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• All Targets

All Targets

Inhibitors & Agonists

• Functionalized E3 Ligand

  Functionalized E3 Ligand (Thalidomide)

  Functionalized E3 Ligand (VH032)

  Functionalized E3 Ligand (Pomalidomide)

  Functionalized E3 Ligand (other)

  Functionalized E3 Ligand (for VHL)

  Functionalized E3 Ligand (Bestatin)

• Linker

  PROTAC Linker

• Functionalized Warhead Ligand

  Bromodomain BET/Warhead Ligand

  Bcr-Abl/Warhead Ligand

  Sirtuin/Warhead Ligand

  FKBP/Warhead Ligand

  mTOR/Warhead Ligand

  CDK/Warhead Ligand

• E3 Ligand Plus Linker

  E3 Ligand Plus Linker (Pomalidomide)

  E3 Ligand Plus Linker (VH032)

  E3 Ligand Plus Linker (Thalidomide)

  E3 Ligand Plus Linker (Lenalidomide)

  E3 Ligand Plus Linker (other)

• PROTACs

  +More

  Bromodomain BET/PROTAC

  VHL/PROTAC

  FKBP/PROTAC

  TRIM/PROTAC

  CDK/PROTAC

  ALK/PROTAC

  ERR/PROTAC

  PTK2/PROTAC

  Raf/PROTAC

  Sirtuin/PROTAC

  CRBN/PROTAC

  Multikinase/PROTAC

  p38/PROTAC

  K-Ras (G12C)/PROTAC

  ERα/PROTAC

  Cdc20/PROTAC

  Bcl-2/PROTAC

  Mcl-1/PROTAC

  FAK/PROTAC

  SGK3/PROTAC

  BTK/PROTAC

  RIP Kinase/PROTAC

  FLT3-ITD/PROTAC

  RAR/PROTAC

  APC/PROTAC

  IAP/PROTAC

  CRABP/PROTAC

  EGFR/PROTAC

  ER/PROTAC

  PCAF/PROTAC

  PD-1 PD-L1/PROTAC

  SHP-2/PROTAC

  STAT/PROTAC

  TBK/PROTAC

  Bcl-xL/PROTAC

  Halo/PROTAC

• ADC

  ADC Linker

  ADC Linker with Payload

  ADC Toxin

• Anti-infection

  +More

  Antibacterial

  Antifungal

  Antiparasitic

  CMV

  Filovirus

  HBV

  HCV

  HIV

  HIV Integrase

  HIV Protease

  HRV

  HSV

  Influenza Virus

  NNRTI

  NRTI

  Orthopoxvirus

  Reverse Transcriptase

  RSV

  SARS-CoV

  CCR

  Dengue Virus

  H37Rv

  HCMV

  HHV

  LpxC

  MCMV

  Neuraminidase

  NS2B-NS3 Protease

  Nucleic Acid Synthesis

  Prion

  SQLE

  Antiviral

  EBV

  MM virus

  NtART

  VZV

  β-lactamase

  FCoV

  3CLpro

  M2 proton channel

  Antiprotozoal

  FIP

  Viral MTase

  PLP

  GraR

  Peroxiredoxin

  BVDV

  SAMHD1

• Apoptosis

  +More

  Apoptosis Inducer

  Bcl-2

  Caspase

  c-Myc

  c-RET

  DAPK

  IAP

  MDM2

  p53

  PD-1/PD-L1

  PERK

  PKD

  Survivin

  Thymidylate Synthase

  TNF-alpha

  G0/G1 switch protein 2

  MDM2/PROTAC

  Mcl-1 (stapled peptide)

  Bim (stapled peptide)

  Bcl-2 (stapled peptide)

  p53/MDM2 (stapled peptide)

