V-9302 HCl is a competitive and selective antagonist of transmembrane glutamine flux that selectively and potently targets the amino acid transporter ASCT2 with IC50 of 9.6 μM.
Defensamide is an activator of SPHK1, and significantly stimulates CAMP mRNA and protein production in KC.
D3-βArr is a positive allosteric TSH Receptor modulator.
Fargesin is a lignan from Magnolia fargesii, an oriental medicine used in the treatment of nasal congestion and sinusitis.
BQR695 is a PI4K specific inhibitor with IC50 value of 80nM.
MK-7246 is a potent and selective CRTH2 antagonist with Ki value of 2.5nM.
Gardiquimod trifluoroacetate is a specific TLR7 agonist.
WIN 18446 is an inhibitor of aldehyde dehydrogenase 1a2 (ALDH1a2) with IC50 of 0.3 μM.
MRTX1257 is a selective, covalent K-Ras G12C inhibitor with oral activity in animal models of cancer.
Spermidine, a precursor of spermine, is a polyamine derived from putrescine and could help stabilize some membranes and nucleic acid structures.
- Elagolix Sodium