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Adenosine Receptor

Adenosine Receptor

Cat. No. Product Name CAS No. Information
CSN24475 Xanthine amine congener hydrochloride 1783977-95-6 XAC is an adenosine receptor antagonist with IC50 value of 16μM for Adenosine Receptor A2.
CSN19829 Trabodenoson 871108-05-3 Trabodenoson is a potent and highly selective adenosine A1 receptor agonist.
CSN16416 Theophylline   58-55-9 Theophylline is a natural product present in tea and cocoa working as a phosphodiesterase inhibitor adenosine receptor blocker and histone deacetylase activator
CSN27356 Taminadenant 1337962-47-6 Taminadenant is an antagonist of adenosine receptor.
CSN23108 SCH442416 316173-57-6 SCH-442416 is a selective adenosine A2A receptor antagonist. SCH-442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively). It displays > 23000-fold selectivity for hA2A over hA1 in vitro with minimal affinity for hA2B and hA3 receptors (IC50 > 10 μM).
CSN15960 Regadenoson 313348-27-5 Regadenoson is a selective adenosine A2A receptor agonist with Ki value of 1.1nM for pig striatum A2A receptor, used as a novel pharmacologic stress agent under clinical development for myocardial perfusion imaging.
CSN21946 Proxyphylline   603-00-9 Proxyphylline is a xanthine-derivatived antagonists of A1 and A2 adenosine receptors, which relaxe smooth muscles, particularly bronchial muscles.
CSN23050 PQ-69 910045-32-8 PQ 69 is a potent and selective A1 receptor inverse agonist taht exhibits high binding affinity at A1 receptor with Kis of 0.07 and 0.96 nM for rat and human receptors respectively.
CSN23113 SDZ WAG 994 130714-47-5 Potent, selective A1 agonist
CSN23153 TC-G 1004 1061747-72-5 Potent and selective A2A antagonist
CSN20000 Neladenoson dalanate 1239309-58-0 Neladenoson dalanate is a potent and selective adenosine A1 receptor agonist, and potentially useful for treatment of cardiovascular diseases.
CSN21751 5'-N-Ethylcarboxamidoadenosine 35920-39-9 NECA, an analog of adenosine, is agonist of adenosine receptors with Kis of 1880, 6660, and 3.5 nM for A1, A2A, and A3, respectively.
CSN22994 N6-Cyclopentyladenosine 41552-82-3 N6-Cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 2.3 nM for human A1 receptor.
CSN25517 N-(2-Hydroxyethyl)adenosine 4338-48-1 N-(2-Hydroxyethyl)adenosine has been studied as an anticonvulsant through the activation of adenosine A1 receptor (AA1R). It attenuates cell death induced by H2O2 through antioxidant action.
CSN24570 MRS1220 183721-15-5 MRS1220 is a potent and highly selective antagonist at the human A3 adenosine receptor. Ki values are 0.65, 305, and 52 nM at hA3, rA1 and rA2A respectively. MRS1220 displays an IC50 > 1 μM for inhibition of binding to rat A3 receptors.
CSN22990 MRS5698 1377273-00-1 MRS 5698 is a high affinity and selective A3 adenosine receptor agonist with Ki ~ 3 nM.
CSN22989 MRS-3777 hemioxalate 1186195-57-2 MRS 3777 Hemioxalate is a high affinity adenosine A3 receptor antagonist with Ki of 47 nM.
CSN22988 MRS 1754 264622-58-4 MRS 1754 is a selective adenosine A2B receptor antagonist with Ki of 1.97 nM for hA2B.
CSN22987 MRS-1706 264622-53-9 MRS 1706 is a potent and selective adenosine A2B receptor inverse agonist with Ki of 1.39 nM.
CSN22873 Rolofylline 136199-02-5 KW 3902 is a Selective adenosine A1 receptor antagonist with Ki of 0.19 nM.
