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Ack1

Ack1

Cat. No. Product Name CAS No. Information
CSN18846 XMD8-87 1234480-46-6 XMD8-87 is a tyrosine kinase nonreceptor 2 TNK2 inhibitor with IC50s of 38 nmolL and 113 nmolL for the D163E and R806Q mutations
CSN18847 XMD16-5 1345098-78-3 XMD16-5 is an inhibitor of TNK2 with IC50 value of 038M potently inhibiting phosphorylation of TNK2 truncation mutations found in solid tumor types
CSN17890 KRCA-0008 1472795-20-2 KRCA-0008 is a potent and selective ALKAck1 inhibitor with IC50 of 12 nM4 nM for ALK and Ack1 respectively and displays drug-like properties without hERG liability
CSN16660 AIM-100 873305-35-2 AIM-100 is a potent and selective Ack1 TNK2 inhibitor with IC50 value of 22nM showing suppression phosphorylation of Tyr267 of the androgen receptor in prostate cancer cells
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