Welcome to CSNpharm! For Research Use Only!
Ack1
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN18846 | XMD8-87 | 1234480-46-6 | XMD8-87 is a tyrosine kinase nonreceptor 2 TNK2 inhibitor with IC50s of 38 nmolL and 113 nmolL for the D163E and R806Q mutations |
| CSN18847 | XMD16-5 | 1345098-78-3 | XMD16-5 is an inhibitor of TNK2 with IC50 value of 038M potently inhibiting phosphorylation of TNK2 truncation mutations found in solid tumor types |
| CSN26520 | Mps1-IN-1 dihydrochloride | 1883548-93-3 | Mps1-IN-1 dihydrochloride is a potent, selective and ATP-competitive Mps1 kinase inhibitor, with an IC50 and a Kd of 367 nM and 27 nM[1]. |
| CSN17890 | KRCA-0008 | 1472795-20-2 | KRCA-0008 is a potent and selective ALKAck1 inhibitor with IC50 of 12 nM4 nM for ALK and Ack1 respectively and displays drug-like properties without hERG liability |
| CSN16660 | AIM-100 | 873305-35-2 | AIM-100 is a potent and selective Ack1 TNK2 inhibitor with IC50 value of 22nM showing suppression phosphorylation of Tyr267 of the androgen receptor in prostate cancer cells |
+1-708-781-1677
+1-708-286-6026
sales@csnpharm.com
