQX disodium 479347-86-9 NBQX Disodium Salt is a potent, selective and competitive AMPA receptor antagonist.
CSN20510 LY3130481 1610802-47-5 LY3130481 is the the first -amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid AMPA receptor antagonist that is dependent on the presence of TARP -8 LY3130481 is fully protective against pentylenetetrazole-induced convulsions in rats without the motor impairment associated with non-TARP-dependent AMPA receptor antagonists
CSN16600 (S)-2-Amino-5-(ethylamino)-5-oxopentanoic acid 3081-61-6 L-theanine is an amino acid found most commonly in tea leaves and binds to ionotropic glutamate receptors in the micromolar range including the AMPA and kainate receptors and to a lesser extent the NMDA receptor
CSN10840 Empirical Formula   492-27-3 Kynurenic Acid is a broad spectrum glutamatergic antagonist which can antagonize NMDA kainate and AMPA receptors
CSN24076 JNJ-61432059 2035814-50-5 JNJ-61432059 is an oral active and selective negative modulator of AMPAR associated with trans-membrane AMPAR regulatory protein (TARP) γ-8, with a pIC50 of 9.7 for GluA1/γ-8. Exhibits time- and dose-dependent AMPAR/γ-8 receptor occupancy in mouse hippocampus, resulting in robust seizure protection in corneal kindling and pentylenetetrazole (PTZ) anticonvulsant models[1].
CSN25362 IDRA 21 22503-72-6 IDRA-21 is a positive AMPA receptor modulator. IDRA-21 inhibits synaptic and extrasynaptic NMDA receptor mediated events in cultured cerebellar granule cells. IDRA 21 enhances ischemic hippocampal neuron injury.
CSN22846 GYKI 52466 102771-26-6 GYKI 52466 2HCl is a selective non-competitive AMPA receptor antagonist with IC50 of 10-20 μM.
CSN21401 Quisqualic acid 52809-07-1 Glutamate receptor agonist acting at AMPA receptors and metabotropic glutamate receptors positively linked to phosphoinositide hydrolysis Sensitizes neurons in hippocampus to depolarization by L-AP6 the so called quis effect
CSN27523 Farampator 211735-76-1 Farampator (CX-691;Org24448) is an AMPA receptor positive modulator.
CSN22784 CX 614 191744-13-5 CX 614 is a positive allosteric modulator of AMPA receptors.
CSN19847 CP-465022 199655-36-2 CP 465022 HCl is a selective, non-competitive AMPA receptor antagonist (IC50 = 25 nM in rat cortical neurons) that displays potent anticonvulsant activity.
CSN12675 Coluracetam   135463-81-9 Coluracetam a nootropic which can increase the potency of AMPA receptors.
CSN22766 7-Nitro-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carbonitrile   115066-14-3 CNQX is a potent and selective non-NMDA iGluR antagonist
CSN24616 ATPA 140158-50-5 ATPA is a selective and potent GluK1 kainate receptor agonist with Ki of 4.3 nM.
CSN10196 Piperidin-1-yl(quinoxalin-6-yl)methanone   154235-83-3 Ampalex is a positive allosteric modulator of AMPAR and is researched as a treatment for Alzheimers disease.
CSN25263 1-BCP 34023-62-6 1-BCP is can modulate AMPA receptor gated currents and enhence memory.
CSN23429 H-Glu-OH   56-86-0 (S)-Glutamic acid acts as an excitatory neurotransmitter in the central nervous system.
CSN22635 (S)-AMPA 83643-88-3 (S)-AMPA is a selective AMPA agonist.
CSN22625 (R)-3,4-DCPG 201730-10-1 (R)-3,4-DCPG is a AMPA receptor antagonist.
CSN51552 Unifiram 272786-64-8
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