  Necroptosis

  C/EBP

  Mcl-1/PROTAC

  Bcl-2/PROTAC

  IAP/PROTAC

  PD-1 PD-L1/PROTAC

  p32

• Autophagy

  Autophagy

  CXCR

  LRRK2

  ULK

  Lysosome

  SPHK

  PPT

  mitoNEET

  TFEB

  LC3

• Cell Cycle

  +More

  APC

  Aurora Kinase

  Casein Kinase

  CDK

  Chk

  c-Myc

  CRISPR/Cas9

  CRM1

  DHFR

  DNA/RNA Synthesis

  DUB

  DYRK

  eIF

  FOX

  G-quadruplex

  Haspin Kinase

  HSP

  IRE1

  Kinesin

  LIMK

  Microtubule/Tubulin

  Mps1

  Nucleoside Antimetabolite/Analog

  p97

  PAK

  PD-1/PD-L1

  PERK

  PLK

  PPAR

  PTEN

  RAD51

  Rho

  ROCK

  Wee1

  BUB

  HSF

  Mad2

  p21

  rRNA synthesis

  E1/E2/E3 Enzyme

  FOXM1

  MKLP

  Cdc25

  TACC

  DOCK

  Clathrin

  MARP

  Lats kinase

  HGF

  Cdc20/PROTAC

  MRE11

  RNA polymerase 1

  DNA polymerase θ

  PBRM

  APC/PROTAC

  PD-1 PD-L1/PROTAC

  RNA polymerase 2

  PKMYT1

• Cytoskeleton

  +More

  Akt

  Bcr-Abl

  Dynamin

  FAK

  Gap Junction Protein

  HSP

  Integrin

  Kinesin

  Microtubule/Tubulin

  Mps1

  Myosin

  PAK

  Wnt

  β-catenin

  N-cadherin

  Selectin

  Arp2/3 Complex

  PKC

  Actin

  Spastin

  Gap Junction

  MLCK

  TACC

  FAK/PROTAC

  Filamin-A

  CYTH

• DNA Damage

  +More

  ATM/ATR

  DNA/RNA Synthesis

  DNA Alkylator/Crosslinker

  DNA-PK

  HDAC

  MTH1

  PARP

  Sirtuin

  Telomerase

  Topoisomerase

  AP endonuclease

  OGG

  ATAD5

  MRE11

  WRN

  BRCA

  RMI1

  RAD52

• Endocrinology/Hormones

  +More

  GHSR

  5 Alpha Reductase

  ACE

  Androgen Receptor

  Aromatase

  ERR

  Glucocorticoid Receptor

  GPCR

  Growth Hormone

  Opioid Receptor

  Progesterone Receptor

  Prolactin

  Renin

  TPO

  TRHR

  Thyroid Hormone Receptor

  AVT receptor

  TTR

  GHRP

  PTGR

  ER/PROTAC

• Epigenetics

  +More

  AMPK

  Aurora Kinase

  CECR2

  DNA Methyltransferase

  Epigenetic Reader Domain

  FACT

  HDAC

  HIF

  Histone Acetyltransferase

  Histone Demethylase

  Histone Methyltransferase

  JAK

  MicroRNA

  PAD

  PARP

  Pim

  PKC

  Sirtuin

  TET

  MBD-containing protein

  EZH2 (stapled peptide)

