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Adenosine Receptor
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN24475 | Xanthine amine congener hydrochloride | 1783977-95-6 | XAC is an adenosine receptor antagonist with IC50 value of 16μM for Adenosine Receptor A2. |
| CSN19829 | Trabodenoson | 871108-05-3 | Trabodenoson is a potent and highly selective adenosine A1 receptor agonist. |
| CSN16416 | Theophylline | 58-55-9 | Theophylline is a natural product present in tea and cocoa working as a phosphodiesterase inhibitor adenosine receptor blocker and histone deacetylase activator |
| CSN27356 | Taminadenant | 1337962-47-6 | Taminadenant is an antagonist of adenosine receptor. |
| CSN23108 | SCH442416 | 316173-57-6 | SCH-442416 is a selective adenosine A2A receptor antagonist. SCH-442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively). It displays > 23000-fold selectivity for hA2A over hA1 in vitro with minimal affinity for hA2B and hA3 receptors (IC50 > 10 μM). |
| CSN15960 | Regadenoson | 313348-27-5 | Regadenoson is a selective adenosine A2A receptor agonist with Ki value of 1.1nM for pig striatum A2A receptor, used as a novel pharmacologic stress agent under clinical development for myocardial perfusion imaging. |
| CSN21946 | Proxyphylline | 603-00-9 | Proxyphylline is a xanthine-derivatived antagonists of A1 and A2 adenosine receptors, which relaxe smooth muscles, particularly bronchial muscles. |
| CSN23050 | PQ-69 | 910045-32-8 | PQ 69 is a potent and selective A1 receptor inverse agonist taht exhibits high binding affinity at A1 receptor with Kis of 0.07 and 0.96 nM for rat and human receptors respectively. |
| CSN23113 | SDZ WAG 994 | 130714-47-5 | Potent, selective A1 agonist |
| CSN23153 | TC-G 1004 | 1061747-72-5 | Potent and selective A2A antagonist |
| CSN20000 | Neladenoson dalanate | 1239309-58-0 | Neladenoson dalanate is a potent and selective adenosine A1 receptor agonist, and potentially useful for treatment of cardiovascular diseases. |
| CSN21751 | 5'-N-Ethylcarboxamidoadenosine | 35920-39-9 | NECA, an analog of adenosine, is agonist of adenosine receptors with Kis of 1880, 6660, and 3.5 nM for A1, A2A, and A3, respectively. |
| CSN22994 | N6-Cyclopentyladenosine | 41552-82-3 | N6-Cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 2.3 nM for human A1 receptor. |
| CSN25517 | N-(2-Hydroxyethyl)adenosine | 4338-48-1 | N-(2-Hydroxyethyl)adenosine has been studied as an anticonvulsant through the activation of adenosine A1 receptor (AA1R). It attenuates cell death induced by H2O2 through antioxidant action. |
| CSN24570 | MRS1220 | 183721-15-5 | MRS1220 is a potent and highly selective antagonist at the human A3 adenosine receptor. Ki values are 0.65, 305, and 52 nM at hA3, rA1 and rA2A respectively. MRS1220 displays an IC50 > 1 μM for inhibition of binding to rat A3 receptors. |
| CSN22990 | MRS5698 | 1377273-00-1 | MRS 5698 is a high affinity and selective A3 adenosine receptor agonist with Ki ~ 3 nM. |
| CSN22989 | MRS-3777 hemioxalate | 1186195-57-2 | MRS 3777 Hemioxalate is a high affinity adenosine A3 receptor antagonist with Ki of 47 nM. |
| CSN22988 | MRS 1754 | 264622-58-4 | MRS 1754 is a selective adenosine A2B receptor antagonist with Ki of 1.97 nM for hA2B. |
| CSN22987 | MRS-1706 | 264622-53-9 | MRS 1706 is a potent and selective adenosine A2B receptor inverse agonist with Ki of 1.39 nM. |
