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5-HT Receptor

5-HT Receptor

Cat. No. Product Name CAS No. Information
CSN12245 Zolmitriptan   139264-17-8 Zolmitriptan is an agonist of 5-HT1B5-HT1D receptors with anti-migraine properties
CSN12542 Ziprasidone 146939-27-7 Ziprasidone is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity.
CSN12748 Ziprasidone HCl 122883-93-6 Ziprasidone hydrochloride is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity, and is used in the treatment of schizophrenia and bipolar disorder.
CSN13510 VUF 10166 155584-74-0 VUF10166 is a potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.
CSN13804 Vilazodone HCl   163521-08-2 Vilazodone HCl is both a selective 5-HT reuptake inhibitor and a partial 5-HT1A receptor agonist.
CSN12174 Urapidil 34661-75-1 Urapidil is a sympatholytic antihypertensive drug
CSN16687 Tropisetron HCl 105826-92-4 Tropisetron HCl is a selective and competitive 5-HT3 receptor antagonist.
CSN12597 Trazodone HCl   25332-39-2 Trazodone HCl is a selective serotonin reuptake inhibitor and 5HT2 receptor antagonist, used as an antidepressant medication.
CSN16779 Tianeptine   72797-41-2 Tianeptine is a unique tricyclic antidepressant, in contrast to SSRIs, which can increase serotonin uptake in the brain and reduce stress-induced atrophy of neuronal dendrites.
CSN16726 Tegaserod Maleate   189188-57-6 Tegaserod Maleate is a potent full agonist at 5-HT4 receptors with an EC50 value of 7 nM, used to treat irritable bowel syndrome associated with constipation and chronic constipation.
CSN12475 Sumatriptan Succinate   103628-48-4 Sumatriptan Succinate can selectively bind to and activate 5-HT1 receptors
CSN11037 Sevoflurane 28523-86-6 Sevoflurane is a sweet-smelling, nonflammable, highly fluorinated methyl isopropyl ether used as an inhalational anaesthetic for induction and maintenance of general anesthesia.
CSN11920 Setiptiline 57262-94-9 Setiptiline is a serotonin receptor antagonist.
CSN16751 SB-742457   607742-69-8 SB-742457 is a selective 5-HT6 receptor antagonist with Ki value of 1.4 nM, showing potential cognition, memory, and learning-enhancing effects.
CSN11875 Rupatadine 158876-82-5 Rupatadine is a potent dual PAFH1 antagonist with Ki of 0.550.1 M (rabbit platelet membranesguinea pig cerebellum membranes).
CSN18707 Rizatriptan Benzoate   145202-66-0 Rizatriptan Benzoate is a triptan-class 5-HT1 receptor agonist, used to treat migraine headaches.
CSN12479 Risperidone   106266-06-2 Risperidone is a multiple-target antipsychotic with high affinity for 5-HT2A and D2 receptors alpha 1 alpha 2 and H1 receptors
CSN22178 PRX933 HCl 639029-42-8 PRX933 HCl is a 5-HT2c receptor agonist.
CSN10104 Pizotifen Malate   5189-11-7 Pizotifen Malate is a benzocycloheptene-based drug used to reduce the frequency of recurrent migraine headacheswith with high affinity for 5-HT and dopamine receptors Kis 794 and 24 nM for 5-HT2C and D2 respectively
CSN18174 Pardoprunox 269718-84-5 Pardoprunox is a partial dopamine D2 (pKi 8.1) and D3 (pKi 8.6) receptor agonist (IA 50 and 67, respectively) and full serotonin 5-HT1A (pKi 8.5) receptor agonist (IA 100), and also binds to D4 (pKi 7.8), 1-adrenergic (pKi 7.8), 2-adrenergic (pKi 7.4), and 5-HT7 receptors (pKi 7.2) with lower affinity.
CSN13827 Palonosetron HCl   135729-62-3 Palonosetron HCl is a carbazole-derived and selective 5-HT3 receptor antagonist.
CSN13137 Ondansetron 99614-02-5 Ondansetron is a serotonin 5-HT3 receptor antagonist used mainly as anantiemetic (to treat nausea and vomiting), often following chemotherapy.
CSN16686 Ondansetron HCl 99614-01-4 Ondansetron is a serotonin 5-HT3 receptor antagonist used mainly as anantiemetic (to treat nausea and vomiting), often following chemotherapy.
CSN15871 Ondansetron HCl 2H2O   103639-04-9 Ondansetron HCl 2H2O is a competitive 5-HT3 receptor antagonist.
CSN11590 Nuciferine 475-83-2 Nuciferine is naturally occuring alkaloid found in the plants Nymphaea caerulea and Nelumbo nucifera as a potent inverse agonist at human 5-HT7 receptor.
CSN20313 NLX-112 208110-64-9 NLX-112 is a potent and efficacious serotonin 5-HT1A receptor agonist potentially for the treatment of drug-induced dyskinesia in patients.