  HES

  FTO

  Sir2p

  PBRM

  PCAF/PROTAC

• GPCR/G Protein

  +More

  Adenosine Receptor

  Adiponectin Receptor

  Adrenergic Receptor

  Angiotensin Receptor

  Bombesin Receptor

  Bradykinin Receptor

  cAMP

  Cannabinoid Receptor

  CaSR

  CCR

  CGRP Receptor

  Cholecystokinin Receptor

  CRTH2

  CXCR

  Dopamine Receptor

  Endothelin Receptor

  GHSR

  Glucagon Receptor

  Glucocorticoid Receptor

  GNRH Receptor

  Guanylate Cyclase

  Hedgehog

  Histamine Receptor

  Imidazoline Receptor

  LPA Receptor

  LTR

  mGluR

  Motilin Receptor

  MT Receptor

  Neurotensin Receptor

  NK Receptor

  NMUR

  Opioid Receptor

  OX Receptor

  OXTR

  P2Y Receptor

  PAFR

  PAR

  PKA

  Prostaglandin Receptor

  Ras

  RGS

  S1P Receptor

  SGLT

  Sigma Receptor

  SSTR

  TSH Receptor

  Urotensin Receptor

  Vasopressin Receptor

  HDR

  CX3CR1

  GPR88

  LHCGR

  Melanocortin Receptor

  RAPGEF4

  SPHK

  5-HT Receptor

  AChR

  ACTH Receptor

  Apelin Receptor

  CRF Receptor

  GPCR

  Gsα

  LPL Receptor

  Neuropeptide Y Receptor

  SRPK

  Gi protein

  GalR

  SOS1

  STK19

  TAAR

  Epac

  G protein

  Endorphin

  SOS1/KRAS (stapled peptide)

  Rab (stapled peptide)

