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5-HT Receptor

5-HT Receptor

Cat. No. Product Name CAS No. Information
CSN12542 Ziprasidone 146939-27-7 Ziprasidone is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity.
CSN12748 Ziprasidone HCl 122883-93-6 Ziprasidone HCl is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity, and is used in the treatment of schizophrenia and bipolar disorder.
CSN12220 Xanthotoxol 2009-24-7 Xanthotoxol, a natural product isolated and purified from the fruits of Cnidium monnieri, has neuroprotection, due to the ability of xanthotoxol to attenuate the expression of pro-inflammatory mediators and thereby inhibit the inflammatory response after cerebral ischemia.
CSN13804 Vilazodone HCl   163521-08-2 Vilazodone HCl is both a selective 5-HT reuptake inhibitor and a partial 5-HT1A receptor agonist.
CSN16687 Tropisetron HCl 105826-92-4 Tropisetron HCl is a selective and competitive 5-HT3 receptor antagonist.
CSN12597 Trazodone HCl   25332-39-2 Trazodone HCl is a selective serotonin reuptake inhibitor and 5HT2 receptor antagonist, used as an antidepressant medication.
CSN16779 Tianeptine   72797-41-2 Tianeptine is a unique tricyclic antidepressant, in contrast to SSRIs, which can increase serotonin uptake in the brain and reduce stress-induced atrophy of neuronal dendrites.
CSN22076 Temanogrel 887936-68-7 Temanogrel is a highly selective 5-HT2A receptor antagonist with Ki of 4.9 nM.
CSN16726 Tegaserod Maleate   189188-57-6 Tegaserod Maleate is a potent full agonist at 5-HT4 receptors with an EC50 value of 7 nM, used to treat irritable bowel syndrome associated with constipation and chronic constipation.
CSN11920 Setiptiline 57262-94-9 Setiptiline is a serotonin receptor antagonist.
CSN16751 SB-742457   607742-69-8 SB-742457 is a selective 5-HT6 receptor antagonist with Ki value of 1.4 nM, showing potential cognition, memory, and learning-enhancing effects.
CSN21989 SB-224289 HCl 180084-26-8 SB-224289 hydrochloride is a selective 5-HT1B receptor antagonist, with anxiolytic effect.
CSN18707 Rizatriptan Benzoate   145202-66-0 Rizatriptan Benzoate is a triptan-class 5-HT1 receptor agonist, used to treat migraine headaches.
CSN19422 Puerarin   3681-99-0 Puerarin, an isoflavones, is antagonist of 5-HT2C receptor and benzodiazepine site that can reduce anxiety symptoms associated with alcohol withdrawal. Puerarin is found in the root of radix puerariae.
CSN22178 PRX933 HCl 639029-42-8 PRX933 HCl is a 5-HT2c receptor agonist.
CSN18174 Pardoprunox 269718-84-5 Pardoprunox is a partial dopamine D2 (pKi 8.1) and D3 (pKi 8.6) receptor agonist (IA 50 and 67, respectively) and full serotonin 5-HT1A (pKi 8.5) receptor agonist (IA 100), and also binds to D4 (pKi 7.8), 1-adrenergic (pKi 7.8), 2-adrenergic (pKi 7.4), and 5-HT7 receptors (pKi 7.2) with lower affinity.
CSN21782 Pancopride 121650-80-4 Pancopride is a selective antagonist of 5-HT3 receptor.
CSN13827 Palonosetron HCl   135729-62-3 Palonosetron HCl is a carbazole-derived and selective 5-HT3 receptor antagonist.
CSN11590 Nuciferine 475-83-2 Nuciferine is naturally occuring alkaloid found in the plants Nymphaea caerulea and Nelumbo nucifera as a potent inverse agonist at human 5-HT7 receptor.
CSN20313 NLX-112 208110-64-9 NLX-112 is a potent and efficacious serotonin 5-HT1A receptor agonist potentially for the treatment of drug-induced dyskinesia in patients.
CSN13092 Nefazodone HCl   82752-99-6 Nefazodone HCl is a 5-HT2A receptor antagonist with Ki of 5.8 nM and an inhibitor of serotonin and noradrenalin uptake with IC50s of 290 and 300 nM respectively, it is an antidepressant drug.
