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AMPAR
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN21669 | H-D-Glu(Gly-OH)-OH | 6729-55-1 | γDGG is a blocker of AMPA receptor. |
| CSN17953 | ZK200775 | 161605-73-8 | ZK200775 is a highly selective AMPAkainate antagonist with little activity against NMDA with Ki values of 3.2 nM, 100 nM, and 8.5 M against quisqualate, kainate, and NMDA, respectively. |
| CSN17630 | ZK200775 Hydrate | 1255517-78-2 | ZK200775 is a highly selective AMPAkainate antagonist with little activity against NMDA and has Ki values of 3.2 nM, 100 nM, and 8.5 M against quisqualate, kainate, and NMDA, respectively. |
| CSN23205 | YM 90K HCl | 154164-30-4 | YM90K hydrochloride is an AMPA receptor antagonist. |
| CSN22000 | YM 872 | 210245-80-0 | YM 872 is an AMPA receptor antagonists and acts as antiepileptic drugs. |
| CSN23175 | UBP 282 | 544697-47-4 | UBP-282 is an α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) and kainate receptor antagonist. |
| CSN24615 | UBP 310 | 902464-46-4 | UBP 310 is an antagonist of GluK1 (formerly GLUK5) kainate receptor with IC50 of 130 nM. |
| CSN24617 | (S)-2-((3-(2-Amino-2-carboxyethyl)-2,6-dioxo-2,3-dihydropyrimidin-1(6H)-yl)methyl)benzoic acid | 745055-91-8 | UBP 302 is a potent and selective GluK1 (formally GluR5)-subunit containing kainate receptor antagonist with KD of 402 nM. |
| CSN13591 | Talampanel | 161832-65-1 | Talampanel, a potent and selective AMPA-receptor antagonist, is a potential antiepileptic drug (AED). |
| CSN20167 | Selurampanel | 912574-69-7 | Selurampanel is a competitive AMPAkainate receptor antagonist drug for epilepsy |
| CSN11876 | (S)-Willardiine | 21416-43-3 | S-Willardiine is a potent agonist of AMPAkainate receptors with EC50 of 448 M |
| CSN19840 | (RS)-AMPA Hydrobromide | 171259-81-7 | RS-AMPA hydrobromide is a class of glutamate agonist structurally related to ibotenic acid |
| CSN13810 | Piracetam | 7491-74-9 | Piracetam is a cyclic derivative of GABA which works as a positive allosteric modulator of the AMPA receptor |
| CSN22487 | PF-4778574 | 1219633-99-4 | PF-4778574 is a positive allosteric modulation of AMPA receptor with EC50 of 45 to 919 nM in differenct cells |
| CSN17813 | PEPA | 141286-78-4 | PEPA is an allosteric modulator of AMPA receptors and binds to the GluA2o and GluA3o LBDs and can be utilized as an indicator of AMPA receptor heterogeneity |
| CSN25561 | PD-161989 | 186268-07-5 | PD-161989 is an AMPA receptor antagonist. |
| CSN23006 | NPEC-caged-(S)-AMPA | 1257323-84-4 | NPEC-caged-(S)-AMPA is an agonist at the AMPA receptor. |
| CSN13580 | Noopept | 157115-85-0 | Noopept is a potent nootropic that improves cognitive ability. |
| CSN22241 | NBQX | 118876-58-7 | NBQX is a potent, selective and competitive AMPAR antagonist, which shows activity of neuroprotective and anticonvulsant. |
| CSN22999 | NBQX Disodium Salt | 479347-86-9 | NBQX Disodium Salt is a potent, selective and competitive AMPA receptor antagonist. |
| CSN17585 | Naspm | 122306-11-0 | Naspm is a potent and selective Ca2 permeable AMPA receptor Ca-perm AMPAR blocker |
| CSN15793 | LY450108 | 376594-67-1 | LY450108 is an alpha-amino-3-hydroxy-5-methyl-4-isoxazole-propionic acid AMPA receptor potentiator |
| CSN20510 | LY3130481 | 1610802-47-5 | LY3130481 is the the first -amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid AMPA receptor antagonist that is dependent on the presence of TARP -8 LY3130481 is fully protective against pentylenetetrazole-induced convulsions in rats without the motor impairment associated with non-TARP-dependent AMPA receptor antagonists |
