AMPAR
Cat. No. | Product Name | CAS No. | Information |
---|---|---|---|
CSN17953 | ZK200775 | 161605-73-8 | ZK200775 is a highly selective AMPAkainate antagonist with little activity against NMDA with Ki values of 3.2 nM, 100 nM, and 8.5 M against quisqualate, kainate, and NMDA, respectively. |
CSN11876 | (S)-Willardiine | 21416-43-3 | S-Willardiine is a potent agonist of AMPAkainate receptors with EC50 of 448 M |
CSN17813 | PEPA | 141286-78-4 | PEPA is an allosteric modulator of AMPA receptors and binds to the GluA2o and GluA3o LBDs and can be utilized as an indicator of AMPA receptor heterogeneity |
CSN13580 | Noopept | 157115-85-0 | Noopept is a potent nootropic that improves cognitive ability. |
CSN22241 | NBQX | 118876-58-7 | NBQX is a potent, selective and competitive AMPAR antagonist, which shows activity of neuroprotective and anticonvulsant. |
CSN22957 | LY 404187 | 211311-95-4 | LY 404187 is a selective positive allosteric modulator of AMPA receptors with IC50s of 015 021 166 and 565 M for GluA2i GluA4i GluA3i and GluA1i respectively |
CSN16600 | L-Theanine | 3081-61-6 | L-theanine is an amino acid found most commonly in tea leaves and binds to ionotropic glutamate receptors in the micromolar range including the AMPA and kainate receptors and to a lesser extent the NMDA receptor |
CSN10840 | Kynurenic Acid | 492-27-3 | Kynurenic Acid is a broad spectrum glutamatergic antagonist which can antagonize NMDA kainate and AMPA receptors |
CSN25362 | IDRA 21 | 22503-72-6 | IDRA-21 is a positive AMPA receptor modulator. IDRA-21 inhibits synaptic and extrasynaptic NMDA receptor mediated events in cultured cerebellar granule cells. IDRA 21 enhances ischemic hippocampal neuron injury. |
CSN21401 | L-Quisqualic Acid | 52809-07-1 | Glutamate receptor agonist acting at AMPA receptors and metabotropic glutamate receptors positively linked to phosphoinositide hydrolysis Sensitizes neurons in hippocampus to depolarization by L-AP6 the so called quis effect |
CSN27523 | Farampator | 211735-76-1 | Farampator (CX-691;Org24448) is an AMPA receptor positive modulator. |
CSN22784 | CX 614 | 191744-13-5 | CX 614 is a positive allosteric modulator of AMPA receptors. |
CSN12675 | Coluracetam | 135463-81-9 | Coluracetam a nootropic which can increase the potency of AMPA receptors. |
CSN22766 | CNQX | 115066-14-3 | CNQX is a potent and selective non-NMDA iGluR antagonist |
CSN22005 | AMP 397 | 188696-80-2 | Becampanel (AMP397) is the first competitive AMPA antagonist and an antiepileptic agent. |
CSN24616 | ATPA | 140158-50-5 | ATPA is a selective and potent GluK1 kainate receptor agonist with Ki of 4.3 nM. |
CSN10196 | Ampalex | 154235-83-3 | Ampalex is a positive allosteric modulator of AMPAR and is researched as a treatment for Alzheimers disease. |
CSN25263 | 1-BCP | 34023-62-6 | 1-BCP is can modulate AMPA receptor gated currents and enhence memory. |
CSN23429 | L-Glutamic Acid | 56-86-0 | (S)-Glutamic acid acts as an excitatory neurotransmitter in the central nervous system. |
CSN22635 | (S)-AMPA | 83643-88-3 | (S)-AMPA is a selective AMPA agonist. |