CSN11473 Mosapride Citrate   112885-42-4 Mosapride Citrate is both a selective 5HT4 agonist and a 5HT3 antagonist, use as a gastroprokinetic agent.
CSN12491 Mosapride   112885-41-3 Mosapride a selective 5HT4 agonist used as a gastroprokinetic agent.
CSN21278 Methiothepin Mesylate 74611-28-2 Methiothepin mesylate is a potent and non-selective 5-HT2 receptor antagonist, with pKds of 7.10 (5-HT1A), 7.28 (5HT1B), 7.56 (5HT1C), 6.99 (5HT1D), 7.0 (5-HT5A), 7.8 (5-HT5B), 8.74 (5-HT6), and 8.99 (5-HT7), and pKis of 8.50 (5HT2A), 8.68 (5HT2B), and 8.35 (5HT2C).
CSN17035 Lumateperone Tosylate 1187020-80-9 Lumateperone tosylate is a 5-HT2A receptor antagonist (Ki 0.54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki 32 nM), and a SERT blocker (Ki 61 nM).
CSN21712 Lintopride 107429-63-0 Lintopride is an antagonist of 5HT4 receptor and moderate antagonist of 5HT3.
CSN21711 Lidanserin 73725-85-6 Lidanserin is antagonist of 5-HT2A and α1-adrenergic receptor.
CSN18311 Isocorynoxeine 51014-29-0 Isocorynoxeine, a major alkaloid found in Uncaria rhynchophylla, exhibits wide beneficial effects on the cardiovascular and cardiocerebral vascular systems.
CSN21695 Irindalone 96478-43-2 Irindalone is an antagonist of serotonin 5-HT2 receptor.
CSN23591 Indole-3-carboxylic acid   771-50-6 Indole-3-carboxylic Acid is a normal urinary indolic tryptophan metabolite with multiple biological roles such as serotonin 5-HT46 receptor antagonist, EphB3 receptor tyrosine kinase inhibitor, vinyl ester pseudotripeptide proteasome inhibitor and potential therapeutic agent for Alzheimers Disease.
CSN11609 Harmine   442-51-3 Harmine is a naturally occuring fluorescent harmala alkaloid isolated plants like Middle Eastern plant harmal which can reversibly inhibit MAOA
CSN20976 Geissoschizine methyl ether 60314-89-8 Geissoschizine methyl ether is a potent serotonin A receptor agonist.
CSN21600 Deramciclane 120444-71-5 Deramciclane is an antagonist of 5-HT2A and inverse agonist of 5-HT2C receptor. It also functions as a GABA reuptake inhibitor.
CSN21594 Dazopride 70181-03-2 Dazopride is an antiemetic agent which acts as a 5-HT3 receptor antagonist and 5-HT4 receptor agonist.
CSN10727 Cyproheptadine Hydrochloride Sesquihydrate   41354-29-4 Cyproheptadine Hydrochloride Sesquihydrate is a serotonin antagonist and a histamine H1 blocker used as antipruritic, appetite stimulant, antiallergic, and for the post-gastrectomy dumping syndrome, etc.
CSN21571 Clocapramine 47739-98-0 Clocapramine is D2 5-HT2A receptors antagonist.
CSN10658 Citalopram Hydrobromide   59729-32-7 Citalopram Hydrobromide is a highly selective and potent 5-HT uptake inhibitor with no effect on noradrenalin or dopamine uptake.
CSN24509 BRL 15572 HCl 1173022-77-9 BRL 15572 HCl is a selective 5-HT Receptor 1D antagonist with a pKi value of 7.9
CSN20672 Aripiprazole Lauroxil 1259305-29-7 Aripiprazole lauroxil is a long-acting injectable atypical antipsychotic. It is an N-acyloxymethyl prodrug of aripiprazole that is administered via intramuscular injection once every four to six weeks for the treatment of schizophrenia.
CSN21450 Abaperidone 183849-43-6 Abaperidone is an antagonist of 5-HT2A receptor and dopamine D2 receptor with IC50s of 6.2 and 17 nM respectively.
CSN21566 (Z)-Thiothixene 3313-26-6 (Z)-Thiothixene is serotonergic receptor antagonist.
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