CSN13092 Nefazodone HCl   82752-99-6 Nefazodone HCl is a 5-HT2A receptor antagonist with Ki of 5.8 nM and an inhibitor of serotonin and noradrenalin uptake with IC50s of 290 and 300 nM respectively, it is an antidepressant drug.
CSN12511 Naratriptan 121679-13-8 Naratriptan is a selective 5-HT1 receptor subtype agonist and is a triptan drug that is used for the treatment of migraine headaches
CSN10097 Naftidrofuryl Oxalate 3200-06-4 Naftidrofuryl oxalate is a drug used in the management of peripheral and cerebral vascular disorders as a vasodilator enhance cellular oxidative capacity and may also be a 5-HT2 receptor antagonist
CSN11473 Mosapride Citrate   112885-42-4 Mosapride Citrate is both a selective 5HT4 agonist and a 5HT3 antagonist, use as a gastroprokinetic agent.
CSN12491 Mosapride   112885-41-3 Mosapride a selective 5HT4 agonist used as a gastroprokinetic agent.
CSN11451 Mirtazapine 85650-52-8 Mirtazapine is a potent tetracyclic antidepressant.
CSN21278 Methiothepin Mesylate 74611-28-2 Methiothepin mesylate is a potent and non-selective 5-HT2 receptor antagonist, with pKds of 7.10 (5-HT1A), 7.28 (5HT1B), 7.56 (5HT1C), 6.99 (5HT1D), 7.0 (5-HT5A), 7.8 (5-HT5B), 8.74 (5-HT6), and 8.99 (5-HT7), and pKis of 8.50 (5HT2A), 8.68 (5HT2B), and 8.35 (5HT2C).
CSN17035 Lumateperone Tosylate 1187020-80-9 Lumateperone tosylate is a 5-HT2A receptor antagonist (Ki 0.54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki 32 nM), and a SERT blocker (Ki 61 nM).
CSN11336 Loxapine succinate salt   27833-64-3 Loxapine succinate salt is an multiple-target antagonist of both D2D4 dopamine receptor and 5-HT2A2B 5-H7 serotonin receptor used as an antipsychotic agent
CSN18968 Latrepirdine 2HCl 97657-92-6 Latrepirdine is an orally active,and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihistamine drug.
CSN13508 Lasmiditan 439239-90-4 Lasmiditan is a high-affinity, highly selective 5-HT1F receptor agonist (Ki2.1 nM), compared with Ki of 1043 nM and 1357 nM at the 5-HT(1B) and 5-HT(1D) receptors, respectively.
CSN11251 Ketanserin Tartrate   83846-83-7 Ketanserin Tartrate is a water soluble selective 5-HT2A and 5-HT1D antagonist
CSN11195 Imipramine HCl 113-52-0 Imipramine HCl is a tricyclic inhibitor of both serotonin and norepinephrine transporters with Ki values of 77 nM and 67 nM respectively
CSN11019 Flibanserin   167933-07-5 Flibanserin is a serotonergic antidepressant used to treat hypoactive sexual desire disorder. It is also a P-Glycoprotein Inhibitor.
CSN10727 Cyproheptadine Hydrochloride Sesquihydrate   41354-29-4 Cyproheptadine Hydrochloride Sesquihydrate is a serotonin antagonist and a histamine H1 blocker used as antipruritic, appetite stimulant, antiallergic, and for the post-gastrectomy dumping syndrome, etc.
CSN10658 Citalopram Hydrobromide   59729-32-7 Citalopram Hydrobromide is a highly selective and potent 5-HT uptake inhibitor with no effect on noradrenalin or dopamine uptake.
CSN21349 Cisapride 260779-88-2 Cisapride is a 5-HT4 serotonin receptor agonist.
CSN10655 Cisapride 81098-60-4 Cisapride is a 5-HT4 agonist which can stimulate intestinal ACh release.
CSN10511 Buspirone HCl 33386-08-2 Buspirone hydrochloride is an anxiolytic psychotropic drug is used to treat generalized anxiety disorder GAD
CSN20672 Aripiprazole Lauroxil 1259305-29-7 Aripiprazole lauroxil is a long-acting injectable atypical antipsychotic. It is an N-acyloxymethyl prodrug of aripiprazole that is administered via intramuscular injection once every four to six weeks for the treatment of schizophrenia.
CSN12463 Aripiprazole   129722-12-9 Aripiprazole is a multiple-target agent used to treat schizophrenia and bipolar disorder working as both a silent antagonist and a high-efficacy partial agonist of D2 receptor as well as works as a partial agonist of 5-HT1A5-HT2A 5-HT2 receptora potent inverse agonist of 5-HT2B receptor a functional antagonist of 5-HT7 receptor
CSN18262 Amitifadine HCl 410074-74-7 Amitifadine hydrochloride is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).
CSN10249 Almotriptan Malate   181183-52-8 Almotriptan Malate a serotonin 5HT-1B1D-receptor agonist with high affinity for the 5-HT(1B) and 5-HT(1D) receptors, used to treat migraine.
CSN10250 Almotriptan 154323-57-6 Almotriptan is a 5-HT1B1D-receptor agonist used to treat migraine
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