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Adenosine Receptor

Adenosine Receptor

Cat. No. Product Name CAS No. Information
CSN12242 ZM241385 139180-30-6 ZM241385 is a high affinity antagonist ligand selective for the adenosine A2A receptor
CSN19381 Xanthine   69-89-6 Xanthine is a natural occuring purine-base adenosine receptor antagonist from which a number of stimulants such as caffeine and theobromine are derived
CSN19829 Trabodenoson 871108-05-3 Trabodenoson is a potent and highly selective adenosine A1 receptor agonist.
CSN13164 Tozadenant   870070-55-6 Tozadenant is a selective adenosine A2A receptor antagonist with Ki values of 115 nM on human A2A and 6 nM on rhesus A2A which can improve motor function in animal models of Parkinsons disease
CSN21258 Tecadenoson 204512-90-3 Tecadenoson is a selective A1 adenosine receptor agonist
CSN11901 SCH-58261 160098-96-4 SCH 58261 is a potent and selective A2a adenosine receptor antagonist with Ki of 23 nM and 2 nM for rat A2a and bovine A2a respectively
CSN15960 Regadenoson 313348-27-5 Regadenoson is a selective adenosine A2A receptor agonist with Ki value of 1.1nM for pig striatum A2A receptor, used as a novel pharmacologic stress agent under clinical development for myocardial perfusion imaging.
CSN23056 PSB 36 524944-72-7 PSB 36 is a potent and selective A1 adenosine receptor antagonist that displays binding affinity of 0.12 nM for rA1.
CSN23054 PSB 0788 1027513-54-7 PSB 0788 is a potent and selective adenosine A2B receptor antagonist with IC50 of 3.64 nM at human A2B receptor.
CSN21946 Proxyphylline   603-00-9 Proxyphylline is a xanthine-derivatived antagonists of A1 and A2 adenosine receptors, which relaxe smooth muscles, particularly bronchial muscles.
CSN11787 Propentofylline 55242-55-2 Propentofylline a xanthine derivative with purported neuroprotective effects acts as a c-AMP phosphodiesterase inhibitor a nerve growth factor stimulator an adenosine transport inhibitor and a non-selective adenosine receptor antagonist
CSN12717 Preladenant   377727-87-2 Preladenant is a highly selective and competitive A2A receptor antagonist with Ki value of 11nM used in trials studying the treatment of brain diseases such as parkinson disease movement disorders antipsychotic agents and parkinsonian disorders
CSN13188 PD117519 96392-15-3 PD117519 is an adenosine agonist
CSN16615 Norisoboldine 23599-69-1 Norisoboldine is an isoquinoline alkaloid isolated and purfied from the roots of Lindera aggregata, which acts as an AhR agonist, and enhances the function of the adenosine A1 receptor.
CSN20000 Neladenoson Dalanate 1239309-58-0 Neladenoson dalanate is a potent and selective adenosine A1 receptor agonist, and potentially useful for treatment of cardiovascular diseases.
CSN21751 NECA 35920-39-9 NECA, an analog of adenosine, is agonist of adenosine receptors with Kis of 1880, 6660, and 3.5 nM for A1, A2A, and A3, respectively.
CSN22994 N6-Cyclopentyladenosine 41552-82-3 N6-Cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 2.3 nM for human A1 receptor.
CSN11502 N6-Cyclohexyladenosine 36396-99-3 N6-Cyclohexyladenosine is a selective A1 receptor agonist EC50 82 nM
CSN18631 N-[(4-Aminophenyl)methyl]adenosine 95523-13-0 N-4-Aminophenylmethyladenosine is an adenosine receptor inhibitor with Ki of 29 nM for rat ecto-5-nucleotidase
CSN22990 MRS 5698 1377273-00-1 MRS 5698 is a high affinity and selective A3 adenosine receptor agonist with Ki ~ 3 nM.
CSN22988 MRS 1754 264622-58-4 MRS 1754 is a selective adenosine A2B receptor antagonist with Ki of 1.97 nM for hA2B.
CSN22987 MRS 1706 264622-53-9 MRS 1706 is a potent and selective adenosine A2B receptor inverse agonist with Ki of 1.39 nM.
