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5-HT Receptor
| Cat. No. | Product Name | CAS No. | Information |
|---|---|---|---|
| CSN12542 | Ziprasidone | 146939-27-7 | Ziprasidone is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. |
| CSN12748 | Ziprasidone HCl | 122883-93-6 | Ziprasidone HCl is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity, and is used in the treatment of schizophrenia and bipolar disorder. |
| CSN12220 | Xanthotoxol | 2009-24-7 | Xanthotoxol, a natural product isolated and purified from the fruits of Cnidium monnieri, has neuroprotection, due to the ability of xanthotoxol to attenuate the expression of pro-inflammatory mediators and thereby inhibit the inflammatory response after cerebral ischemia. |
| CSN13804 | Vilazodone HCl | 163521-08-2 | Vilazodone HCl is both a selective 5-HT reuptake inhibitor and a partial 5-HT1A receptor agonist. |
| CSN16687 | Tropisetron HCl | 105826-92-4 | Tropisetron HCl is a selective and competitive 5-HT3 receptor antagonist. |
| CSN12597 | Trazodone HCl | 25332-39-2 | Trazodone HCl is a selective serotonin reuptake inhibitor and 5HT2 receptor antagonist, used as an antidepressant medication. |
| CSN16779 | Tianeptine | 72797-41-2 | Tianeptine is a unique tricyclic antidepressant, in contrast to SSRIs, which can increase serotonin uptake in the brain and reduce stress-induced atrophy of neuronal dendrites. |
| CSN22076 | Temanogrel | 887936-68-7 | Temanogrel is a highly selective 5-HT2A receptor antagonist with Ki of 4.9 nM. |
| CSN16726 | Tegaserod Maleate | 189188-57-6 | Tegaserod Maleate is a potent full agonist at 5-HT4 receptors with an EC50 value of 7 nM, used to treat irritable bowel syndrome associated with constipation and chronic constipation. |
| CSN11920 | Setiptiline | 57262-94-9 | Setiptiline is a serotonin receptor antagonist. |
| CSN16751 | SB-742457 | 607742-69-8 | SB-742457 is a selective 5-HT6 receptor antagonist with Ki value of 1.4 nM, showing potential cognition, memory, and learning-enhancing effects. |
| CSN21989 | SB-224289 HCl | 180084-26-8 | SB-224289 hydrochloride is a selective 5-HT1B receptor antagonist, with anxiolytic effect. |
| CSN18707 | Rizatriptan Benzoate | 145202-66-0 | Rizatriptan Benzoate is a triptan-class 5-HT1 receptor agonist, used to treat migraine headaches. |
| CSN19422 | Puerarin | 3681-99-0 | Puerarin, an isoflavones, is antagonist of 5-HT2C receptor and benzodiazepine site that can reduce anxiety symptoms associated with alcohol withdrawal. Puerarin is found in the root of radix puerariae. |
| CSN22178 | PRX933 HCl | 639029-42-8 | PRX933 HCl is a 5-HT2c receptor agonist. |
| CSN18174 | Pardoprunox | 269718-84-5 | Pardoprunox is a partial dopamine D2 (pKi 8.1) and D3 (pKi 8.6) receptor agonist (IA 50 and 67, respectively) and full serotonin 5-HT1A (pKi 8.5) receptor agonist (IA 100), and also binds to D4 (pKi 7.8), 1-adrenergic (pKi 7.8), 2-adrenergic (pKi 7.4), and 5-HT7 receptors (pKi 7.2) with lower affinity. |
| CSN21782 | Pancopride | 121650-80-4 | Pancopride is a selective antagonist of 5-HT3 receptor. |
| CSN13827 | Palonosetron HCl | 135729-62-3 | Palonosetron HCl is a carbazole-derived and selective 5-HT3 receptor antagonist. |
| CSN11590 | Nuciferine | 475-83-2 | Nuciferine is naturally occuring alkaloid found in the plants Nymphaea caerulea and Nelumbo nucifera as a potent inverse agonist at human 5-HT7 receptor. |
| CSN20313 | NLX-112 | 208110-64-9 | NLX-112 is a potent and efficacious serotonin 5-HT1A receptor agonist potentially for the treatment of drug-induced dyskinesia in patients. |