  SOS

  Calcitonin Receptor

  SUCNR1

  FSHR

  FPR

• Immunology/Inflammation

  +More

  CCR

  Complement System

  COX

  CRTH2

  CXCR

  FLAP

  Histamine Receptor

  IFNAR

  IL Receptor

  IRAK

  LTR

  MALT1

  NADPH Oxidase

  NLR

  NOS

  Nrf2

  PD-1/PD-L1

  PGE Synthase

  ROS

  SIK

  STING

  Thrombopoietin Receptor

  TLR

  Calcineurin

  Complement Receptor

  GM-CSF

  IFN

  IL

  IRF3

  MIF

  S100A9

  THPO

  TSPO

  cGAS

  Immunology & Inflammation Related

  LTA4H

  MyD88

  macrophage/microglia

  NPR

  NFAT

  FPR

  CYPA

  CD80

  Scavenger receptor

  NOT

  CD28-B7

  Endorphin

  LanC-like protein

  PG Synthase

  XBP1

  S100β

  Complement C3

  VISTA

  CD147

  NETosis

  SAMHD1

  CD38

• JAK/STAT Signaling

  EGFR

  JAK

  Pim

  STAT

  EGFR/PROTAC

  STAT/PROTAC

• LIF/Stat3

  LIF

• MAPK/ERK Pathway

  +More

  ERK

  JNK

  KLF

  MEK

  MLK

  MNK

  p38 MAPK

  Raf

  RSK

  ZAK

  Cot/tpl2

  MAP3K12

  MAP4K4

  AP-1

  HPK1

  TAOK

  MK2

  MAP4K6

• Membrane Transporter/Ion Channel

  +More

  AMPAR

  BCRP

  CFTR

  Chloride Channel

  CRAC Channel

  CRM1

  EAAT2

  HCN Channel

  MAT

  MCT

  Na+/Ca2+ Exchanger

  NKCC

  P2X Receptor

  P-gp

  Potassium Channel

  Proton Pump

  Sodium Channel

  TRPV

  URAT1

  VDAC

  GABA Receptor

  IBAT

  Oct

  SGLT

  AChR

  ATPase

  Calcium Channel

  EAAT1

  GlyT1

  Na+/K+ ATPase

  NBC

  NMDAR

  SV2

  TRP Channel

  SLC

  PIEZO1

  Glutamate transporter

  UCP

  ENT

  GABA transporter

  Glycine transporter

  Kainate receptor

  ABC Transporter

  Adaptor-associated kinase 1

  ABC Transporter

  ANT

  AKK1

  Efflux pump

  Clathrin

  Piezo

  OCTN

  AQP

  VRAC

  OAT

  sinus node I(f) channel

  GluR

  Transferrin Receptor

  NPC1L1

  CD147

  Organic Anion Transporter

  ARF

• Metabolic Enzyme

  +More

  15-PGDH

  ACC

  ACE

  Adenosine Deaminase

  Adenosine Kinase

  AhR

  ALDH

  Aldose Reductase

  Aminopeptidase

  ATP Citrate Lyase

  Carbonic Anhydrase

  Cathepsin

  CETP

  COMT

  CPA

  Decarboxylase

  Dehydrogenase

  DGAT

  DHFR

  Elastase

  Enolase

  FAAH

  FABP

  Factor Xa

  FAS

  Ferroptosis

  FXR

  Glucokinase

  GLUT1

  GSNOR

  GST

  Hexokinase

  HIF

  HIV Integrase

  HMGCR

  HSP

  Hydroxylase

  IDH

  IDO

  Lipase

  Lipoxygenase

  LXR

  MAO

  Mineralocorticoid Receptor

  NAE

  NAMPT

  Neprilysin

  P450

  PAI-1

  PDE

  PDHK

  PGC-1α

  Phospholipase

  Procollagen C Proteinase

  RAR/RXR

  Renin

  ROR

  SCD

  SGK

  Thioredoxin

  Thrombin

  Transferase

  VD/VDR

  Xanthine Oxidase

  Cholesterol Transporter

  CYP51

  Gluconeogenesis

  Glucosidase

  Glutaminase C

  Glycogenin

  Glyoxalase

  Ketohexokinase

  LDL

  Mitochondrial Electron Transport Chain

  Mitochondrial Metabolism

  MPC

  NQO1

  PGAM1

  PKM2

  Pyruvate Kinase

  TDO

  TGH

  Transketolase

  αKGD

  β-D-glucosidase

  2OG Oxygenase

  3-PGDH

  ACAT

  ACMSD

  Adenosylhomocysteinase

  AKR1B10

  Arginase

  ATP synthase

  Fumarate hydratase

  Steroid Sulfatase

  Phosphorylase

  Clp protease

  Galactosidases

  Heme polymerase

  Hydrolase

  MetAP

  NPR

  PFK

  FBPase

  ACS

  D-amino acid oxidase

  NQO2

  P448

  SOD2

  SPT

  Srx

  AO

  Proprotein convertases

  E-NTPDase

  ABHD12

  5 Alpha Reductase

  APOE

  Carboxylesterase

  CPSI

  GLUT

  QR

  sEH

  GPx

  G0/G1 switch protein 2

  GMPS

  CYPA

  PvdQ acylase

  BDK

  Creatine kinase

  NPP

  VDR (stapled peptide)

