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Adrenergic Receptor
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN24606 | ZD 7114 HCl | 129689-28-7 | ZD 7114 hydrochloride is an agonist of β3-adrenoceptor. |
| CSN24046 | Xamoterol | 81801-12-9 | Xamoterol hemifumarate is a selective partial agonist of β1-adrenoceptor. |
| CSN24598 | WB 4101 HCl | 2170-58-3 | WB 4101 hydrochloride is a selective antagonist of α1A-adrenergic receptor. |
| CSN21863 | Tiodazosin | 66969-81-1 | Tiodazosin is a potent competitive postsynaptic alpha adrenergic receptor antagonist. |
| CSN24706 | Tampramine fumarate | 83166-18-1 | Tampramine is a tricyclic antidepressant (TCA). It acts as a selective norepinephrine reuptake inhibitor and has negligible affinity for adrenergic, histaminergic, and muscarinic receptors. |
| CSN24608 | Talsupram HCl | 25487-28-9 | Talsupram hydrochloride is a selective noradrenalin re-uptake inhibitor. |
| CSN24600 | SNAP 5089 HCl | 157066-77-8 | SNAP 5089 is a selective antagonist of α1A-adrenoceptor. |
| CSN24736 | SNAP 5089 | 157066-76-7 | SNAP 5089 is a selective antagonist of the subtype α1A-adrenoceptor. It binds with high affinity to α1A-adrenoceptor with a Ki value of 0.35 nM. |
| CSN24580 | SKF 86466 HCl | 86129-54-6 | SKF 86466 hydrochloride is selective antagonist of pre- (Ki= 13 nM) and post-junctional (Ki= 17 nM) α2-adrenoceptors with antihypertensive activity in rat model. |
| CSN24586 | RX 821002 HCl | 109544-45-8 | RX 821002 hydrochloride is a selective antagonist of α2-adrenoceptor with low affinity for imidazoline sites. The pKd values for α2D and α2A subtypes are 9.7 and 8.2 respectively. |
| CSN24579 | RS 79948 HCl | 186002-54-0 | RS 79948 hydrochloride is an antagonist of α2-adrenoreceptor with Kd values are 0.18, 0.19 and 0.42 nM for α2B, α2C and α2A, respectively in rat. It can increase insulin secretion. |
| CSN24576 | RS 17053 HCl | 169505-93-5 | RS 17053 hydrochloride is a selective antagonist of α1A-adrenoceptor with pKi and pA2 estimate of 9.1 - 9.9. |
| CSN26507 | OPC-28326 HCl hydrate | 167626-17-7 | OPC-28326 is an adrenergic receptor antagonist potentially for the treatment of intermittent claudication and Raynaud's Syndrome |
| CSN24594 | Naftopidil HCl | 1164469-60-6 | Naftopidil hydrochloride is antagonist of α1-adrenoceptor and has weak antagonism at post-junctional α2 receptors with persistent antihypertensive activity. |
| CSN26574 | O-Desmethyl Mebeverine alcohol | 155172-67-1 | Mebeverine metabolite O-desmethyl Mebeverine alcohol is a metabolite of Mebeverine, which is a potent α1 repector inhibitor, causing relaxation of the gastrointestinal tract. |
| CSN21712 | Lintopride | 107429-63-0 | Lintopride is an antagonist of 5HT4 receptor and moderate antagonist of 5HT3. |
| CSN24584 | JP 1302 2HCl | 1259314-65-2 | JP 1302 dihydrochloride is an antagonist of α2C-adrenoceptor with Ki value of 28 nM. |
| CSN22006 | Isoxsuprine-monoester-1 | 67160-74-1 | Isoxsuprine-monoester-1, a monoester of isoxsuprine, is a long acting peripheral vasodilator. |
| CSN21958 | Indanazoline | 40507-78-6 | Indanazoline is a sympathomimetic imidazoline derivative and shows vasoconstrictive action . |
| CSN24602 | Imiloxan HCl | 81167-22-8 | Imiloxan hydrochloride is a highly selective antagonist of α2-adrenoceptor. |
| CSN24605 | ICI 89406 | 53671-71-9 | ICI 89406 is a β-adrenergic antagonist and low efficacy partial agonist; does not affect resting cardiac parameters. |
