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AChR

AChR

Cat. No. Product Name CAS No. Information
CSN24514 α-Conotoxin PnIA 705300-84-1 α-Conotoxin PnIA is a selective antagonist of α3β2 nAChR receptors (IC50 = 9.56 nM) and α7 receptors (IC50 = 252 nM).
CSN24553 α-Conotoxin M II 175735-93-0 α-Conotoxin MII is a potent and selective α3β2 and β3 nAChR antagonist.
CSN24544 α-Conotoxin EI 170663-33-9 α-Conotoxin EI is a selective antagonist of neuromuscular nicotinic receptors α1β1γδ with IC50 of 187 nM.
CSN24535 α-Conotoxin Au IB 216299-21-7 α-Conotoxin AuIB is a selective antagonist of α3β4 nicotinic acetylcholine receptors.
CSN24539 Zamifenacin fumarate 127308-98-9 Zamifenacin fumarate is a selective M3 muscarinic receptor antagonist with pKi value of 8.52.
CSN24545 VU 10010 633283-39-3 VU 10010 is a selective allosteric potentiator of M4 acetylcholine receptor.
CSN24529 VU 0238429 1160247-92-6 VU 0238429 is a selective positive allosteric modulator of M5 receptors with EC50 values of 1.16, >30 and >30 μM at M5, M1 and M3 receptors respectively.
CSN21894 Vinconate 70704-03-9 Vinconate is an indolonaphthyridine derivative and can stimulate the muscariic acetylcholine receptor.
CSN21914 Tiotropium Bromide H2O 411207-31-3 Tiotropium Bromide is an considsered a long acting muscarinic receptor antagonist (LAMA) and is used clinically as an inhaled bronchodilator for COPD and asthma.
CSN21862 SA-504 35035-05-3 Timepidium bromide is an anticholinergic agent.
CSN21860 tigloidine 495-83-0 Tigloidin is an analogue of atropine with anticholinergic activity.
CSN21851 Tematropium 113932-41-5 Tematropium (CDDD3602) is a soft anticholinergics.
CSN23115 SIB 1553A HCl 191611-89-9 SIB-1553A is a nicotinic acetylcholine receptor agonist potentially for the treatment of Alzheimer’s disease (AD).
CSN24554 SEN 12333 874450-44-9 SEN 12333 is a selective agonist of α7 nicotinic acetylcholine receptor (nAChR) with EC50 and Ki of 1.6 μM, 260 nM in rat. It also displays functional antagonism at histamine H3 receptors (IC50 = 103 nM).
CSN24694 (R)-N-(Quinuclidin-3-yl)-2,3-dihydrobenzo[b][1,4]dioxine-6-carboxamide fumarate 527680-57-5 Selective α7 nAChR agonist
CSN23842 Scopolamine N-Oxide HydrobroMide Monohydrate N/A Scopolamine N-oxide hydrobromide is an antagonist of the muscarinic acetylcholine.
CSN24550 RuBi-Nicotine 1256362-30-7 RuBi-Nicotine is a caged nicotine that is nicotinic acetylcholine receptor (nAChR) agonist.
CSN21821 Rapacuronium 156137-99-4 Rapacuronium is an allosteric modulator of muscarinic acetylcholine receptor (mAChR). It is an aminosteroidal nondepolarizing neuromuscular blocking agent and used as a anesthesia.
CSN25236 Pirmenol 68252-19-7 Pirmenol inhibited the muscarinic acetylcholine receptor-operated K+ current (I[K.ACh]) in atrial cells and on experimental atrial fibrillation in isolated guinea-pig hearts.
CSN24691 (R)-N-(Furo[2,3-c]pyridin-5-ylmethyl)quinuclidin-3-amine 478149-53-0 PHA-543613 acts as a potent and selective agonist for the α7 subtype of neural nicotinic acetylcholine receptors, with a high level of brain penetration and good oral bioavailability. It is under development as a possible treatment for cognitive deficits in schizophrenia.
CSN24541 Perlapine 1977-11-3 Perlapine is a potent muscarinic DREADD agonist.
