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5-HT Receptor
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN12245 | Zolmitriptan | 139264-17-8 | Zolmitriptan is an agonist of 5-HT1B5-HT1D receptors with anti-migraine properties |
| CSN12542 | Ziprasidone | 146939-27-7 | Ziprasidone is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. |
| CSN12748 | Ziprasidone HCl | 122883-93-6 | Ziprasidone hydrochloride is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity, and is used in the treatment of schizophrenia and bipolar disorder. |
| CSN13510 | VUF 10166 | 155584-74-0 | VUF10166 is a potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower. |
| CSN13804 | Vilazodone HCl | 163521-08-2 | Vilazodone HCl is both a selective 5-HT reuptake inhibitor and a partial 5-HT1A receptor agonist. |
| CSN12174 | Urapidil | 34661-75-1 | Urapidil is a sympatholytic antihypertensive drug |
| CSN16687 | Tropisetron HCl | 105826-92-4 | Tropisetron HCl is a selective and competitive 5-HT3 receptor antagonist. |
| CSN12597 | Trazodone HCl | 25332-39-2 | Trazodone HCl is a selective serotonin reuptake inhibitor and 5HT2 receptor antagonist, used as an antidepressant medication. |
| CSN16779 | Tianeptine | 72797-41-2 | Tianeptine is a unique tricyclic antidepressant, in contrast to SSRIs, which can increase serotonin uptake in the brain and reduce stress-induced atrophy of neuronal dendrites. |
| CSN16726 | Tegaserod Maleate | 189188-57-6 | Tegaserod Maleate is a potent full agonist at 5-HT4 receptors with an EC50 value of 7 nM, used to treat irritable bowel syndrome associated with constipation and chronic constipation. |
| CSN12475 | Sumatriptan Succinate | 103628-48-4 | Sumatriptan Succinate can selectively bind to and activate 5-HT1 receptors |
| CSN11037 | Sevoflurane | 28523-86-6 | Sevoflurane is a sweet-smelling, nonflammable, highly fluorinated methyl isopropyl ether used as an inhalational anaesthetic for induction and maintenance of general anesthesia. |
| CSN11920 | Setiptiline | 57262-94-9 | Setiptiline is a serotonin receptor antagonist. |
| CSN16751 | SB-742457 | 607742-69-8 | SB-742457 is a selective 5-HT6 receptor antagonist with Ki value of 1.4 nM, showing potential cognition, memory, and learning-enhancing effects. |
| CSN11875 | Rupatadine | 158876-82-5 | Rupatadine is a potent dual PAFH1 antagonist with Ki of 0.550.1 M (rabbit platelet membranesguinea pig cerebellum membranes). |
| CSN18707 | Rizatriptan Benzoate | 145202-66-0 | Rizatriptan Benzoate is a triptan-class 5-HT1 receptor agonist, used to treat migraine headaches. |
| CSN12479 | Risperidone | 106266-06-2 | Risperidone is a multiple-target antipsychotic with high affinity for 5-HT2A and D2 receptors alpha 1 alpha 2 and H1 receptors |
| CSN22178 | PRX933 HCl | 639029-42-8 | PRX933 HCl is a 5-HT2c receptor agonist. |
| CSN10104 | Pizotifen Malate | 5189-11-7 | Pizotifen Malate is a benzocycloheptene-based drug used to reduce the frequency of recurrent migraine headacheswith with high affinity for 5-HT and dopamine receptors Kis 794 and 24 nM for 5-HT2C and D2 respectively |
| CSN18174 | Pardoprunox | 269718-84-5 | Pardoprunox is a partial dopamine D2 (pKi 8.1) and D3 (pKi 8.6) receptor agonist (IA 50 and 67, respectively) and full serotonin 5-HT1A (pKi 8.5) receptor agonist (IA 100), and also binds to D4 (pKi 7.8), 1-adrenergic (pKi 7.8), 2-adrenergic (pKi 7.4), and 5-HT7 receptors (pKi 7.2) with lower affinity. |
| CSN13827 | Palonosetron HCl | 135729-62-3 | Palonosetron HCl is a carbazole-derived and selective 5-HT3 receptor antagonist. |
| CSN13137 | Ondansetron | 99614-02-5 | Ondansetron is a serotonin 5-HT3 receptor antagonist used mainly as anantiemetic (to treat nausea and vomiting), often following chemotherapy. |
| CSN16686 | Ondansetron HCl | 99614-01-4 | Ondansetron is a serotonin 5-HT3 receptor antagonist used mainly as anantiemetic (to treat nausea and vomiting), often following chemotherapy. |
| CSN15871 | Ondansetron HCl 2H2O | 103639-04-9 | Ondansetron HCl 2H2O is a competitive 5-HT3 receptor antagonist. |
| CSN11590 | Nuciferine | 475-83-2 | Nuciferine is naturally occuring alkaloid found in the plants Nymphaea caerulea and Nelumbo nucifera as a potent inverse agonist at human 5-HT7 receptor. |
| CSN20313 | NLX-112 | 208110-64-9 | NLX-112 is a potent and efficacious serotonin 5-HT1A receptor agonist potentially for the treatment of drug-induced dyskinesia in patients. |
