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Adrenergic Receptor

Adrenergic Receptor

Cat. No. Product Name CAS No. Information
CSN24606 ZD 7114 HCl 129689-28-7 ZD 7114 hydrochloride is an agonist of β3-adrenoceptor.
CSN24046 Xamoterol 81801-12-9 Xamoterol hemifumarate is a selective partial agonist of β1-adrenoceptor.
CSN24598 WB 4101 HCl 2170-58-3 WB 4101 hydrochloride is a selective antagonist of α1A-adrenergic receptor.
CSN21863 Tiodazosin 66969-81-1 Tiodazosin is a potent competitive postsynaptic alpha adrenergic receptor antagonist.
CSN24706 Tampramine fumarate 83166-18-1 Tampramine is a tricyclic antidepressant (TCA). It acts as a selective norepinephrine reuptake inhibitor and has negligible affinity for adrenergic, histaminergic, and muscarinic receptors.
CSN24608 Talsupram HCl 25487-28-9 Talsupram hydrochloride is a selective noradrenalin re-uptake inhibitor.
CSN24600 SNAP 5089 HCl 157066-77-8 SNAP 5089 is a selective antagonist of α1A-adrenoceptor.
CSN24736 SNAP 5089 157066-76-7 SNAP 5089 is a selective antagonist of the subtype α1A-adrenoceptor. It binds with high affinity to α1A-adrenoceptor with a Ki value of 0.35 nM.
CSN24580 SKF 86466 HCl 86129-54-6 SKF 86466 hydrochloride is selective antagonist of pre- (Ki= 13 nM) and post-junctional (Ki= 17 nM) α2-adrenoceptors with antihypertensive activity in rat model.
CSN24586 RX 821002 HCl 109544-45-8 RX 821002 hydrochloride is a selective antagonist of α2-adrenoceptor with low affinity for imidazoline sites. The pKd values for α2D and α2A subtypes are 9.7 and 8.2 respectively.
CSN24579 RS 79948 HCl 186002-54-0 RS 79948 hydrochloride is an antagonist of α2-adrenoreceptor with Kd values are 0.18, 0.19 and 0.42 nM for α2B, α2C and α2A, respectively in rat. It can increase insulin secretion.
CSN24576 RS 17053 HCl 169505-93-5 RS 17053 hydrochloride is a selective antagonist of α1A-adrenoceptor with pKi and pA2 estimate of 9.1 - 9.9.
CSN26507 OPC-28326 HCl hydrate 167626-17-7 OPC-28326 is an adrenergic receptor antagonist potentially for the treatment of intermittent claudication and Raynaud's Syndrome
CSN24594 Naftopidil HCl 1164469-60-6 Naftopidil hydrochloride is antagonist of α1-adrenoceptor and has weak antagonism at post-junctional α2 receptors with persistent antihypertensive activity.
CSN26574 O-Desmethyl Mebeverine alcohol 155172-67-1 Mebeverine metabolite O-desmethyl Mebeverine alcohol is a metabolite of Mebeverine, which is a potent α1 repector inhibitor, causing relaxation of the gastrointestinal tract.
CSN21712 Lintopride 107429-63-0 Lintopride is an antagonist of 5HT4 receptor and moderate antagonist of 5HT3.
CSN24584 JP 1302 2HCl 1259314-65-2 JP 1302 dihydrochloride is an antagonist of α2C-adrenoceptor with Ki value of 28 nM.
CSN22006 Isoxsuprine-monoester-1 67160-74-1 Isoxsuprine-monoester-1, a monoester of isoxsuprine, is a long acting peripheral vasodilator.
CSN21958 Indanazoline 40507-78-6 Indanazoline is a sympathomimetic imidazoline derivative and shows vasoconstrictive action .
CSN24602 Imiloxan HCl 81167-22-8 Imiloxan hydrochloride is a highly selective antagonist of α2-adrenoceptor.
CSN24605 ICI 89406 53671-71-9 ICI 89406 is a β-adrenergic antagonist and low efficacy partial agonist; does not affect resting cardiac parameters.