CSN24528 PD 102807 23062-91-1 PD 102807 is a selective M4 muscarinic receptor antagonist with IC50 values of 91, 6559, 3441, 950 and 7412 nM for human M4, M1, M2, M3, and M5 receptors respectively.
CSN24547 Oxotremorine sesquifumarate 17360-35-9 Oxotremorine sesquifumarate is a muscarinic agonist.
CSN24546 N,N,N-Trimethyl-4-(2-oxopyrrolidin-1-yl)but-2-yn-1-aminium iodide 3854-04-4 Oxotremorine M iodide is a potent and selective muscarinic acetylcholine receptor (mAChR) agonist. Oxotremorine M iodide potentiates NMDA receptors by muscarinic receptor dependent and independent mechanisms[1].
CSN21769 Nuvenzepine 96487-37-5 Nuvenzepine is an antagonist of musccarinic M3 which is used to treat gastrospasm.
CSN24692 3-(3-Bromothiophen-2-yl)-8-methyl-8-azabicyclo[3.2.1]oct-2-ene fumarate 216853-60-0 NS3861 is an α3β2 full agonist and an α3β4 partial agonist.
CSN24538 McN-A 343 55-45-8 McN-A 343 is a selective muscarinic M1 receptor agonist.
CSN24690 1,4-Diazabicyclo[3.2.2]nonan-4-yl(5-(3-(trifluoromethyl)phenyl)furan-2-yl)methanone hydrochloride 753499-14-8 High affinity α7 nAChR partial agonist; anti-inflammatory
CSN22004 ENS-163 phosphate 117707-51-4 ENS-163 phosphate is a selective muscarinic M1 receptor agonist.
CSN21625 Elucaine 25314-87-8 Elucaine is an antagonist of muscarinic acetylcholine receptor with anti-ulcerative activity.
CSN24537 DMP 543 160588-45-4 DMP 543 is a sitmulator of acetylcholine release. It can enhance K+-stimulated [3H]-ACh release from rat hippocampal slices (EC50 = 700 nM) and increase release of dopamine and glutamate (EC50 = 0.25 and 0.22 μM, respectively). 
CSN20950 delsoline 509-18-2 Delsoline is found in the roots of aonitum carmichaeli debx with hypotensive effects.
CSN24540 DAU 5884 HCl 131780-48-8 DAU 5884 HCl is a selective muscarinic M3 receptor antagonist.
CSN21591 Darenzepine 84629-61-8 Darenzepine is an inhibitor of muscarinic receptor.
CSN22098 Ambutonium Bromide 115-51-5 Ambutonium bromide is an acetylcholine antagonist.
CSN24516 A 85380 dihydrochloride 174740-86-4 A 85380 dihydrochloride is a high affinity and selective agonist of α4β2 nACh receptor with Ki of 0.05.
CSN24536 5-Iodo-A-85380 dihydrochloride 1217837-17-6 5-Iodo-A-85380 dihydrochloride is selective agonist of the α4β2 and α6β2 nicotinic acetylcholine receptors.
CSN24533 4-Acetyl-1,1-dimethylpiperazinium iodide 75667-84-4 4-Acetyl-1,1-dimethylpiperazinium iodide is a nAChR agonist with Ki of 29.9 nM at α4β2.
CSN24530 (¡À)-Anatoxin A fumarat 1219922-30-1 (¡À)-Anatoxin A fumarat is a potent nicotinic agonist with Ki values of 1.25 and 1840 nM for α4β2 and α7 nicotinic receptors respectively.
CSN25275 (S)-PNU-282987 HCl 128311-08-0 (S)-PNU-282987 is the an absolute stereochemistry form of PNU-282987.
CSN25570 (-)-(S)-B-973B 2244989-34-0 (-)-(S)-B-973B is positive allosteric modulator of α7 nAChRs with EC50 of ~0.3 μM.
CSN25357 Ethyl (triphenylphosphoranylidene) acetate 1099-45-2
CSN25425 LY 2033298 New 886047-13-8
CSN25424 Cyclopentolate HCl 5870-29-1
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