  NQO

  XBP1

  AKR

  HMG-CoA synthase

  RBP

  FTO

  D6D

  OGT

  ADP-ribosyltransferase

  ERAP

  LRH-1

  PASK

  PME-NMT

  PDE-NMT

  PEPCK

  Cardiolipin Peroxidase

  Aconitate hydratase

  Asparagine synthetase

  SGK3/PROTAC

  RAR/PROTAC

  OPA1

  NNMT

  6PGD

  CSE

  GAPDH

  HPSE

  PARG

  PI5P4K

  PKM1

  GCS

  LOX

  3MST

  Beta-glucuronidase

  FPR

  cGMP

• Neuronal Signaling

  +More

  AChE

  Adenosine Kinase

  Adrenergic Receptor

  AMPAR

  Amyloid-β

  CaMK

  CGRP Receptor

  COMT

  COX

  DAT

  Dopamine Receptor

  FAAH

  GABA Receptor

  GlyT1

  Histamine Receptor

  Imidazoline Receptor

  MAO

  mGluR

  MT Receptor

  NK Receptor

  NMDAR

  Opioid Receptor

  OX Receptor

  P2X Receptor

  P-gp

  Secretase

  SSRIs

  Substance P

  RyR1

  Choline

  Cholinesterase

  Enkephalinase

  GluCls

  Glucosylceramide Synthase

  Glutamate Release

  NET

  PSD-95

  RAGE

  SERT

  Sortilin

  5-HT Receptor

  AA-amyloid

  AChR

  PIEZO1

  Amylin receptor

  QC

  AQP4

  TAAR

  TLX

  CHT

  GABA transporter

  Glycine transporter

  Kainate receptor

  Endorphin

  S100β

  GluR

  NGF

  Ryanodine Receptor-1

  VIP

• PI3K/Akt/mTOR

  +More

  Akt

  AMPK

  ATM/ATR

  DNA-PK

  GSK-3

  MELK

  mTOR

  PDK-1

  PI3K

  PI4K

  PIKfyve

  PTEN

  RSK

  FOXO

  PHLPP

  PDK-4

  PDK

• Protease

  +More

  Caspase

  Cysteine Protease

  DPP4

  Glutaminase

  HIV Protease

  MMP

  Proteasome

  Secretase

  Ser/Thr Protease

  NEP

  PE

  Aspartic Protease

  Tyrosinase

  DPP2

  Dipeptidase 1

• Protein Tyrosine Kinase/RTK

  +More

  Ack1

  ALK

  Bcr-Abl

  BMX Kinase

  BTK

  c-FMS

  c-Kit

  c-Met/HGFR

  c-RET

  DDR1/DDR2 Receptor

  DYRK

  EGFR

  Ephrin Receptor

  FAK

  FGFR

  FLT3

  HER2

  IGF-1R

  Insulin Receptor

  ITK

  PDGFR

  PKA

  PTK

  Pyk2

  Ros1

  Src

  Syk

  TAM Receptor

  Tie-2

  Trk Receptor

  VEGFR

  CSK

  FLT4

  BRK

  MERTK

  FGF

  Tec

  ErbB

  BTK/PROTAC

  FLT3-ITD/PROTAC

  EGFR/PROTAC

  LTK

  INSRR

  GAK

• Stem Cells/Wnt

  +More

  Casein Kinase

  ERK

  Gli

  GSK-3

  Hedgehog

  JAK

  MST

  Notch

  PKA

  PORCN

  ROCK

  Secretase

  sFRP-1

  Smo

  STAT

  Wnt

  YAP

  β-catenin

  BMI-1

  Stemness Kinase

  TGF-beta Receptor

  14-3-3

  AAK1

  CREB

  Hes1

  β-catenin (stapled peptide)

  Notch (stapled peptide)

  PKA/AKAP (stapled peptide)

  MARP

  LIN28

  LRH-1

  HPK1

  STAT/PROTAC

  Notum

  MAP4K6

• TGF-beta/Smad

  TGF-beta Receptor

  Smad

  TGF-beta

  Smurf

  MARP

  Bcr-Abl

• Ubiquitin

  APC

  DUB

  NAE

  p97

  Proteasome

  E1/E2/E3 Enzyme

  SUMO

  FBXO

  Functionalized E3 Ligand (Bestatin)

  DCN

• Natural Product

  +More

  Alkaloids

  Cerebrosides

  Chalcones

  Coumarins

  Diterpenoids

  Flavonoids

  Iridoids

  Lignans

  Lipids

  Miscellaneous

  Monoterpenoids

  Naphthols

  Other Terpenoids

  Others-NP

  Phenols

  Phenylpropanoids

  Quinones

  Saccharides

  Sesquiterpenoids

  Steroids

  Tetraterpenoids

  Thiophenes

  Triterpenoids

  Xanthones

  Glycoside

  Terpenoids

• NF-κB

  +More

  HDAC

  IKK

  MALT1

  NF-κB

  NOD1

  Nrf2

  PPAR

  RIP Kinase

  TAK1

  Pirin

  LUBAC

  RIP Kinase/PROTAC

  TBK/PROTAC

• Biochemical Reagent

  Intermediate and Others

  Biochemical Assay Reagent

  Dye Reagent

  Cationic & Neutral Lipids

  Dendrimers

  LNA

• PROTAC

  E1/E2/E3 Enzyme

  Others-PROTAC

  MDM2/PROTAC

• Stapled Peptide

  +More

  Mcl-1 (stapled peptide)

  β-catenin (stapled peptide)

  EZH2 (stapled peptide)

  SOS1/KRAS (stapled peptide)

  Notch (stapled peptide)

  PKA/AKAP (stapled peptide)

  Beclin 1 (stapled peptide)

  Bim (stapled peptide)

  Bcl-2 (stapled peptide)

  p53/MDM2 (stapled peptide)

  RAP1/TRF2 (stapled peptide)

  Rab (stapled peptide)