| CSN22873 | Rolofylline | 136199-02-5 | KW 3902 is a Selective adenosine A1 receptor antagonist with Ki of 0.19 nM. |
| CSN22860 | ISAM-140 | 932191-62-3 | ISAM 140 is a high affinity A2B receptor antagonist with Ki of 3.49 nM. |
| CSN23107 | SCH 202676 Hydrobromide | 265980-25-4 | Inhibitor of ligand binding to G-protein-coupled receptors |
| CSN16958 | Piclidenoson | 152918-18-8 | IB-MECA is an agonist of the adenosine A3 receptor with EC50 values of 0.11 M. IB-MECA is a potent and selective A3 adenosine receptor agonist with Ki value of 1.1, 54 and 56 nM for A3, A1 and A2A receptors, respectively, which possessing cardioprotective effect and reduces infarct size upon reperfusion in rats. |
| CSN22848 | HEMADO | 403842-38-6 | HEMADO is a high affinity and selective adenosine A3 receptor agonist with Ki of 1.1 nM for human A3. |
| CSN17618 | GR79236 | 124555-18-6 | GR79236 is a highly potent and selective adenosine A1 receptor agonist (Ki 3.1 nM) that has analgesic and anti-inflammatory actions in humans and animals. |
| CSN23120 | Derenofylline | 251945-92-3 | Derenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. Derenofylline suppresses cardiac fibrosis and attenuates albuminuria without affecting blood pressure in rats[1]. |
| CSN21199 | Ciforadenant(CPI-444) | 1202402-40-1 | CPI-444 is an orally administered antagonist of the adenosine A2A receptor. Upon oral administration, CPI-444 binds to adenosine A2A receptors expressed on the surface of immune cells, including T-lymphocytes, natural killer (NK) cells, macrophages and dendritic cells (DCs). |
| CSN24568 | CGS 15943 | 104615-18-1 | CGS 15943 is a potent adenosine receptor antagonist with Ki values of 3.5, 4.2, 16 and 51 nM for human A1, A2A, A2B and A3 receptors respectively. |
| CSN23897 | BAY-545 | 1699717-32-2 | BAY-545 is a structure-optimizd adenosine receptor A2B antagonist with IC50 value of of 59 nM. |
| CSN24164 | BAY-218 | 2162982-11-6 | BAY-218 is an AHR antagonist. |
| CSN27286 | BAY 2416964 | 2242464-44-2 | BAY 2416964 is an antagonist of aryl hydrocarbon receptor (AhR) with IC50 of 341 nM. |
| CSN23524 | Adenosine | 58-61-7 | Adenosine is a nucleoside that is composed of adenine and d-ribose and plays many important biological roles in addition to being components of DNA and RNA. |
| CSN25244 | Adenosine amine congener | 96760-69-9 | Adenosine amine congener hydrate is a potent aqueous-soluble A1 adenosine receptor agonist with Ki value of 0.85nM for binding against [3H]N6-cyclohexyladenosine in rat cerebral cortex membranes. |
| CSN24753 | AB928 | 2239273-34-6 | AB928 is a dual A2aR/A2bR antagonist that inhibits A2aR and A2bR with an equilibrium binding constant of 1.4 and 2 nM, respectively. |
| CSN18264 | A2AR-agonist-1 | 41552-95-8 | A2AR-agonist-1 is a potent A2AR and ENT1 agonist with Ki of 4.39 and 3.47 for A2AR and ENT1. |
| CSN17107 | Namodenoson (CF-102) | 163042-96-4 | 2-Cl-IB-MECA is a highly selective A3 adenosine receptor agonist with Ki value of 0.33nM, displaying 2500- and 1400-fold selectivity over A1 and A2A receptors, respectively. |
| CSN22645 | (2R,3R,4S,5R)-2-(2-Chloro-6-(cyclopentylamino)-9H-purin-9-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | 37739-05-2 | 2-Chloro-N6-cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 0.8 nM for human A1. |
| CSN51551 | 4-Nitrophenyl hydrogen phenylphosphonate | 57072-35-2 |
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