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Cat. No. Product Name CAS No. Information
CSN10004 Cladribine  4291-63-8 Cladribine is an adenosine deaminase inhibitor used to treat hairy cell leukemia and multiple sclerosis. For U266, RPMI8226, and MM1.S cells, its IC50
CSN10240 Aliskiren  173334-57-1 Aliskiren is a renin inhibitor with IC50 of 1.5 nM.
CSN10349 Atazanavir  198904-31-3 Atazanavir is a protease inhibitor used as an antiretroviral medication to treat and prevent HIVAIDS.
CSN10369 Azilsartan  147403-03-0 Azilsartan is an orally available angiotensin II type 1 AT1 receptor antagonist with IC50 value of 26 nM
CSN10496 Ambrisentan  177036-94-1 Ambrisentan is an oral, once-daily endothelin receptor antagonist that is selective for the endothelin type A receptor (IC50s 0.251, 0.316, 0.398, 25
CSN10538 Caffeic Acid Phenethyl Ester  104594-70-9 Caffeic acid phenethyl ester, a natural product isolated and purified from the barks of Cinnamomum cassia Presl, is a potent and specific inhibitor of
CSN10852 DMXAA  117570-53-3 DMXAA is an apoptosis inducer with anti-vascular activity. It can inhibit STING and enzyme DT-diaphorase (Ki 20 M).
CSN10931 Erlotinib  183321-74-6 Erlotinib is an EGFR inhibitor with IC50 of 2 nM, > 1000-fold more sensitive for EGFR than human c-Src or v-Abl.
CSN11084 Gefitinib  184475-35-2 Gefitinibis an EGFR inhibitor for Tyr1173, Tyr992, Tyr1173 and Tyr992 in the NR6wtEGFR and NR6W cells with IC50 of 37 nM, 37nM, 26 nM and 57 nM, respe
CSN11131 GW9662  22978-25-2 GW9662 selectively antagonizes PPAR with IC50 of 3.3 nM. It can inhibit the growth of mammary cancer cells.
CSN11187 GM6001  142880-36-2 GM6001 is a broad spectrum MMPs inhibitor for MMP-1, MMP-2, MMP-3, MMP-7, MMP-8, MMP-9, MMP-12, MMP-14, and MMP-26 with Ki of 0.4 nM, 0.5 nM, 27 nM, 3
CSN11190 Imatinib  152459-95-5 Imatinib is a multi-target inhibitor of v-Abl, c-Kit and PDGFR with IC50 of 0.6 M, 0.1 M and 0.1 M in cell-free or cell-based assays, respectively.
CSN11280 Lenalidomide  191732-72-6 Lenalidomide a analog of thalidomide is TNF- secretion inhibitor with IC50 of 13 nM
CSN11339 Lubiprostone  136790-76-6 Lubiprostone is an ClC-2 chloride channel activator used in the treatment of idiopathic chronic constipation.
CSN11455 Montelukast Sodium  151767-02-1 Montelukast Sodium is a potent, selective and competitive LTR1 antagonist with IC50 value 5 nM, possesssing anti-inflammatory and bronchodilating act
CSN11667 Pemetrexed  137281-23-3 Pemetrexed is an antifolate and antimetabolite for TSthymidylate synthase DHFRdihydrofolate reductase and GARFTglycinamide ribonucleotide formyltransf
CSN11857 Roflumilast  162401-32-3 Roflumilast is a selective and long-acting inhibitor of PDE-4 with IC50 of 0.8 nM.
CSN11862 Roscovitine  186692-46-6 Roscovitine is a potent and selective CDK inhibitor for Cdc2, CDK2 and CDK5 with IC50 of 0.65 μM, 0.7 μM and 0.16 μM and shows little effect on CDK4/6
CSN11899 SB-203580  152121-47-6 SB-203580 is a p38 MAPK inhibitor with IC50 of 0.3-0.5 M.
CSN12170 Tyrphostin AG 879  148741-30-4 Tyrphostin AG 879 potently inhibits HER2ErbB2 with IC50 of 1 M 100- and 500-fold higher selective to ErbB2 than PDGFR and EGFR
CSN12304 BSI-201  160003-66-7 BSI-201 is a PARP1 inhibitor with demonstrated effectiveness in triple-negative breast cancer (TNBC).
CSN12327 Pixantrone Dimaleate  144675-97-8 Pixantrone dimaleate is a topoisomerase II inhibitor and DNA intercalator with anti-tumor activity Pixantrone dimaleate is an experimental antineoplas
CSN12330 Piceatannol  10083-24-6 Piceatannol a natural stilbene is selective Syk inhibitor extracted from the rhizomes of Polygonum cuspidatum Sieb et Zucc
CSN12357 PD153035  153436-54-5 PD153035 is EGFR inhibitor with Ki and IC50 of 5.2 pM and 29 pM and could rapidly suppress autophosphorylation of EGFR.
