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AMPAR
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN21669 | gamma-DGG | 6729-55-1 | γDGG is a blocker of AMPA receptor. |
| CSN17953 | Fanapanel | 161605-73-8 | ZK200775 is a highly selective AMPAkainate antagonist with little activity against NMDA with Ki values of 3.2 nM, 100 nM, and 8.5 M against quisqualate, kainate, and NMDA, respectively. |
| CSN17630 | Fanapanel hydrate | 1255517-78-2 | ZK200775 is a highly selective AMPAkainate antagonist with little activity against NMDA and has Ki values of 3.2 nM, 100 nM, and 8.5 M against quisqualate, kainate, and NMDA, respectively. |
| CSN22000 | Zonampanel | 210245-80-0 | YM 872 is an AMPA receptor antagonists and acts as antiepileptic drugs. |
| CSN23175 | UBP-282 | 544697-47-4 | UBP-282 is an α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) and kainate receptor antagonist. |
| CSN24615 | UBP310 | 902464-46-4 | UBP 310 is an antagonist of GluK1 (formerly GLUK5) kainate receptor with IC50 of 130 nM. |
| CSN24617 | UBP 302 | 745055-91-8 | UBP 302 is a potent and selective GluK1 (formally GluR5)-subunit containing kainate receptor antagonist with KD of 402 nM. |
| CSN24618 | U-54494AHYDROCHLORIDE | 112465-94-8 | U-54494A hydrochloride is a selective non-competitive AMPA receptor antagonist with IC50 of 10-20 mM. |
| CSN13864 | Sunifiram | 314728-85-3 | Sunifiram is a piperazine derived ampakine-like drug(acting via AMPA receptors) which has nootropic effects in animal studies with significantly higher potency than piracetam. |
| CSN20167 | Selurampanel | 912574-69-7 | Selurampanel is a competitive AMPAkainate receptor antagonist drug for epilepsy |
| CSN11876 | (S)-Willardiine | 21416-43-3 | S-Willardiine is a potent agonist of AMPAkainate receptors with EC50 of 448 M |
| CSN19840 | (RS)-AMPA Hydrobromide | 171259-81-7 | RS-AMPA hydrobromide is a class of glutamate agonist structurally related to ibotenic acid |
| CSN24155 | Philanthotoxin 74 dihydrochloride | 1227301-51-0 | Philanthotoxin 74 dihydrochloride (PhTx 74) is an AMPAR antagonist; inhibits GluR3 and GluR1 with IC50s of 263 and 296 nM, respectively. |
| CSN22487 | PF-4778574 | 1219633-99-4 | PF-4778574 is a positive allosteric modulation of AMPA receptor with EC50 of 45 to 919 nM in differenct cells |
| CSN32485 | Pesampator | 1258963-59-5 | PF-04958242 is an AMPA receptor positive allosteric modulator. |
| CSN17813 | PEPA | 141286-78-4 | PEPA is an allosteric modulator of AMPA receptors and binds to the GluA2o and GluA3o LBDs and can be utilized as an indicator of AMPA receptor heterogeneity |
| CSN23006 | NPEC-caged-(S)-AMPA | 1257323-84-4 | NPEC-caged-(S)-AMPA is an agonist at the AMPA receptor. |
| CSN13580 | Omberacetam | 157115-85-0 | Noopept is a potent nootropic that improves cognitive ability. |
| CSN22241 | NBQX | 118876-58-7 | NBQX is a potent, selective and competitive AMPAR antagonist, which shows activity of neuroprotective and anticonvulsant. |
| CSN22999 | NBQX disodium | 479347-86-9 | NBQX Disodium Salt is a potent, selective and competitive AMPA receptor antagonist. |
| CSN20510 | LY3130481 | 1610802-47-5 | LY3130481 is the the first -amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid AMPA receptor antagonist that is dependent on the presence of TARP -8 LY3130481 is fully protective against pentylenetetrazole-induced convulsions in rats without the motor impairment associated with non-TARP-dependent AMPA receptor antagonists |
| CSN16600 | L-Theanine | 3081-61-6 | L-theanine is an amino acid found most commonly in tea leaves and binds to ionotropic glutamate receptors in the micromolar range including the AMPA and kainate receptors and to a lesser extent the NMDA receptor |
| CSN10840 | Kynurenic acid | 492-27-3 | Kynurenic Acid is a broad spectrum glutamatergic antagonist which can antagonize NMDA kainate and AMPA receptors |
| CSN24076 | JNJ-61432059 | 2035814-50-5 | JNJ-61432059 is an oral active and selective negative modulator of AMPAR associated with trans-membrane AMPAR regulatory protein (TARP) γ-8, with a pIC50 of 9.7 for GluA1/γ-8. Exhibits time- and dose-dependent AMPAR/γ-8 receptor occupancy in mouse hippocampus, resulting in robust seizure protection in corneal kindling and pentylenetetrazole (PTZ) anticonvulsant models[1]. |
| CSN25362 | IDRA 21 | 22503-72-6 | IDRA-21 is a positive AMPA receptor modulator. IDRA-21 inhibits synaptic and extrasynaptic NMDA receptor mediated events in cultured cerebellar granule cells. IDRA 21 enhances ischemic hippocampal neuron injury. |
| CSN22846 | GYKI 52466 | 102771-26-6 | GYKI 52466 2HCl is a selective non-competitive AMPA receptor antagonist with IC50 of 10-20 μM. |
| CSN21401 | Quisqualic acid | 52809-07-1 | Glutamate receptor agonist acting at AMPA receptors and metabotropic glutamate receptors positively linked to phosphoinositide hydrolysis Sensitizes neurons in hippocampus to depolarization by L-AP6 the so called quis effect |
| CSN27523 | Farampator | 211735-76-1 | Farampator (CX-691;Org24448) is an AMPA receptor positive modulator. |
| CSN22784 | CX 614 | 191744-13-5 | CX 614 is a positive allosteric modulator of AMPA receptors. |
| CSN12675 | Coluracetam | 135463-81-9 | Coluracetam a nootropic which can increase the potency of AMPA receptors. |
| CSN22766 | CNQX | 115066-14-3 | CNQX is a potent and selective non-NMDA iGluR antagonist |
| CSN24616 | ATPA | 140158-50-5 | ATPA is a selective and potent GluK1 kainate receptor agonist with Ki of 4.3 nM. |
| CSN10196 | CX516 | 154235-83-3 | Ampalex is a positive allosteric modulator of AMPAR and is researched as a treatment for Alzheimers disease. |
| CSN25263 | 1-BCP | 34023-62-6 | 1-BCP is can modulate AMPA receptor gated currents and enhence memory. |
| CSN23429 | L-Glutamic acid | 56-86-0 | (S)-Glutamic acid acts as an excitatory neurotransmitter in the central nervous system. |
| CSN22635 | (S)-AMPA | 83643-88-3 | (S)-AMPA is a selective AMPA agonist. |
| CSN22625 | (R)-3,4-DCPG | 201730-10-1 | (R)-3,4-DCPG is a AMPA receptor antagonist. |
| CSN51552 | 2-((4-Fluorophenyl)sulfonyl)hexahydropyrrolo[1,2-a]pyrazin-6(2H)-one | 272786-64-8 |
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