CSN19808 LAS38096 851371-22-7 LAS38096 is a potent selective and efficacious A2B adenosine receptor antagonist
CSN16958 IB-MECA   152918-18-8 IB-MECA is an agonist of the adenosine A3 receptor with EC50 values of 0.11 M. IB-MECA is a potent and selective A3 adenosine receptor agonist with Ki value of 1.1, 54 and 56 nM for A3, A1 and A2A receptors, respectively, which possessing cardioprotective effect and reduces infarct size upon reperfusion in rats.
CSN22848 HEMADO 403842-38-6 HEMADO is a high affinity and selective adenosine A3 receptor agonist with Ki of 1.1 nM for human A3.
CSN17618 GR79236 124555-18-6 GR79236 is a highly potent and selective adenosine A1 receptor agonist (Ki 3.1 nM) that has analgesic and anti-inflammatory actions in humans and animals.
CSN10909 Enprofylline 41078-02-8 Enprofylline is a xanthine derivative used in the treatment of asthma, which acts as a bronchodilator.
CSN22792 DPCPX 102146-07-6 DPCPX is a potent and selective A1 adenosine receptor antagonist, both in vitro and in vivo, with Ki of 3.9 nM for human A1.
CSN22838 CVT-6883 752222-83-6 CVT-6883 is a selective antagonist of adenosine A2B receptors with Ki of 22 nM for human A2B.
CSN21199 CPI444 1202402-40-1 CPI-444 is an orally administered antagonist of the adenosine A2A receptor. Upon oral administration, CPI-444 binds to adenosine A2A receptors expressed on the surface of immune cells, including T-lymphocytes, natural killer (NK) cells, macrophages and dendritic cells (DCs).
CSN10605 CGS 21680 120225-54-9 CGS 21680 is an adenosine A2 receptor agonist with IC50 of 22 nM exhibits 140-fold over A1 receptor
CSN18682 CGS 21680 HCl 124431-80-7 CGS 21680 HCl is A2A adenosine receptor agonist with Ki value of 27 nM which can be used to distinguish A2A- and A2B-mediated effect and shows affinity for both A1 and A3 adenosine receptors
CSN10537 Capadenoson 544417-40-5 Capadenoson is an oral active potent and selective adenosine A1 receptor agonist
CSN24164 BAY-218 2162982-11-6 BAY-218 is an AHR antagonist.
CSN22708 BAY 60-6583 910487-58-0 BAY 60-6583 is a potent adenosine A2B receptor agonist with EC50 of 2.83 nM for murine A2B receptor.
CSN21201 AZD4635 1321514-06-0 AZD4635 is an A2AR antagonist which can reverse adenosine mediated T cell suppression
CSN21468 Alloxazine 490-59-5 Alloxazine is a selective antagonist of A2B adenosine receptor.
CSN21333 Adenosine Antagonist-1 431040-19-6 Adenosine antagonist-1 is an adenosine A3 receptor AA3R antagonist
CSN12871 Acefylline   652-37-9 Acefylline is an adenosine receptor antagonist, a stimulant drug of the xanthine chemical class.
CSN18264 A2AR-Agonist-1 41552-95-8 A2AR-agonist-1 is a potent A2AR and ENT1 agonist with Ki of 4.39 and 3.47 for A2AR and ENT1.
CSN17107 2-Cl-IB-MECA   163042-96-4 2-Cl-IB-MECA is a highly selective A3 adenosine receptor agonist with Ki value of 0.33nM, displaying 2500- and 1400-fold selectivity over A1 and A2A receptors, respectively.
CSN22645 2-Chloro-N6-cyclopentyladenosine 37739-05-2 2-Chloro-N6-cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist with Ki of 0.8 nM for human A1.
CSN22617 (±)-5'-Chloro-5'-deoxy-ENBA 103626-26-2 (±)-5'-Chloro-5'-deoxy-ENBA is a highly selective adenosine A1 receptor agonist with Ki of 0.51 nM.
CSN23108 SCH 442416 316173-57-6
CSN23113 SDZ WAG 994 130714-47-5
CSN23120 SLV 320 251945-92-3
CSN23153 TC-G 1004 1061747-72-5
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