CSN12358 AG-1478  153436-53-4 AG-1478 selectively inhibits EGFR with IC50 of 3 nM in cell-free assay.
CSN12447 Fondaparinux Sodium  114870-03-0 Fondaparinux sodium is a pentasaccharide inhibitor of antithrombin-dependent factor Xa (IC50 40 nM). It can bind to antithrombin III.
CSN12489 Pioglitazone HCl  112529-15-4 Pioglitazone HCl is a selective agonist of PPARγ with EC50 of 0.93 μM which is used to treat diabetes.
CSN12500 Combretastatin A4  117048-59-6 Combretastatin A4 is a tubulin polymerization inhibitor with Kd value of 04 M for binding to -tubulin
CSN12559 Tenofovir  147127-20-6 Tenofovir is an antiretroviral drug known as nucleotide analogue reverse transcriptase inhibitors (NRTIs), which block reverse transcriptase, a crucia
CSN12570 Rosiglitazone Maleate  155141-29-0 Rosiglitazone maleate is the maleate form of rosiglitazone which is a high-affinity selective agonist of the peroxisome proliferator-activated recepto
CSN12700 PD153035 HCl  183322-45-4 PD153035 HCl is an reversible inhibitor of EGFR with Ki and IC50 of 5.2 pM and 29 pM.
CSN12964 Cabazitaxel  183133-96-2 Cabazitaxel is a semi-synthetic derivative of the natural taxoid 10-deacetylbaccatin III with potential antineoplastic activity. Cabazitaxel exerts it
CSN13185 Pomalidomide  19171-19-8 Pomalidomide can inhibit LPS-induced TNF- release with IC50 of 13 nM in PBMCs.
CSN13562 Triapine  143621-35-6 Triapine is a ribonucleotide reductase inhibitor and a CDK inhibtor.
CSN16276 PF-06840003  198474-05-4 PF-06840003 is a highly selective orally bioavailable IDO-1 inhibitor with IC50 of 041 M
CSN16424 Licochalcone A  58749-22-7 Licochalcone A an estrogenic flavanoid can be an inhibitor of p-glycoprotein and has anti-inflammatory actions
CSN16694 Metformin HCl  1115-70-4 Metformin HCl, a widely used anti-diabetic drug has potential efficacy as an anti-cancer drug, decreasing hyperglycemia in hepatocytes primarily by su
CSN16698 Alendronate Sodium Trihydrate  121268-17-5 Alendronate Sodium Trihydrate is an inhibitor of farnesyl diphosphate synthase with IC50 of 460 nM. It is used to treat osteoporosis.
CSN16708 Calcifediol  19356-17-3 Calcifediol is an active metabolite of vitamin D It can inhibit the secretion of parathyroid hormone with 2 nM and commonly used as an indicator of bo
CSN16716 Everolimus  159351-69-6 Everolimus is a mTOR inhibitor of FKBP12 with IC50 of 1.6-2.4 nM.
CSN16720 Fingolimod HCl  162359-56-0 Fingolimod HCl is a S1P antagonist with IC50 of 0.033 nM.
CSN16725 Erlotinib HCl  183319-69-9 Erlotinib HCl is a directly acting inhibitor of human EGFR tyrosine kinase with an IC50 of 2 nM.
CSN19413 Polydatin  27208-80-6 Polydatin, extracted from the roots ofPolygonum cuspidatumSieb, a widely used traditional Chinese remedies, possesses anti-inflammatory activity in se
CSN19473 Bexarotene  153559-49-0 Bexarotene is a selective agonist of RXR IC50 24 nM RXR IC50 25 nM and RXR IC50 33 nM with antineoplastic activity
CSN19160 H 89 2HCl  130964-39-5 H 89 2HCl is a potent and selective inhibitor of cyclic AMP-dependent protein kinase (protein kinase A) with IC50 of 48 nM. It also shows weak inhibit
CSN16987 ABT-751  141430-65-1 ABT-751 can inhibit microtubule polymerization through binding to -tubulin on the colchine site
CSN12943 Marimastat  154039-60-8 Marimastat is a competitive and broad-spectrum MMP inhibitor with IC50 values of 3, 5, 6, 9 and 13 nM for MMP-9, MMP-1, MMP-2, MMP-14 and MMP-7, respe
CSN10894 Elacridar  143664-11-3 Elacridar is a P-glycoprotein inhibitor, and has been used both in vitro and in vivo as a tool inhibitor of P-glycoprotein (Pgp) to investigate the ro
CSN11329 Lopinavir  192725-17-0 Lopinavir is an antiretroviral of the protease inhibitor class, as well as an inhibitor of P-Glycoprotein, Cytochrome P450 3A and Organic Anion Transp
CSN13587 Ritonavir  155213-67-5 Ritonavir is both an HIV protease inhibitor and a Cytochrome P450 3A inhibitor.
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