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5-HT Receptor

5-HT Receptor

Cat. No. Product Name CAS No. Information
CSN12199 Vilazodone 163521-12-8 Vilazodone is a combined serotonin specific reuptake inhibitor (SSRI) and 5-HT1A receptor partial agonist currently under clinical evaluation for the treatment of major depression.
CSN23171 Tropanserin 85181-40-4 Tropanserin is a selective 5-HT3 receptor antagonist.
CSN12086 Tiamenidine 31428-61-2 Thioridazine is an antipsychotic drug used in the treatment of schizophrenia and psychosis shows D4 selectivity or serotonin antagonism
CSN23197 WAY 629 HCl 57756-44-2 Selective 5-HT2C agonist
CSN23140 Tandospirone HCl 99095-10-0 Selective 5-HT1A partial agonist
CSN23208 Zimelidine 2HCl 60525-15-7 Selective 5-HT uptake inhibitor
CSN23095 SB 215505 162100-15-4 SB215505 is a potent 5-HT2B/2C receptor antagonist (pKi values are 8.3, 7.66 and 6.77 for 5-HT2B, 5-HT2C and 5-HT2A respectively). It Increases wakefulness and motor activity in rats.
CSN23105 SB 699551 864741-95-7 SB 699551 is a selective 5-ht5a receptor antagonist (pKi values are 8.3, < 6.0, < 6.0, < 6.0, < 5.5 and < 5.5 for 5-ht5a, 5-HT1B/D, 5-HT2A, 5-HT2C, 5-HT1A and 5-HT7 receptors respectively).
CSN23096 SB 221284 196965-14-7 SB 221284 is potent, selective 5-HT2C/2B receptor antagonist. SB 221284 are pKi values are 6.4, 7.9 and 8.6 for 5-HT2A, 2B and 2C receptors respectively.
CSN17113 Promethazine HCl   58-33-3 Promethazine HCl is the effective antagonist of the H1 receptor and moderate antagonist of mACh receptor.
CSN23130 SR 57227 HCl 77145-61-0 Potent and selective 5-HT3 agonist
CSN27301 Phenylbiguanide 102-02-3 Phenylbiguanide is a 5-HT3 receptor selective agonist with an EC50 of 3.0±0.1 μM.
CSN18173 Pardoprunox HCl 269718-83-4 Pardoprunox HCl is a partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) and D3 receptor (pKi = 8.6) partial agonist and 5-HT1A receptor (pKi = 8.5) full agonist.
CSN27393 Paliperidone palmitate 199739-10-1 Paliperidone palmitate (9-Hydroxyrisperidone palmitate), an atypical long-acting antipsychotic agent, is an ester prodrug of Paliperidone. Paliperidone is a dopamine antagonist and 5-HT2A antagonist of the atypical antipsychotic class. Paliperidone palmitate shows efficacy against schizophrenia.
CSN27188 p-MPPI HCl 220643-77-6 p-MPPI is a novel 5-HT Receptor 1A receptor antagonist. It produced a significant and dose-related anxiolytic profile in male mice.
CSN27303 Org-12962   132834-56-1 Org-12962 is a potent, selective and orally active 5-HT2C receptor agonist with a pEC50 value of 7.01. Org-12962 also exhibits high effacy for the 5-HT2A and 5-HT2B receptor with pEC50s of 6.38 and 6.28, respectively.Org-12962 displays antiaversive effects in a rat model of panic-like anxiety.
CSN26151 LY344864 racemate 186543-64-6 LY344864 racemate is the racemate form of LY344864. LY344864 is a selective receptor agonist with an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.
CSN25658 Elopiprazole 115464-77-2 Elopiprazole is an antipsychotic drug of the phenylpiperazine class.
CSN27302 Dehydroaripiprazole   129722-25-4 Dehydroaripiprazole (OPC-14857) is an active metabolite of Aripiprazole. Aripiprazole is an antipsychotic agent and is metabolized by CYP3A4 and CYP2D6 forming mainly Dehydroaripiprazole. Dehydroaripiprazole has with antipsychotic activity equivalent to Aripiprazole.
CSN17079 Colfosceril Palmitate 63-89-8 Colfosceril palmitate is a drug used as a pulmonary surfactant. It is also a key conponent of LNP as an effective delivery vehicle of mRNA.
CSN23078 RS 67506 HCl 168986-61-6 5-HT4 partial agonist
CSN23074 RS 23597-190 HCl 149719-06-2 5-HT4 antagonist
CSN23076 RS 39604 HCl 167710-87-4 5-HT4 antagonist
CSN23090 SB 200646 HCl 143797-62-0 5-HT2C/2B antagonist
CSN23080 RU 24969 Hemisuccinate 66611-27-6 5-HT1A and 5-HT1B agonist
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