  VDR (stapled peptide)

  β-arrestin/β-adaptin (stapled peptide)

• Others

  +More

  Phosphatase

  SRPK

  RyR1

  Cardiovascular Agent

  CBFβ-SMMHC

  Choleretic

  Diabetes

  Diuretic

  DNA Stain

  DprE1

  DUE-B

  E2F

  ECE

  ENT1

  ERO1

  FANCJ

  FAP

  Fer/FerT

  FPP synthase

  Fucosyltransferase

  Fungicide

  Galectin-3

  GBF1

  GCase

  HIPK2

  Histidine Kinase

  HPPD

  Importin β

  Insecticide

  LAT1

  MITF

  MLKL

  MPO

  MPTP

  MTP

  MTTP

  Muscle Relaxant

  Neuroprotection/Neurogenic Agents

  NMD

  NO Synthesis

  Nonsense-Suppressing Agent

  Nur77

  O-GlcNAcase

  Oligomer

  Osteoclasts/Bone/Osteogenesis

  Oxidosqualene Cyclase

  PAX2

  PBR

  PCA1

  PCSK9

  PDX1

  PEPT

  PFKFB3

  PHD

  Photosensitizer

  PIN1

  PKG

  Platelet

  PME-1

  PNP

  PREP

  Protein Synthesis

  PXR

  RasGAP

  Rev-ErbA

  RPE65

  SAP

  Serine Hydrolase

  Spermine Synthase

  SPPL2a

  SQS

  SREBP

  STK33

  Sweetener

  Tgase

  TIR1

  TNK

  TRIO

  UGT1A1

  Urease

  Vanin

  VAP-1

  VDA

  XOR

  Analgetic

  Anesthetic

  Anti-Coagulant/Procoagulant Agent

  Antispasmodic Agent

  Anti-Thyroid Agent

  Antitussive Agent

  Anti-ulcer

  BoNT A

  Cancer Stem Cells

  CD73

  CerK

  Chelating Agent

  Choline Kinase

  Differentiation/IPS

  DinG helicase

  CAR

  ITPKA

  Legumain

  Others-Others

  OxPhos

  Vitamin

  eEF2

  NT

  FBXO3

  GMPS

  metalloendopeptidase

  TXNRD1

  ATAD5

  PANK

  O-glycosylation

  DcpS

  GRK

  VPS4B

  TNIK

  RUNX

  HRGP

  20-HETE

  Cardiac transcription factor

  AIMP2-DX2

  PAM complex

  IMP1

  Quorum Sensing

  ASGPR

  SMARC

  PU.1

  HNF4α

  PNA

  PMO/MNA

  FLAT

  MALAT1

  VPS

  BBOX

  GTPCH

  FATP

  IKZF1

  IKZF2

  OSC

• Product Types:

  API

  Natural Products

  All Targets

  All Products

Researach Areas

• Others-Field:

• Cardiovascular DiseaseMetabolic Disease:

• Natural Product:

• Endocrinology:

• Others:

• Neurological Disease:

• Neurological Disease Cardiovascular Disease:

• Immunology/Inflammation:

• Cardiovascular Disease:

• Cancer:

  +More

  Leukemia

  Lymphoma

  Skin Cancer

  Pancreatic Cancer

  Multiple Myeloma

  Kidney (Renal Cell) Cancer

  Liver Cancer

  Thyroid Cancer

  Colon Cancer/Rectal Cancer

  Lung Cancer

  Ovarian Cancer

  Cervical Cancer

  Breast Cancer

  Prostate Cancer

• Infection:

  Influenza Virus

  HIV

  HBV

  HCV

• Inflammation:

  Pain

  Allergy

  Rheumatoid Arthritis

  Asthma

• Metabolic Disease:

  Obesity

  Diabetes

Antibody Drug Conjugates

• • Cytotoxins
  • Chemical linker and Intermidates
  • Payload with Linker
  • PEG analogs

Proteins/Peptides

• • Cytokines
  • Growth Factors
  • Chemokines
  • Neurotrophins
  • Hormones