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5-HT Receptor
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN12220 | Xanthotoxol | 2009-24-7 | Xanthotoxol, a natural product isolated and purified from the fruits of Cnidium monnieri, has neuroprotection, due to the ability of xanthotoxol to attenuate the expression of pro-inflammatory mediators and thereby inhibit the inflammatory response after cerebral ischemia. |
| CSN23195 | WAY 208466 2HCl | 1207064-61-6 | WAY-208466 2HCl is a selective serotonin 5-HT6 receptor agonist. |
| CSN23171 | Tropanserin | 85181-40-4 | Tropanserin is a selective 5-HT3 receptor antagonist. |
| CSN23100 | SB 258719 HCl | 1217674-10-6 | Selective 5-HT7 antagonist |
| CSN23114 | SGS 518 Oxalate | 445441-27-0 | Selective 5-HT6 antagonist |
| CSN23197 | WAY 629 HCl | 57756-44-2 | Selective 5-HT2C agonist |
| CSN23112 | SDZ SER 082 Fumarate | 1417343-80-6 | Selective 5-HT2B/2C antagonist |
| CSN23140 | Tandospirone HCl | 99095-10-0 | Selective 5-HT1A partial agonist |
| CSN23208 | Zimelidine 2HCl | 60525-15-7 | Selective 5-HT uptake inhibitor |
| CSN23095 | SB 215505 | 162100-15-4 | SB215505 is a potent 5-HT2B/2C receptor antagonist (pKi values are 8.3, 7.66 and 6.77 for 5-HT2B, 5-HT2C and 5-HT2A respectively). It Increases wakefulness and motor activity in rats. |
| CSN23104 | SB 399885 HCl | 402713-81-9 | SB-399885 hydrochloride is a 5-HT6 receptor antagonist. |
| CSN23105 | SB 699551 | 864741-95-7 | SB 699551 is a selective 5-ht5a receptor antagonist (pKi values are 8.3, < 6.0, < 6.0, < 6.0, < 5.5 and < 5.5 for 5-ht5a, 5-HT1B/D, 5-HT2A, 5-HT2C, 5-HT1A and 5-HT7 receptors respectively). |
| CSN23098 | SB 243213 HCl | 200940-23-4 | SB 243213 hydrochloride is a selective and high-affinity 5-hydroxytryptamine (5-HT)2C receptor antagonist with a pKi of 9.37 and a pKb of 9.8 for human 5-HT2C receptor. SB 243213 hydrochloride has improved anxiolytic profile[1]. |
| CSN23096 | SB 221284 | 196965-14-7 | SB 221284 is potent, selective 5-HT2C/2B receptor antagonist. SB 221284 are pKi values are 6.4, 7.9 and 8.6 for 5-HT2A, 2B and 2C receptors respectively. |
| CSN23094 | SB 206553 HCl | 1197334-04-5 | SB 206553 HCl is a potent and selective 5-HT2B/5-HT2C receptor antagonist (rat 5-HT2B pA2 = 8.89, human 5-HT2C pKi = 7.92). It displays > 80-fold selectivity over all other 5-HT receptor subtypes and a variety of other receptors (pKi < 6). |
| CSN23093 | SB 204741 | 152239-46-8 | SB 204741 is potent and selective 5-HT2B receptor antagonist (pA2 = 7.95). It displays ≥ 135-fold selectivity over 5-HT2C (pKi = 5.82), 5-HT2A (pKi < 5.2), 5-HT1A, 1D, 1E, 5-HT3 and 5-HT4 receptors. |
| CSN23092 | SB 204070 | 148688-01-1 | SB 204070A is a highly selective 5-HT4 receptor antagonist. |
| CSN23091 | SB 203186 HCl | 207572-69-8 | SB 203186 HCl is potent 5-HT4 receptor antagonist with high affinity for human atrial 5-HT4 receptors. |
| CSN23073 | RS 102221 HCl | 187397-18-8 | RS-102221 HCl is a highly potent, selective 5-HT2C receptor antagonist. |
| CSN23066 | Ro 04-6790 | 202466-68-0 | Ro 04-6790 is a potent and selective 5-HT6 receptor antagonist (pKi values are 7.26 and 7.35 at rat and human 5-HT6 receptors respectively). Ro 04-6790 displays no affinity at a range of other receptors (IC50 > 10 μM). |
| CSN19422 | Puerarin | 3681-99-0 | Puerarin, an isoflavones, is antagonist of 5-HT2C receptor and benzodiazepine site that can reduce anxiety symptoms associated with alcohol withdrawal. Puerarin is found in the root of radix puerariae. |
| CSN23099 | SB 258585 HCl | 1216468-02-8 | Potent, selective 5-HT6 antagonist |
| CSN23130 | SR 57227 HCl | 77145-61-0 | Potent and selective 5-HT3 agonist |
| CSN23193 | WAY 161503 HCl | 276695-22-8 | Potent and selective 5-HT2C agonist |
| CSN18311 | Isocorynoxeine | 51014-29-0 | Isocorynoxeine, a major alkaloid found in Uncaria rhynchophylla, exhibits wide beneficial effects on the cardiovascular and cardiocerebral vascular systems. |
| CSN23084 | S 14506 HCl | 286369-38-8 | Highly potent 5-HT1A agonist; displays unique binding mechanism |
| CSN23194 | WAY 181187 Oxalate | 1883548-85-3 | High affinity and selective 5-HT6 agonist |
| CSN20976 | Geissoschizine methyl ether | 60314-89-8 | Geissoschizine methyl ether is a potent serotonin A receptor agonist. |
| CSN14586 | Galanolactone | 115753-79-2 | Galanolactone, a natural product isolated and purified from the rhizomes of Zingiber officinale Roscoe with cytotoxic activity, has anti-5-HT effect, a diterpenoid isolated from ginger, is related to antagonism of 5-HT3 receptors, exerts anti-obesity effect through down regulation of adipogenic transcription factors and adipogenic marker genes, and inhibits nitric oxide production with IC(50) values ranging from 5.5 to 28.5 μM. |
| CSN24769 | F-15599 | 635323-95-4 | F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist with Ki value of 3.4nM. |
| CSN21571 | Clocapramine | 47739-98-0 | Clocapramine is D2 5-HT2A receptors antagonist. |
| CSN23783 | AVN492 | 1220646-23-0 | AVN492 is a selective antagonist of 5-HT6R with Ki of 91 pM. |
| CSN21450 | Abaperidone | 183849-43-6 | Abaperidone is an antagonist of 5-HT2A receptor and dopamine D2 receptor with IC50s of 6.2 and 17 nM respectively. |
| CSN23078 | RS 67506 HCl | 168986-61-6 | 5-HT4 partial agonist |
| CSN23074 | RS 23597-190 HCl | 149719-06-2 | 5-HT4 antagonist |
| CSN23076 | RS 39604 HCl | 167710-87-4 | 5-HT4 antagonist |
| CSN23077 | RS 56812 HCl | 143339-12-2 | 5-HT3 partial agonist |
| CSN23090 | SB 200646 HCl | 143797-62-0 | 5-HT2C/2B antagonist |
| CSN23085 | S 32212 HCl | 847871-78-7 | 5-HT2C inverse agonist; α2-adrenoceptor antagonist |
| CSN23080 | RU 24969 Hemisuccinate | 66611-27-6 | 5-HT1A and 5-HT1B agonist |
| CSN21566 | (Z)-Thiothixene | 3313-26-6 | (Z)-Thiothixene is serotonergic receptor antagonist. |
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