| CSN24607 | HEAT HCl | 30007-39-7 | HEAT HCl is a very selective α1-adrenoceptor antagonist. |
| CSN26499 | Fiduxosin free base | 208993-54-8 | Fiduxosin is an alpha(1)-adrenoceptor antagonist with higher affinity for alpha(1A)-adrenoceptors and for alpha(1D)-adrenoceptors than for alpha(1B)-adrenoceptors. |
| CSN24610 | Efaroxan HCl | 89197-00-2 | Efaroxan hydrochloride is an antagonist of α2 adrenoceptor and imidazoline I1 receptor ligand. The pKi values are 7.87, 7.42, 5.74, 7.28 and < 5 for α2A, α2B, α2C, I1 and I2 receptors, respectively. |
| CSN26575 | Detomidine carboxylic acid | 115664-39-6 | Detomidine carboxylic acid is the major urinary metabolite of Detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic sedative. Detomidine also has cardiac and respiratory effects and an antidiuretic action[1][2]. |
| CSN26579 | Dabuzalgron | 219311-44-1 | Dabuzalgron (previously codenamed R-450; Ro-115-1240) is a novel partial alphaA/IL receptor agonist that is administered in its hydrochloride form to control urethral smooth muscle contraction. The hemodynamic changes in the drug are very small and it is a potential drug for the treatment of stress urinary incontinence. |
| CSN26578 | Clonidine(200mg) | 4205-90-7 | Clonidine (also known as Catapres, Kapvay, Nexiclon, and Clophelin) is a sympathomimetic medication used to treat high blood pressure, attention deficit hyperactivity disorder, anxiety disorders, withdrawal (from either alcohol, opioids, or smoking), migraine, menopausal flushing, diarrhea, and certain pain conditions. It is classified as a centrally acting α2 adrenergic agonist and imidazoline receptor agonist that has been in clinical use for over 40 years. |
| CSN24596 | Cirazoline HCl | 40600-13-3 | Cirazoline hydrochloride is a selective agonist of alpha1-adrenoceptor. |
| CSN33167 | Bucindolol | 71119-11-4 | Bucindolol is a high-affinity, competitive beta blocker. |
| CSN24591 | BRL 37344 Sodium Salt | 127299-93-8 | BRL 37344 sodium salt is selective β3 adrenoceptor agonist with Ki values of 287, 1750 and 1120 nM for β3, β1 and β2 receptors respectively. |
| CSN24601 | B-HT 933 2HCl | 36067-72-8 | B-HT 933 dihydrochloride is selective agonist of α2-adrenoceptor. |
| CSN24197 | Arotinolol HCl | 68377-91-3 | Arotinolol is a blocker of both α- and β-receptor, and also acts as a β3 receptor agonist. It is used in the treatment of high blood pressure and essential tremor. |
| CSN24583 | ARC 239 2HCl | 55974-42-0 | ARC 239 dihydrochloride is a selective antagonist of α2B adrenoceptor with pKD values of 8.8, 6.7 and 6.4 for α2B, α2A, and α2D receptors respectively. |
| CSN24581 | A 80426 mesylate | 152148-64-6 | A 80426 mesylate is antagonist of α2-adrenoceptor and selective 5-HT uptake inhibitor with Ki values of 2.01 and 3.77 nM respectively. It also displays low affinity at homologous GPCRs. |
| CSN24599 | A 61603 hydrobromide | 107756-30-9 | A 61603 hydrobromide is a selective α1A-adrenergic receptor agonist. |
| CSN24609 | 3-MPPI | 133399-65-2 | 3-MPPI is a very potent ligand for α1 sites and regulates smooth muscle contraction. The pKi values for α1B, α1D, α1A adrenoceptors are 8.74, 9.44, 9.57 respectively. It also binds to 5-HT1A sites (Ki = 50 nM). |
| CSN24595 | 2-PMDQ | 139047-55-5 | 2-PMDQ is a selective α1-adrenoceptor antagonist with antihypertensive effect. |
| CSN24597 | 2-MPMDQ | 149847-77-8 | 2-MPMDQ is a selective antagonist of α1-AR adrenoceptor and can act as a hypotensive. |
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