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Adrenergic Receptor

Adrenergic Receptor

Cat. No. Product Name CAS No. Information
CSN24598 WB 4101 HCl 2170-58-3 WB 4101 hydrochloride is a selective antagonist of α1A-adrenergic receptor.
CSN21863 Tiodazosin 66969-81-1 Tiodazosin is a potent competitive postsynaptic alpha adrenergic receptor antagonist.
CSN24706 Tampramine fumarate 83166-18-1 Tampramine is a tricyclic antidepressant (TCA). It acts as a selective norepinephrine reuptake inhibitor and has negligible affinity for adrenergic, histaminergic, and muscarinic receptors.
CSN24608 Talsupram HCl 25487-28-9 Talsupram hydrochloride is a selective noradrenalin re-uptake inhibitor.
CSN24600 SNAP 5089 HCl 157066-77-8 SNAP 5089 is a selective antagonist of α1A-adrenoceptor.
CSN24736 SNAP 5089 157066-76-7 SNAP 5089 is a selective antagonist of the subtype α1A-adrenoceptor. It binds with high affinity to α1A-adrenoceptor with a Ki value of 0.35 nM.
CSN24580 SKF 86466 HCl 86129-54-6 SKF 86466 hydrochloride is selective antagonist of pre- (Ki= 13 nM) and post-junctional (Ki= 17 nM) α2-adrenoceptors with antihypertensive activity in rat model.
CSN11918 Sertindole 106516-24-9 Sertindole, a neuroleptic, is one of the antipsychotic medications available, with a high affinity for dopamine D2, serotonin 5-HT2A, 5-HT2C, and α1-adrenergic receptors.
CSN24586 2-Methoxyidazoxan monohydrochloride 109544-45-8 RX 821002 hydrochloride is a selective antagonist of α2-adrenoceptor with low affinity for imidazoline sites. The pKd values for α2D and α2A subtypes are 9.7 and 8.2 respectively.
CSN24576 RS 17053 hydrochloride 169505-93-5 RS 17053 hydrochloride is a selective antagonist of α1A-adrenoceptor with pKi and pA2 estimate of 9.1 - 9.9.
CSN24584 JP1302 dihydrochloride 1259314-65-2 JP 1302 dihydrochloride is an antagonist of α2C-adrenoceptor with Ki value of 28 nM.
CSN21958 Indanazoline 40507-78-6 Indanazoline is a sympathomimetic imidazoline derivative and shows vasoconstrictive action .
CSN24602 Imiloxan HCl 81167-22-8 Imiloxan hydrochloride is a highly selective antagonist of α2-adrenoceptor.
CSN26499 Fiduxosin 208993-54-8 Fiduxosin is an alpha(1)-adrenoceptor antagonist with higher affinity for alpha(1A)-adrenoceptors and for alpha(1D)-adrenoceptors than for alpha(1B)-adrenoceptors.
CSN33116 Esreboxetine 98819-76-2 Esreboxetine is a selective norepinephrine reuptake inhibitor.
CSN24610 Efaroxan hydrochloride 89197-00-2 Efaroxan hydrochloride is an antagonist of α2 adrenoceptor and imidazoline I1 receptor ligand. The pKi values are 7.87, 7.42, 5.74, 7.28 and < 5 for α2A, α2B, α2C, I1 and I2 receptors, respectively.
CSN26575 Detomidine carboxylic acid 115664-39-6 Detomidine carboxylic acid is the major urinary metabolite of Detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic sedative. Detomidine also has cardiac and respiratory effects and an antidiuretic action[1][2].
CSN26579 Dabuzalgron 219311-44-1 Dabuzalgron (previously codenamed R-450; Ro-115-1240) is a novel partial alphaA/IL receptor agonist that is administered in its hydrochloride form to control urethral smooth muscle contraction. The hemodynamic changes in the drug are very small and it is a potential drug for the treatment of stress urinary incontinence.
CSN26578 Clonidine 4205-90-7 Clonidine (also known as Catapres, Kapvay, Nexiclon, and Clophelin) is a sympathomimetic medication used to treat high blood pressure, attention deficit hyperactivity disorder, anxiety disorders, withdrawal (from either alcohol, opioids, or smoking), migraine, menopausal flushing, diarrhea, and certain pain conditions. It is classified as a centrally acting α2 adrenergic agonist and imidazoline receptor agonist that has been in clinical use for over 40 years.
CSN24596 Cirazoline hydrochloride 40600-13-3 Cirazoline hydrochloride is a selective agonist of alpha1-adrenoceptor.
CSN24601 Azepexole dihydrochloride 36067-72-8 B-HT 933 dihydrochloride is selective agonist of α2-adrenoceptor.
CSN24583 ARC 239 dihydrochloride 55974-42-0 ARC 239 dihydrochloride is a selective antagonist of α2B adrenoceptor with pKD values of 8.8, 6.7 and 6.4 for α2B, α2A, and α2D receptors respectively.
CSN32920 Ampreloxetine 1227056-84-9 Ampreloxetine is a norepinephrine reuptake inhibitor.
CSN32921 Ampreloxetine HCl 1227056-87-2 Ampreloxetine is a norepinephrine reuptake inhibitor.
CSN24599 A-61603 107756-30-9 A 61603 hydrobromide is a selective α1A-adrenergic receptor agonist.
CSN24609 3-MPPI 133399-65-2 3-MPPI is a very potent ligand for α1 sites and regulates smooth muscle contraction. The pKi values for α1B, α1D, α1A adrenoceptors are 8.74, 9.44, 9.57 respectively. It also binds to 5-HT1A sites (Ki = 50 nM).
CSN24595 2-PMDQ 139047-55-5 2-PMDQ is a selective α1-adrenoceptor antagonist with antihypertensive effect.
CSN24597 2-MPMDQ 149847-77-8 2-MPMDQ is a selective antagonist of α1-AR adrenoceptor and can act as a hypotensive.
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