CSN24607 HEAT HCl 30007-39-7 HEAT HCl is a very selective α1-adrenoceptor antagonist.
CSN26499 Fiduxosin free base 208993-54-8 Fiduxosin is an alpha(1)-adrenoceptor antagonist with higher affinity for alpha(1A)-adrenoceptors and for alpha(1D)-adrenoceptors than for alpha(1B)-adrenoceptors.
CSN24610 Efaroxan HCl 89197-00-2 Efaroxan hydrochloride is an antagonist of α2 adrenoceptor and imidazoline I1 receptor ligand. The pKi values are 7.87, 7.42, 5.74, 7.28 and < 5 for α2A, α2B, α2C, I1 and I2 receptors, respectively.
CSN26575 Detomidine carboxylic acid 115664-39-6 Detomidine carboxylic acid is the major urinary metabolite of Detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic sedative. Detomidine also has cardiac and respiratory effects and an antidiuretic action[1][2].
CSN26579 Dabuzalgron 219311-44-1 Dabuzalgron (previously codenamed R-450; Ro-115-1240) is a novel partial alphaA/IL receptor agonist that is administered in its hydrochloride form to control urethral smooth muscle contraction. The hemodynamic changes in the drug are very small and it is a potential drug for the treatment of stress urinary incontinence.
CSN26578 Clonidine(200mg) 4205-90-7 Clonidine (also known as Catapres, Kapvay, Nexiclon, and Clophelin) is a sympathomimetic medication used to treat high blood pressure, attention deficit hyperactivity disorder, anxiety disorders, withdrawal (from either alcohol, opioids, or smoking), migraine, menopausal flushing, diarrhea, and certain pain conditions. It is classified as a centrally acting α2 adrenergic agonist and imidazoline receptor agonist that has been in clinical use for over 40 years.
CSN24596 Cirazoline HCl 40600-13-3 Cirazoline hydrochloride is a selective agonist of alpha1-adrenoceptor.
CSN33167 Bucindolol 71119-11-4 Bucindolol is a high-affinity, competitive beta blocker.
CSN24591 BRL 37344 Sodium Salt 127299-93-8 BRL 37344 sodium salt is selective β3 adrenoceptor agonist with Ki values of 287, 1750 and 1120 nM for β3, β1 and β2 receptors respectively.
CSN24601 B-HT 933 2HCl 36067-72-8 B-HT 933 dihydrochloride is selective agonist of α2-adrenoceptor.
CSN24197 Arotinolol HCl 68377-91-3 Arotinolol is a blocker of both α- and β-receptor, and also acts as a β3 receptor agonist. It is used in the treatment of high blood pressure and essential tremor.
CSN24583 ARC 239 2HCl 55974-42-0 ARC 239 dihydrochloride is a selective antagonist of α2B adrenoceptor with pKD values of 8.8, 6.7 and 6.4 for α2B, α2A, and α2D receptors respectively.
CSN24581 A 80426 mesylate 152148-64-6 A 80426 mesylate is antagonist of α2-adrenoceptor and selective 5-HT uptake inhibitor with Ki values of 2.01 and 3.77 nM respectively. It also displays low affinity at homologous GPCRs.
CSN24599 A 61603 hydrobromide 107756-30-9 A 61603 hydrobromide is a selective α1A-adrenergic receptor agonist.
CSN24609 3-MPPI 133399-65-2 3-MPPI is a very potent ligand for α1 sites and regulates smooth muscle contraction. The pKi values for α1B, α1D, α1A adrenoceptors are 8.74, 9.44, 9.57 respectively. It also binds to 5-HT1A sites (Ki = 50 nM).
CSN24595 2-PMDQ 139047-55-5 2-PMDQ is a selective α1-adrenoceptor antagonist with antihypertensive effect.
CSN24597 2-MPMDQ 149847-77-8 2-MPMDQ is a selective antagonist of α1-AR adrenoceptor and can act as a hypotensive.
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