| CSN16600 | L-Theanine | 3081-61-6 | L-theanine is an amino acid found most commonly in tea leaves and binds to ionotropic glutamate receptors in the micromolar range including the AMPA and kainate receptors and to a lesser extent the NMDA receptor |
| CSN10840 | Kynurenic Acid | 492-27-3 | Kynurenic Acid is a broad spectrum glutamatergic antagonist which can antagonize NMDA kainate and AMPA receptors |
| CSN24076 | JNJ-61432059 | 2035814-50-5 | JNJ-61432059 is an oral active and selective negative modulator of AMPAR associated with trans-membrane AMPAR regulatory protein (TARP) γ-8, with a pIC50 of 9.7 for GluA1/γ-8. Exhibits time- and dose-dependent AMPAR/γ-8 receptor occupancy in mouse hippocampus, resulting in robust seizure protection in corneal kindling and pentylenetetrazole (PTZ) anticonvulsant models[1]. |
| CSN21937 | GYKI53655 HCl | 143692-48-2 | GYKI53655 hydrochloride is an α-amino-3-hydroxy-5-methylisoxazole-4-propionic acid (AMPA) antagonist. |
| CSN22846 | GYKI 52466 2HCl | 102771-26-6 | GYKI 52466 2HCl is a selective non-competitive AMPA receptor antagonist with IC50 of 10-20 μM. |
| CSN21401 | L-Quisqualic Acid | 52809-07-1 | Glutamate receptor agonist acting at AMPA receptors and metabotropic glutamate receptors positively linked to phosphoinositide hydrolysis Sensitizes neurons in hippocampus to depolarization by L-AP6 the so called quis effect |
| CSN10853 | DNQX | 2379-57-9 | DNQX is a selective non-NMDA iGluR antagonist |
| CSN12690 | CX-546 | 215923-54-9 | CX-546 is a AMPAR potentiator which can destabilize the desensitized receptor conformation |
| CSN22784 | CX 614 | 191744-13-5 | CX 614 is a positive allosteric modulator of AMPA receptors. |
| CSN19847 | CP 465022 | 199655-36-2 | CP 465022 HCl is a selective, non-competitive AMPA receptor antagonist (IC50 = 25 nM in rat cortical neurons) that displays potent anticonvulsant activity. |
| CSN12675 | Coluracetam | 135463-81-9 | Coluracetam a nootropic which can increase the potency of AMPA receptors. |
| CSN22766 | CNQX | 115066-14-3 | CNQX is a potent and selective non-NMDA iGluR antagonist |
| CSN22767 | CNQX Disodium Salt | 479347-85-8 | CNQX Disodium Salt is a AMPA/kainate antagonist and also available as part of the Kainate Receptor. |
| CSN18250 | CMPDA | 380607-77-2 | CMPDA is a positive allosteric modulator of AMPA receptors with EC50s of 454 42 nM634 56 nM for GluA2iGluA2o receptor |
| CSN22005 | AMP 397 | 188696-80-2 | Becampanel (AMP397) is the first competitive AMPA antagonist and an antiepileptic agent. |
| CSN24616 | ATPA | 140158-50-5 | ATPA is a selective and potent GluK1 kainate receptor agonist with Ki of 4.3 nM. |
| CSN10315 | Aniracetam | 72432-10-1 | Aniracetam is an allosteric modulator of AMPAR which can reduce glutamate receptor desensitization and potentiate metabotropic glutamate receptor activity |
| CSN10196 | Ampalex | 154235-83-3 | Ampalex is a positive allosteric modulator of AMPAR and is researched as a treatment for Alzheimers disease. |
| CSN25263 | 1-BCP | 34023-62-6 | 1-BCP is can modulate AMPA receptor gated currents and enhence memory. |
| CSN13605 | β-ODAP | 5302-45-4 | -ODAP is an analog of glutamic acid present in Lathyrus sativus grass pea that activates AMPA receptors |
| CSN23429 | L-Glutamic Acid | 56-86-0 | (S)-Glutamic acid acts as an excitatory neurotransmitter in the central nervous system. |
| CSN22635 | (S)-AMPA | 83643-88-3 | (S)-AMPA is a selective AMPA agonist. |
| CSN17690 | (S)-(-)-5-Fluorowillardiine HCl | 1321546-70-6 | (S)-(-)-5-Fluorowillardiine HCl is a potent and specific AMPAR agonist. |
| CSN22625 | (R)-3,4-DCPG | 201730-10-1 | (R)-3,4-DCPG is a AMPA receptor antagonist. |
| CSN25362 | IDRA 21 | 22503-72-6 |
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