| CSN13092 | Nefazodone HCl | 82752-99-6 | Nefazodone HCl is a 5-HT2A receptor antagonist with Ki of 5.8 nM and an inhibitor of serotonin and noradrenalin uptake with IC50s of 290 and 300 nM respectively, it is an antidepressant drug. |
| CSN12511 | Naratriptan | 121679-13-8 | Naratriptan is a selective 5-HT1 receptor subtype agonist and is a triptan drug that is used for the treatment of migraine headaches |
| CSN10097 | Naftidrofuryl Oxalate | 3200-06-4 | Naftidrofuryl oxalate is a drug used in the management of peripheral and cerebral vascular disorders as a vasodilator enhance cellular oxidative capacity and may also be a 5-HT2 receptor antagonist |
| CSN11473 | Mosapride Citrate | 112885-42-4 | Mosapride Citrate is both a selective 5HT4 agonist and a 5HT3 antagonist, use as a gastroprokinetic agent. |
| CSN12491 | Mosapride | 112885-41-3 | Mosapride a selective 5HT4 agonist used as a gastroprokinetic agent. |
| CSN11451 | Mirtazapine | 85650-52-8 | Mirtazapine is a potent tetracyclic antidepressant. |
| CSN21278 | Methiothepin Mesylate | 74611-28-2 | Methiothepin mesylate is a potent and non-selective 5-HT2 receptor antagonist, with pKds of 7.10 (5-HT1A), 7.28 (5HT1B), 7.56 (5HT1C), 6.99 (5HT1D), 7.0 (5-HT5A), 7.8 (5-HT5B), 8.74 (5-HT6), and 8.99 (5-HT7), and pKis of 8.50 (5HT2A), 8.68 (5HT2B), and 8.35 (5HT2C). |
| CSN17035 | Lumateperone Tosylate | 1187020-80-9 | Lumateperone tosylate is a 5-HT2A receptor antagonist (Ki 0.54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki 32 nM), and a SERT blocker (Ki 61 nM). |
| CSN11336 | Loxapine succinate salt | 27833-64-3 | Loxapine succinate salt is an multiple-target antagonist of both D2D4 dopamine receptor and 5-HT2A2B 5-H7 serotonin receptor used as an antipsychotic agent |
| CSN18968 | Latrepirdine 2HCl | 97657-92-6 | Latrepirdine is an orally active,and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihistamine drug. |
| CSN13508 | Lasmiditan | 439239-90-4 | Lasmiditan is a high-affinity, highly selective 5-HT1F receptor agonist (Ki2.1 nM), compared with Ki of 1043 nM and 1357 nM at the 5-HT(1B) and 5-HT(1D) receptors, respectively. |
| CSN11251 | Ketanserin Tartrate | 83846-83-7 | Ketanserin Tartrate is a water soluble selective 5-HT2A and 5-HT1D antagonist |
| CSN11195 | Imipramine HCl | 113-52-0 | Imipramine HCl is a tricyclic inhibitor of both serotonin and norepinephrine transporters with Ki values of 77 nM and 67 nM respectively |
| CSN11019 | Flibanserin | 167933-07-5 | Flibanserin is a serotonergic antidepressant used to treat hypoactive sexual desire disorder. It is also a P-Glycoprotein Inhibitor. |
| CSN10727 | Cyproheptadine Hydrochloride Sesquihydrate | 41354-29-4 | Cyproheptadine Hydrochloride Sesquihydrate is a serotonin antagonist and a histamine H1 blocker used as antipruritic, appetite stimulant, antiallergic, and for the post-gastrectomy dumping syndrome, etc. |
| CSN10658 | Citalopram Hydrobromide | 59729-32-7 | Citalopram Hydrobromide is a highly selective and potent 5-HT uptake inhibitor with no effect on noradrenalin or dopamine uptake. |
| CSN21349 | Cisapride | 260779-88-2 | Cisapride is a 5-HT4 serotonin receptor agonist. |
| CSN10655 | Cisapride | 81098-60-4 | Cisapride is a 5-HT4 agonist which can stimulate intestinal ACh release. |
| CSN10511 | Buspirone HCl | 33386-08-2 | Buspirone hydrochloride is an anxiolytic psychotropic drug is used to treat generalized anxiety disorder GAD |
| CSN20672 | Aripiprazole Lauroxil | 1259305-29-7 | Aripiprazole lauroxil is a long-acting injectable atypical antipsychotic. It is an N-acyloxymethyl prodrug of aripiprazole that is administered via intramuscular injection once every four to six weeks for the treatment of schizophrenia. |
| CSN12463 | Aripiprazole | 129722-12-9 | Aripiprazole is a multiple-target agent used to treat schizophrenia and bipolar disorder working as both a silent antagonist and a high-efficacy partial agonist of D2 receptor as well as works as a partial agonist of 5-HT1A5-HT2A 5-HT2 receptora potent inverse agonist of 5-HT2B receptor a functional antagonist of 5-HT7 receptor |
| CSN18262 | Amitifadine HCl | 410074-74-7 | Amitifadine hydrochloride is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI). |
| CSN10249 | Almotriptan Malate | 181183-52-8 | Almotriptan Malate a serotonin 5HT-1B1D-receptor agonist with high affinity for the 5-HT(1B) and 5-HT(1D) receptors, used to treat migraine. |
| CSN10250 | Almotriptan | 154323-57-6 | Almotriptan is a 5-HT1B1D-receptor agonist used to treat migraine |
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