CSN22860 ISAM-140 932191-62-3 ISAM 140 is a high affinity A2B receptor antagonist with Ki of 3.49 nM.
CSN23107 SCH 202676 Hydrobromide 265980-25-4 Inhibitor of ligand binding to G-protein-coupled receptors
CSN16958 Piclidenoson   152918-18-8 IB-MECA is an agonist of the adenosine A3 receptor with EC50 values of 0.11 M. IB-MECA is a potent and selective A3 adenosine receptor agonist with Ki value of 1.1, 54 and 56 nM for A3, A1 and A2A receptors, respectively, which possessing cardioprotective effect and reduces infarct size upon reperfusion in rats.
CSN22848 HEMADO 403842-38-6 HEMADO is a high affinity and selective adenosine A3 receptor agonist with Ki of 1.1 nM for human A3.
CSN17618 GR79236 124555-18-6 GR79236 is a highly potent and selective adenosine A1 receptor agonist (Ki 3.1 nM) that has analgesic and anti-inflammatory actions in humans and animals.
CSN22792 DPCPX 102146-07-6 DPCPX is a potent and selective A1 adenosine receptor antagonist, both in vitro and in vivo, with Ki of 3.9 nM for human A1.
CSN23120 Derenofylline 251945-92-3 Derenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. Derenofylline suppresses cardiac fibrosis and attenuates albuminuria without affecting blood pressure in rats[1].
CSN22838 GS-6201 752222-83-6 CVT-6883 is a selective antagonist of adenosine A2B receptors with Ki of 22 nM for human A2B.
CSN21199 Ciforadenant(CPI-444) 1202402-40-1 CPI-444 is an orally administered antagonist of the adenosine A2A receptor. Upon oral administration, CPI-444 binds to adenosine A2A receptors expressed on the surface of immune cells, including T-lymphocytes, natural killer (NK) cells, macrophages and dendritic cells (DCs).
CSN24568 CGS 15943 104615-18-1 CGS 15943 is a potent adenosine receptor antagonist with Ki values of 3.5, 4.2, 16 and 51 nM for human A1, A2A, A2B and A3 receptors respectively.
CSN23897 BAY-545 1699717-32-2 BAY-545 is a structure-optimizd adenosine receptor A2B antagonist with IC50 value of of 59 nM.
CSN24164 BAY-218   2162982-11-6 BAY-218 is an AHR antagonist.
CSN22708 BAY 60-6583 910487-58-0 BAY 60-6583 is a potent adenosine A2B receptor agonist with EC50 of 2.83 nM for murine A2B receptor.
CSN27286 BAY 2416964 2242464-44-2 BAY 2416964 is an antagonist of aryl hydrocarbon receptor (AhR) with IC50 of 341 nM.
CSN23524 Adenosine   58-61-7 Adenosine is a nucleoside that is composed of adenine and d-ribose and plays many important biological roles in addition to being components of DNA and RNA.
CSN25244 Adenosine amine congener 96760-69-9 Adenosine amine congener hydrate is a potent aqueous-soluble A1 adenosine receptor agonist with Ki value of 0.85nM for binding against [3H]N6-cyclohexyladenosine in rat cerebral cortex membranes.
CSN24753 AB928 2239273-34-6 AB928 is a dual A2aR/A2bR antagonist that inhibits A2aR and A2bR with an equilibrium binding constant of 1.4 and 2 nM, respectively.
CSN18264 A2AR-agonist-1 41552-95-8 A2AR-agonist-1 is a potent A2AR and ENT1 agonist with Ki of 4.39 and 3.47 for A2AR and ENT1.
CSN17107 Namodenoson (CF-102)   163042-96-4 2-Cl-IB-MECA is a highly selective A3 adenosine receptor agonist with Ki value of 0.33nM, displaying 2500- and 1400-fold selectivity over A1 and A2A receptors, respectively.
CSN22645 2-Chloro-N6-cyclopentyladenosine 37739-05-2 2-Chloro-N6-cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 0.8 nM for human A1.
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