| CSN13092 | Nefazodone HCl | 82752-99-6 | Nefazodone HCl is a 5-HT2A receptor antagonist with Ki of 5.8 nM and an inhibitor of serotonin and noradrenalin uptake with IC50s of 290 and 300 nM respectively, it is an antidepressant drug. |
| CSN11473 | Mosapride Citrate | 112885-42-4 | Mosapride Citrate is both a selective 5HT4 agonist and a 5HT3 antagonist, use as a gastroprokinetic agent. |
| CSN12491 | Mosapride | 112885-41-3 | Mosapride a selective 5HT4 agonist used as a gastroprokinetic agent. |
| CSN21278 | Methiothepin Mesylate | 74611-28-2 | Methiothepin mesylate is a potent and non-selective 5-HT2 receptor antagonist, with pKds of 7.10 (5-HT1A), 7.28 (5HT1B), 7.56 (5HT1C), 6.99 (5HT1D), 7.0 (5-HT5A), 7.8 (5-HT5B), 8.74 (5-HT6), and 8.99 (5-HT7), and pKis of 8.50 (5HT2A), 8.68 (5HT2B), and 8.35 (5HT2C). |
| CSN17035 | Lumateperone Tosylate | 1187020-80-9 | Lumateperone tosylate is a 5-HT2A receptor antagonist (Ki 0.54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki 32 nM), and a SERT blocker (Ki 61 nM). |
| CSN21712 | Lintopride | 107429-63-0 | Lintopride is an antagonist of 5HT4 receptor and moderate antagonist of 5HT3. |
| CSN21711 | Lidanserin | 73725-85-6 | Lidanserin is antagonist of 5-HT2A and α1-adrenergic receptor. |
| CSN18311 | Isocorynoxeine | 51014-29-0 | Isocorynoxeine, a major alkaloid found in Uncaria rhynchophylla, exhibits wide beneficial effects on the cardiovascular and cardiocerebral vascular systems. |
| CSN21695 | Irindalone | 96478-43-2 | Irindalone is an antagonist of serotonin 5-HT2 receptor. |
| CSN23591 | Indole-3-carboxylic acid | 771-50-6 | Indole-3-carboxylic Acid is a normal urinary indolic tryptophan metabolite with multiple biological roles such as serotonin 5-HT46 receptor antagonist, EphB3 receptor tyrosine kinase inhibitor, vinyl ester pseudotripeptide proteasome inhibitor and potential therapeutic agent for Alzheimers Disease. |
| CSN11609 | Harmine | 442-51-3 | Harmine is a naturally occuring fluorescent harmala alkaloid isolated plants like Middle Eastern plant harmal which can reversibly inhibit MAOA |
| CSN20976 | Geissoschizine methyl ether | 60314-89-8 | Geissoschizine methyl ether is a potent serotonin A receptor agonist. |
| CSN21600 | Deramciclane | 120444-71-5 | Deramciclane is an antagonist of 5-HT2A and inverse agonist of 5-HT2C receptor. It also functions as a GABA reuptake inhibitor. |
| CSN21594 | Dazopride | 70181-03-2 | Dazopride is an antiemetic agent which acts as a 5-HT3 receptor antagonist and 5-HT4 receptor agonist. |
| CSN10727 | Cyproheptadine Hydrochloride Sesquihydrate | 41354-29-4 | Cyproheptadine Hydrochloride Sesquihydrate is a serotonin antagonist and a histamine H1 blocker used as antipruritic, appetite stimulant, antiallergic, and for the post-gastrectomy dumping syndrome, etc. |
| CSN21571 | Clocapramine | 47739-98-0 | Clocapramine is D2 5-HT2A receptors antagonist. |
| CSN10658 | Citalopram Hydrobromide | 59729-32-7 | Citalopram Hydrobromide is a highly selective and potent 5-HT uptake inhibitor with no effect on noradrenalin or dopamine uptake. |
| CSN24509 | BRL 15572 HCl | 1173022-77-9 | BRL 15572 HCl is a selective 5-HT Receptor 1D antagonist with a pKi value of 7.9 |
| CSN20672 | Aripiprazole Lauroxil | 1259305-29-7 | Aripiprazole lauroxil is a long-acting injectable atypical antipsychotic. It is an N-acyloxymethyl prodrug of aripiprazole that is administered via intramuscular injection once every four to six weeks for the treatment of schizophrenia. |
| CSN21450 | Abaperidone | 183849-43-6 | Abaperidone is an antagonist of 5-HT2A receptor and dopamine D2 receptor with IC50s of 6.2 and 17 nM respectively. |
| CSN21566 | (Z)-Thiothixene | 3313-26-6 | (Z)-Thiothixene is serotonergic receptor antagonist. |
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